TW200418482A - Method of treatment of transplant rejection - Google Patents

Method of treatment of transplant rejection Download PDF

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Publication number
TW200418482A
TW200418482A TW092132613A TW92132613A TW200418482A TW 200418482 A TW200418482 A TW 200418482A TW 092132613 A TW092132613 A TW 092132613A TW 92132613 A TW92132613 A TW 92132613A TW 200418482 A TW200418482 A TW 200418482A
Authority
TW
Taiwan
Prior art keywords
alkyl
methyl
amine
amino
group
Prior art date
Application number
TW092132613A
Other languages
English (en)
Chinese (zh)
Inventor
Paul Steven Changelian
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TW200418482A publication Critical patent/TW200418482A/zh

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Transplantation (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
TW092132613A 2002-11-26 2003-11-20 Method of treatment of transplant rejection TW200418482A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42978402P 2002-11-26 2002-11-26

Publications (1)

Publication Number Publication Date
TW200418482A true TW200418482A (en) 2004-10-01

Family

ID=32393587

Family Applications (1)

Application Number Title Priority Date Filing Date
TW092132613A TW200418482A (en) 2002-11-26 2003-11-20 Method of treatment of transplant rejection

Country Status (15)

Country Link
US (1) US7250420B2 (https=)
EP (1) EP1572213A1 (https=)
JP (1) JP2006509000A (https=)
KR (1) KR20050086784A (https=)
CN (1) CN1717236A (https=)
AU (1) AU2003276591A1 (https=)
BR (1) BR0316487A (https=)
CA (1) CA2507392A1 (https=)
MX (1) MXPA05005576A (https=)
MY (1) MY137250A (https=)
NZ (1) NZ539901A (https=)
PL (1) PL378246A1 (https=)
TW (1) TW200418482A (https=)
WO (1) WO2004047843A1 (https=)
ZA (1) ZA200503811B (https=)

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Also Published As

Publication number Publication date
US7250420B2 (en) 2007-07-31
JP2006509000A (ja) 2006-03-16
ZA200503811B (en) 2006-07-26
CN1717236A (zh) 2006-01-04
CA2507392A1 (en) 2004-06-10
MY137250A (en) 2009-01-30
WO2004047843A1 (en) 2004-06-10
AU2003276591A1 (en) 2004-06-18
MXPA05005576A (es) 2005-07-27
KR20050086784A (ko) 2005-08-30
BR0316487A (pt) 2005-10-11
US20040116449A1 (en) 2004-06-17
PL378246A1 (pl) 2006-03-20
NZ539901A (en) 2007-09-28
EP1572213A1 (en) 2005-09-14

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