TW264477B - - Google Patents

Info

Publication number
TW264477B
TW264477B TW082101890A TW82101890A TW264477B TW 264477 B TW264477 B TW 264477B TW 082101890 A TW082101890 A TW 082101890A TW 82101890 A TW82101890 A TW 82101890A TW 264477 B TW264477 B TW 264477B
Authority
TW
Taiwan
Prior art keywords
hydrogen
hydroxy
hydroxysulfonyloxy
methyl
compounds
Prior art date
Application number
TW082101890A
Other languages
English (en)
Chinese (zh)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of TW264477B publication Critical patent/TW264477B/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64—Cyclic peptides containing only normal peptide links
    • C07K7/66—Gramicidins S, C; Tyrocidins A, B, C; Related peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Virology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
TW082101890A 1992-03-19 1993-03-15 TW264477B (OSRAM)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US85411792A 1992-03-19 1992-03-19
US99239092A 1992-12-16 1992-12-16

Publications (1)

Publication Number Publication Date
TW264477B true TW264477B (OSRAM) 1995-12-01

Family

ID=27127211

Family Applications (1)

Application Number Title Priority Date Filing Date
TW082101890A TW264477B (OSRAM) 1992-03-19 1993-03-15

Country Status (25)

Country Link
EP (1) EP0561639B1 (OSRAM)
JP (3) JP3519754B2 (OSRAM)
KR (1) KR100256036B1 (OSRAM)
CN (1) CN1036715C (OSRAM)
AT (1) ATE217635T1 (OSRAM)
AU (2) AU3534193A (OSRAM)
BR (1) BR9301232A (OSRAM)
CA (1) CA2091663C (OSRAM)
CZ (1) CZ288974B6 (OSRAM)
DE (2) DE122008000006I2 (OSRAM)
DK (1) DK0561639T3 (OSRAM)
ES (1) ES2174843T3 (OSRAM)
FI (1) FI118768B (OSRAM)
HU (2) HU225783B1 (OSRAM)
IL (3) IL105048A (OSRAM)
LU (1) LU91406I2 (OSRAM)
MX (1) MX9301457A (OSRAM)
MY (1) MY136593A (OSRAM)
NL (1) NL300334I2 (OSRAM)
NO (1) NO930948L (OSRAM)
NZ (3) NZ512085A (OSRAM)
PT (1) PT561639E (OSRAM)
RU (1) RU2129562C1 (OSRAM)
TW (1) TW264477B (OSRAM)
YU (1) YU49108B (OSRAM)

Families Citing this family (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5430018A (en) * 1991-10-17 1995-07-04 Merck & Co., Inc. Cyclohexapeptide with basic nitrogen containing alkylamide groups
US6743777B1 (en) 1992-03-19 2004-06-01 Eli Lilly And Company Cyclic peptide antifungal agents and process for preparation thereof
CA2091663C (en) * 1992-03-19 2007-10-30 Frederick Joseph Burkhardt Cyclic peptide antifungal agents and process for preparation thereof
US5378804A (en) * 1993-03-16 1995-01-03 Merck & Co., Inc. Aza cyclohexapeptide compounds
US5948753A (en) * 1993-05-04 1999-09-07 Merck & Co., Inc. Cyclohexapeptidyl propanolamine compounds
EP0697879A4 (en) * 1993-05-04 1998-01-14 Merck & Co Inc AMINOALKYL ETHER DERIVATIVES OF CYCLOHEXAPEPTIDES
WO1995008341A1 (en) * 1993-09-22 1995-03-30 Merck & Co., Inc. Antifungal and anti-pneumocystis compounds, compositions containing such compounds, and methods of use
US5516757A (en) * 1994-09-16 1996-05-14 Merck & Co., Inc. Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use
EP0781141B1 (en) * 1994-09-16 2002-09-04 Merck & Co. Inc. Aza cyclohexapeptide compounds
US5514651A (en) * 1994-09-16 1996-05-07 Merck & Co., Inc. Aza cyclohexapeptide compounds
JP2897427B2 (ja) * 1994-10-07 1999-05-31 藤沢薬品工業株式会社 抗微生物活性を有する環状ヘキサペプチド化合物
US5516756A (en) * 1994-10-31 1996-05-14 Merck & Co., Inc. Aza cyclohexapeptide compounds
CA2211138A1 (en) * 1995-01-26 1996-08-01 Merck & Co., Inc. Novel antifungal cyclohexapeptides
US5646111A (en) * 1995-04-07 1997-07-08 Eli Lilly And Company Cyclic peptide antifungal Agents
US5629290A (en) * 1995-05-26 1997-05-13 Eli Lilly And Company Cyclic peptide antifungal agents
US5652213A (en) * 1995-05-26 1997-07-29 Eli Lilly And Company Cyclic peptide antifungal agents
US5786325A (en) * 1995-05-26 1998-07-28 Eli Lilly And Company Cyclic peptide antifungal agents and methods of making and using
US5618787A (en) * 1995-05-26 1997-04-08 Eli Lilly And Company Cyclic peptide antifungal agents
US5629289A (en) * 1995-07-25 1997-05-13 Eli Lilly And Company Cyclic peptide antifungal agents
AU1851797A (en) * 1996-02-01 1997-08-22 Eli Lilly And Company Cyclic peptide antifungal agents
US5693611A (en) * 1996-02-01 1997-12-02 Eli Lilly And Company Cyclic peptide antifungal agents
JPH09227422A (ja) * 1996-02-12 1997-09-02 Rolic Ag シクロペンチル誘導体
US5696084A (en) * 1996-08-16 1997-12-09 Abbott Laboratories Amino-lipopetide antifungal agents
AUPO381496A0 (en) * 1996-11-25 1996-12-19 Fujisawa Pharmaceutical Co., Ltd. New compound
FR2784993B1 (fr) * 1998-10-26 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme fongicides
UA72200C2 (uk) 1997-12-10 2005-02-15 Авентіс Фарма С.А. Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція
AU2003200556B2 (en) * 1997-12-10 2005-12-01 Novexel Echinocandin derivative and their preparation method
AUPP172898A0 (en) * 1998-02-09 1998-03-05 Fujisawa Pharmaceutical Co., Ltd. New compound
JP2002509444A (ja) * 1998-03-16 2002-03-26 藤沢薬品工業株式会社 Ｗｆ１４５７３またはその塩、それらの製法および用途
JP2002528388A (ja) 1998-08-20 2002-09-03 イーライ リリー アンド カンパニー 環改変された環状ペプチドアナログ
US6506726B1 (en) 1998-12-09 2003-01-14 Eli Lilly And Company Purification of Echinocandin cyclopeptide compounds
DE19907904A1 (de) 1999-02-24 2000-08-31 Clariant Gmbh Verfahren zur Herstellung von [1,1':4',1"]-Terphenylverbindungen
WO2000052037A1 (en) 1999-03-03 2000-09-08 Eli Lilly And Company Echinocandin/carbohydrate complexes
ATE338060T1 (de) 1999-03-03 2006-09-15 Lilly Co Eli Bildung und anionenaustausch von inneren kristallinen ammoniumsalzen des echinocandins b
DK1582204T3 (da) * 1999-03-03 2013-11-04 Lilly Co Eli Echinocandin-farmaceutiske formuleringer, der indeholder miceldannende overfladeaktive stoffer
CA2362482A1 (en) 1999-03-03 2000-09-08 Eli Lilly And Company Processes for making pharmaceutical oral ecb formulations and compositions
AU2001232319B2 (en) * 2000-02-18 2005-01-13 Meiji Seika Kaisha, Ltd. Phenoxyalkylamine derivates useful as opioid delta receptor ligands
FR2833596B1 (fr) * 2001-12-14 2005-02-18 Aventis Pharma Sa Procede de preparation de derives d'echinocandine
US6991800B2 (en) 2002-06-13 2006-01-31 Vicuron Pharmaceuticals Inc. Antifungal parenteral products
WO2004099170A2 (en) * 2003-04-30 2004-11-18 The Institutes For Pharmaceutical Discovery, Llc Phenyl substituted carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
KR101551207B1 (ko) * 2008-09-04 2015-09-08 롬엔드하스전자재료코리아유한회사 신규한 유기 발광 화합물 및 이를 발광재료로서 채용하고 있는 유기 발광 소자
CN102464704B (zh) * 2010-11-05 2013-12-11 上海医药工业研究院 一种化合物及其制备方法和用途
PL3677252T3 (pl) * 2012-03-19 2024-01-08 Cidara Therapeutics, Inc. Schematy dawkowania dla związków z klasy echinokandyn
ES2694561T3 (es) 2015-02-23 2018-12-21 Selectchemie Ag Composición de anidulafungina
JP6866583B2 (ja) * 2016-07-05 2021-04-28 Dic株式会社 液晶化合物
CN116903706B (zh) * 2023-06-13 2024-05-17 深圳市祥根生物有限公司 一种棘白菌素类药物及其制备方法和用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE886575A (fr) * 1979-12-13 1981-06-10 Lilly Co Eli Derives de noyaux peptidiques cycliques, leur preparation et leur utilisation comme agents antifongiques
BE886576A (fr) * 1979-12-13 1981-06-10 Lilly Co Eli Derives de noyaux peptidiques cycliques, leur preparation et leur utilisation comme agents antifongiques
CA2037957A1 (en) * 1990-03-12 1991-09-13 Merck & Co., Inc. N-acylated cyclohexapeptide compounds
GB2241956A (en) * 1990-03-16 1991-09-18 Merck & Co Inc N-acylated cyclohexapeptide compounds
US5330973A (en) * 1990-03-19 1994-07-19 Merck & Co., Inc. Lipopeptide derivatives
IL97347A0 (en) * 1990-03-19 1992-05-25 Merck & Co Inc Lipopeptide derivatives and antimicrobial compositions containing them
US5310726A (en) * 1990-03-19 1994-05-10 Merck & Co., Inc. Lipopeptide compounds
CA2091663C (en) * 1992-03-19 2007-10-30 Frederick Joseph Burkhardt Cyclic peptide antifungal agents and process for preparation thereof

Also Published As

Publication number Publication date
NO930948D0 (no) 1993-03-16
CA2091663A1 (en) 1993-09-20
AU689391B2 (en) 1998-03-26
DE122008000006I2 (de) 2011-07-21
JP3520071B2 (ja) 2004-04-19
NZ299314A (en) 2001-09-28
NZ512085A (en) 2003-08-29
BR9301232A (pt) 1993-09-21
JP2004115540A (ja) 2004-04-15
CZ288974B6 (cs) 2001-10-17
MY136593A (en) 2008-10-31
NZ247149A (en) 1996-10-28
CN1036715C (zh) 1997-12-17
HU9300785D0 (en) 1993-06-28
HU211562A9 (en) 1995-12-28
ES2174843T3 (es) 2002-11-16
NL300334I1 (nl) 2008-03-03
JP3519754B2 (ja) 2004-04-19
JP2002226500A (ja) 2002-08-14
IL122315A0 (en) 1998-04-05
FI931202L (fi) 1993-09-20
FI931202A0 (fi) 1993-03-18
FI118768B (fi) 2008-03-14
HU225783B1 (en) 2007-09-28
JPH0656892A (ja) 1994-03-01
DK0561639T3 (da) 2002-06-17
NL300334I2 (nl) 2008-05-01
DE69331922T2 (de) 2002-08-29
NO930948L (no) 1993-09-20
LU91406I2 (fr) 2008-03-10
RU2129562C1 (ru) 1999-04-27
IL105048A0 (en) 1993-07-08
CA2091663C (en) 2007-10-30
IL122315A (en) 2002-03-10
YU49108B (sh) 2004-03-12
HUT63637A (en) 1993-09-28
EP0561639A1 (en) 1993-09-22
IL105048A (en) 2001-06-14
KR930019694A (ko) 1993-10-18
EP0561639B1 (en) 2002-05-15
KR100256036B1 (ko) 2000-05-01
PT561639E (pt) 2002-10-31
ATE217635T1 (de) 2002-06-15
DE69331922D1 (de) 2002-06-20
DE122008000006I1 (de) 2008-04-17
AU6552996A (en) 1996-12-05
MX9301457A (es) 1994-02-28
YU18593A (sh) 1996-10-09
AU3534193A (en) 1993-09-23
CN1080926A (zh) 1994-01-19
CZ41693A3 (en) 1994-07-13

Similar Documents

Publication Publication Date Title
TW264477B (OSRAM)
SG49607A1 (en) 1-methylcarbapenem derivatives and process for preparation thereof
NZ332136A (en) Phenylalkylcarboxylic acid derivatives useful for treating hyperglycemia
ZA927606B (en) Antifungal agent.
MY116862A (en) New processes for preparing pesticidal intermediates
HUT60232A (en) Process for producing diiododiethylether derivatives
CY1385A (en) N-naphthoylglycine derivatives
GR3001955T3 (en) N-phenethylaminoalkyl-benzamide anti-arrhythmia agents
HUT71513A (en) 2-substituted-(3-chlorophenyl)-3,6-diazahexanoic acid derivatives for producing alkil-trazodone derivatives and process for producing them
EP0555479A4 (OSRAM)
GR3023827T3 (en) Indole-sulfonamides as antitumor agents.
IL103202A0 (en) Method for treating hypertension
TW275629B (OSRAM)
GR76446B (OSRAM)
EP0272849A3 (en) Use of 2-oxo-imidazolidine derivatives in the treatment of kidney diseases
HUT70219A (en) 1-phenylpyrrolidone derivatives, intermediates for producing them and producing them
LU88449I2 (fr) Fleroxacine et ses dérivés pharmaceutiquement acceptables.

Legal Events

Date Code Title Description
MK4A Expiration of patent term of an invention patent