TR199800624T1 - Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi. - Google Patents
Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi.Info
- Publication number
- TR199800624T1 TR199800624T1 TR1998/00624T TR9800624T TR199800624T1 TR 199800624 T1 TR199800624 T1 TR 199800624T1 TR 1998/00624 T TR1998/00624 T TR 1998/00624T TR 9800624 T TR9800624 T TR 9800624T TR 199800624 T1 TR199800624 T1 TR 199800624T1
- Authority
- TR
- Turkey
- Prior art keywords
- revleri
- kullan
- erythronolid
- deosaminil
- buynar
- Prior art date
Links
- YVTFLQUPRIIRFE-QUMKBVJLSA-N erythronolide A Chemical compound CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O YVTFLQUPRIIRFE-QUMKBVJLSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 229940088710 antibiotic agent Drugs 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001732 carboxylic acid derivatives Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
R' nin 18'e kadar karbon atomu içerdigi bir karboksilik asit bakiyesi oldugu formül (I)'i havi bilesikler tarif edilmektedir. Formül (I)'i havi bilesikler antibiyotiklerin hazirlanmasinda kullanilabilir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9511861A FR2739620B1 (fr) | 1995-10-09 | 1995-10-09 | Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs |
Publications (1)
Publication Number | Publication Date |
---|---|
TR199800624T1 true TR199800624T1 (tr) | 1998-06-22 |
Family
ID=9483377
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR1998/00624T TR199800624T1 (tr) | 1995-10-09 | 1996-10-08 | Yeni 5-0- deosaminil 6-0-metil eritronolid a türevleri, bunlarin kullanimi. |
Country Status (33)
Country | Link |
---|---|
US (1) | US6011142A (tr) |
EP (1) | EP0854879B1 (tr) |
JP (1) | JP4327248B2 (tr) |
KR (1) | KR100451063B1 (tr) |
CN (1) | CN1067401C (tr) |
AP (1) | AP888A (tr) |
AR (1) | AR004688A1 (tr) |
AT (1) | ATE212034T1 (tr) |
AU (1) | AU708351B2 (tr) |
BG (1) | BG63752B1 (tr) |
BR (1) | BR9610959A (tr) |
CA (1) | CA2231562C (tr) |
CZ (1) | CZ293430B6 (tr) |
DE (1) | DE69618607T2 (tr) |
DK (1) | DK0854879T3 (tr) |
EA (1) | EA000765B1 (tr) |
EE (1) | EE03878B1 (tr) |
ES (1) | ES2171722T3 (tr) |
FR (1) | FR2739620B1 (tr) |
GE (1) | GEP20032899B (tr) |
HU (1) | HUP9900136A3 (tr) |
IL (1) | IL123613A0 (tr) |
MX (1) | MX9802655A (tr) |
NO (1) | NO312592B1 (tr) |
PL (1) | PL183645B1 (tr) |
PT (1) | PT854879E (tr) |
RO (1) | RO118874B1 (tr) |
SI (1) | SI0854879T1 (tr) |
SK (1) | SK283619B6 (tr) |
TR (1) | TR199800624T1 (tr) |
UA (1) | UA52621C2 (tr) |
WO (1) | WO1997013774A2 (tr) |
ZA (1) | ZA966666B (tr) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2777282B1 (fr) * | 1998-04-08 | 2001-04-20 | Hoechst Marion Roussel Inc | Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments |
MXPA01010524A (es) * | 1999-04-16 | 2002-03-14 | Kosan Biosciences Inc | Agentes macrolidos anti-infecciosos. |
US6399582B1 (en) | 1999-04-16 | 2002-06-04 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
US6590083B1 (en) | 1999-04-16 | 2003-07-08 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
GB0031312D0 (en) * | 2000-12-21 | 2001-02-07 | Glaxo Group Ltd | Macrolides |
EP2772254A3 (en) | 2003-03-10 | 2015-03-11 | Optimer Pharmaceuticals, Inc. | Novel Antibacterial Agents |
JP5698979B2 (ja) * | 2007-10-25 | 2015-04-08 | センプラ ファーマシューティカルズ,インコーポレイテッド | マクロライド系抗菌剤の調製プロセス |
CN105616437A (zh) * | 2008-10-24 | 2016-06-01 | 森普拉制药公司 | 使用含三唑的大环内酯的生物防御 |
US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
CN108310000A (zh) | 2009-09-10 | 2018-07-24 | 森普拉制药公司 | 治疗疟疾、结核病和mac疾病的方法 |
EP3009442B1 (en) | 2010-03-22 | 2019-06-19 | Cempra Pharmaceuticals, Inc. | Crystalline forms of a macrolide, and uses therefor |
DK2571506T3 (en) | 2010-05-20 | 2017-08-28 | Cempra Pharmaceuticals Inc | PROCEDURES FOR THE MANUFACTURE OF MACROLIDES AND KETOLIDES AND INTERMEDIATES |
US9815863B2 (en) | 2010-09-10 | 2017-11-14 | Cempra Pharmaceuticals, Inc. | Hydrogen bond forming fluoro ketolides for treating diseases |
RU2658050C2 (ru) | 2012-03-27 | 2018-06-19 | Семпра Фармасьютикалз, Инк. | Парентеральные составы для введения макролидных антибиотиков |
JP6426696B2 (ja) | 2013-03-14 | 2018-11-21 | センプラ ファーマシューティカルズ,インコーポレイテッド | 呼吸器疾患の治療のための方法および製剤 |
CA2907085A1 (en) | 2013-03-15 | 2014-09-18 | Cempra Pharmaceuticals, Inc. | Convergent processes for preparing macrolide antibacterial agents |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3923784A (en) * | 1973-09-10 | 1975-12-02 | Hoffmann La Roche | Erythromycin a derivatives |
US4518590A (en) * | 1984-04-13 | 1985-05-21 | Pfizer Inc. | 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method |
US4742049A (en) * | 1986-06-04 | 1988-05-03 | Abbott Laboratories | Semisynthetic erythromycin antibiotics |
KR880009960A (ko) * | 1987-02-24 | 1988-10-06 | 데이빗 로버츠 | 화학적 화합물 |
US5523399A (en) * | 1991-12-27 | 1996-06-04 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
US5631355A (en) * | 1992-04-22 | 1997-05-20 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide a derivatives |
FR2692579B1 (fr) * | 1992-06-19 | 1995-06-02 | Roussel Uclaf | Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments. |
CA2154550A1 (en) * | 1993-01-26 | 1994-08-04 | Yoko Misawa | 5-o-desosaminylerythronolide derivatives |
-
1995
- 1995-10-09 FR FR9511861A patent/FR2739620B1/fr not_active Expired - Fee Related
-
1996
- 1996-08-06 ZA ZA9606666A patent/ZA966666B/xx unknown
- 1996-08-10 UA UA98041836A patent/UA52621C2/uk unknown
- 1996-10-07 AR ARP960104634A patent/AR004688A1/es not_active Application Discontinuation
- 1996-10-08 PL PL96326001A patent/PL183645B1/pl not_active IP Right Cessation
- 1996-10-08 ES ES96933501T patent/ES2171722T3/es not_active Expired - Lifetime
- 1996-10-08 RO RO98-00826A patent/RO118874B1/ro unknown
- 1996-10-08 EP EP96933501A patent/EP0854879B1/fr not_active Expired - Lifetime
- 1996-10-08 SK SK431-98A patent/SK283619B6/sk unknown
- 1996-10-08 PT PT96933501T patent/PT854879E/pt unknown
- 1996-10-08 US US09/051,378 patent/US6011142A/en not_active Ceased
- 1996-10-08 WO PCT/FR1996/001567 patent/WO1997013774A2/fr not_active Application Discontinuation
- 1996-10-08 HU HU9900136A patent/HUP9900136A3/hu unknown
- 1996-10-08 GE GEAP19964227A patent/GEP20032899B/en unknown
- 1996-10-08 IL IL12361396A patent/IL123613A0/xx not_active IP Right Cessation
- 1996-10-08 AU AU72208/96A patent/AU708351B2/en not_active Expired
- 1996-10-08 KR KR10-1998-0702581A patent/KR100451063B1/ko not_active IP Right Cessation
- 1996-10-08 BR BR9610959A patent/BR9610959A/pt not_active Application Discontinuation
- 1996-10-08 SI SI9630452T patent/SI0854879T1/xx unknown
- 1996-10-08 EA EA199800280A patent/EA000765B1/ru not_active IP Right Cessation
- 1996-10-08 CN CN96197514A patent/CN1067401C/zh not_active Expired - Lifetime
- 1996-10-08 DK DK96933501T patent/DK0854879T3/da active
- 1996-10-08 CA CA002231562A patent/CA2231562C/fr not_active Expired - Lifetime
- 1996-10-08 AT AT96933501T patent/ATE212034T1/de active
- 1996-10-08 JP JP51476697A patent/JP4327248B2/ja not_active Expired - Lifetime
- 1996-10-08 EE EE9800109A patent/EE03878B1/xx not_active IP Right Cessation
- 1996-10-08 TR TR1998/00624T patent/TR199800624T1/tr unknown
- 1996-10-08 AP APAP/P/1998/001216A patent/AP888A/en active
- 1996-10-08 CZ CZ19981055A patent/CZ293430B6/cs not_active IP Right Cessation
- 1996-10-08 DE DE69618607T patent/DE69618607T2/de not_active Expired - Lifetime
-
1998
- 1998-03-25 BG BG102350A patent/BG63752B1/bg unknown
- 1998-04-03 MX MX9802655A patent/MX9802655A/es unknown
- 1998-04-08 NO NO19981630A patent/NO312592B1/no not_active IP Right Cessation
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