TR199800624T1 - Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi. - Google Patents

Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi.

Info

Publication number
TR199800624T1
TR199800624T1 TR1998/00624T TR9800624T TR199800624T1 TR 199800624 T1 TR199800624 T1 TR 199800624T1 TR 1998/00624 T TR1998/00624 T TR 1998/00624T TR 9800624 T TR9800624 T TR 9800624T TR 199800624 T1 TR199800624 T1 TR 199800624T1
Authority
TR
Turkey
Prior art keywords
revleri
kullan
erythronolid
deosaminil
buynar
Prior art date
Application number
TR1998/00624T
Other languages
English (en)
Inventor
Bonnet Alain
Chappert Bernadette
Lagouardat Jacques
Original Assignee
Hoechst Marion Roussel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel filed Critical Hoechst Marion Roussel
Publication of TR199800624T1 publication Critical patent/TR199800624T1/tr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

R' nin 18'e kadar karbon atomu içerdigi bir karboksilik asit bakiyesi oldugu formül (I)'i havi bilesikler tarif edilmektedir. Formül (I)'i havi bilesikler antibiyotiklerin hazirlanmasinda kullanilabilir.
TR1998/00624T 1995-10-09 1996-10-08 Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi. TR199800624T1 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
TR199800624T1 true TR199800624T1 (tr) 1998-06-22

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1998/00624T TR199800624T1 (tr) 1995-10-09 1996-10-08 Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi.

Country Status (33)

Country Link
US (1) US6011142A (tr)
EP (1) EP0854879B1 (tr)
JP (1) JP4327248B2 (tr)
KR (1) KR100451063B1 (tr)
CN (1) CN1067401C (tr)
AP (1) AP888A (tr)
AR (1) AR004688A1 (tr)
AT (1) ATE212034T1 (tr)
AU (1) AU708351B2 (tr)
BG (1) BG63752B1 (tr)
BR (1) BR9610959A (tr)
CA (1) CA2231562C (tr)
CZ (1) CZ293430B6 (tr)
DE (1) DE69618607T2 (tr)
DK (1) DK0854879T3 (tr)
EA (1) EA000765B1 (tr)
EE (1) EE03878B1 (tr)
ES (1) ES2171722T3 (tr)
FR (1) FR2739620B1 (tr)
GE (1) GEP20032899B (tr)
HU (1) HUP9900136A3 (tr)
IL (1) IL123613A0 (tr)
MX (1) MX9802655A (tr)
NO (1) NO312592B1 (tr)
PL (1) PL183645B1 (tr)
PT (1) PT854879E (tr)
RO (1) RO118874B1 (tr)
SI (1) SI0854879T1 (tr)
SK (1) SK283619B6 (tr)
TR (1) TR199800624T1 (tr)
UA (1) UA52621C2 (tr)
WO (1) WO1997013774A2 (tr)
ZA (1) ZA966666B (tr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
MXPA01010524A (es) * 1999-04-16 2002-03-14 Kosan Biosciences Inc Agentes macrolidos anti-infecciosos.
US6399582B1 (en) 1999-04-16 2002-06-04 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
EP2772254A3 (en) 2003-03-10 2015-03-11 Optimer Pharmaceuticals, Inc. Novel Antibacterial Agents
JP5698979B2 (ja) * 2007-10-25 2015-04-08 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライド系抗菌剤の調製プロセス
CN105616437A (zh) * 2008-10-24 2016-06-01 森普拉制药公司 使用含三唑的大环内酯的生物防御
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
CN108310000A (zh) 2009-09-10 2018-07-24 森普拉制药公司 治疗疟疾、结核病和mac疾病的方法
EP3009442B1 (en) 2010-03-22 2019-06-19 Cempra Pharmaceuticals, Inc. Crystalline forms of a macrolide, and uses therefor
DK2571506T3 (en) 2010-05-20 2017-08-28 Cempra Pharmaceuticals Inc PROCEDURES FOR THE MANUFACTURE OF MACROLIDES AND KETOLIDES AND INTERMEDIATES
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
RU2658050C2 (ru) 2012-03-27 2018-06-19 Семпра Фармасьютикалз, Инк. Парентеральные составы для введения макролидных антибиотиков
JP6426696B2 (ja) 2013-03-14 2018-11-21 センプラ ファーマシューティカルズ,インコーポレイテッド 呼吸器疾患の治療のための方法および製剤
CA2907085A1 (en) 2013-03-15 2014-09-18 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
KR880009960A (ko) * 1987-02-24 1988-10-06 데이빗 로버츠 화학적 화합물
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
US5631355A (en) * 1992-04-22 1997-05-20 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide a derivatives
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
CA2154550A1 (en) * 1993-01-26 1994-08-04 Yoko Misawa 5-o-desosaminylerythronolide derivatives

Also Published As

Publication number Publication date
EP0854879B1 (fr) 2002-01-16
JP4327248B2 (ja) 2009-09-09
ES2171722T3 (es) 2002-09-16
SK43198A3 (en) 1998-11-04
AR004688A1 (es) 1999-03-10
JPH11513401A (ja) 1999-11-16
WO1997013774A2 (fr) 1997-04-17
ZA966666B (en) 1997-08-06
ATE212034T1 (de) 2002-02-15
GEP20032899B (en) 2003-02-25
NO981630D0 (no) 1998-04-08
CA2231562A1 (fr) 1997-04-17
NO981630L (no) 1998-04-08
BG63752B1 (bg) 2002-11-29
BR9610959A (pt) 1999-03-02
FR2739620A1 (fr) 1997-04-11
CA2231562C (fr) 2006-11-28
NO312592B1 (no) 2002-06-03
CN1199403A (zh) 1998-11-18
IL123613A0 (en) 1998-10-30
AU7220896A (en) 1997-04-30
DE69618607D1 (de) 2002-02-21
FR2739620B1 (fr) 1997-12-19
AP888A (en) 2000-11-10
EA000765B1 (ru) 2000-04-24
US6011142A (en) 2000-01-04
EE03878B1 (et) 2002-10-15
AU708351B2 (en) 1999-08-05
PL326001A1 (en) 1998-08-17
HUP9900136A1 (hu) 1999-05-28
SI0854879T1 (en) 2002-08-31
BG102350A (en) 1999-03-31
CZ293430B6 (cs) 2004-04-14
PT854879E (pt) 2002-07-31
EP0854879A2 (fr) 1998-07-29
CZ105598A3 (cs) 1998-07-15
KR19990064100A (ko) 1999-07-26
PL183645B1 (pl) 2002-06-28
CN1067401C (zh) 2001-06-20
KR100451063B1 (ko) 2004-12-17
WO1997013774A3 (fr) 1997-05-29
EA199800280A1 (ru) 1998-10-29
SK283619B6 (sk) 2003-10-07
HUP9900136A3 (en) 2000-04-28
UA52621C2 (uk) 2003-01-15
MX9802655A (es) 1998-11-30
DK0854879T3 (da) 2002-05-06
RO118874B1 (ro) 2003-12-30
EE9800109A (et) 1998-10-15
DE69618607T2 (de) 2002-08-14

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