MX9802655A - Nuevos derivados de la 5-0-desosaminil-6-metil-eritronolida a, su procedimiento de preparacion y su aplicacion para la preparacion de productos biologicamente activos. - Google Patents

Nuevos derivados de la 5-0-desosaminil-6-metil-eritronolida a, su procedimiento de preparacion y su aplicacion para la preparacion de productos biologicamente activos.

Info

Publication number
MX9802655A
MX9802655A MX9802655A MX9802655A MX9802655A MX 9802655 A MX9802655 A MX 9802655A MX 9802655 A MX9802655 A MX 9802655A MX 9802655 A MX9802655 A MX 9802655A MX 9802655 A MX9802655 A MX 9802655A
Authority
MX
Mexico
Prior art keywords
deosaminyl
derivatives
novel
preparation
biologically active
Prior art date
Application number
MX9802655A
Other languages
English (en)
Inventor
Alain Bonnet
Bernadette Chappert
Jacques Lagouardat
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of MX9802655A publication Critical patent/MX9802655A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

La invencion tiene por objetivo los compuestos de la formula (I), en los cuales R representan el residuo de un ácido carboxílico que contiene hasta 18átomos de carbono. Los productos de la formula (I) pueden ser utilizados para preparar productos antibioticos.
MX9802655A 1995-10-09 1998-04-03 Nuevos derivados de la 5-0-desosaminil-6-metil-eritronolida a, su procedimiento de preparacion y su aplicacion para la preparacion de productos biologicamente activos. MX9802655A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
MX9802655A true MX9802655A (es) 1998-11-30

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9802655A MX9802655A (es) 1995-10-09 1998-04-03 Nuevos derivados de la 5-0-desosaminil-6-metil-eritronolida a, su procedimiento de preparacion y su aplicacion para la preparacion de productos biologicamente activos.

Country Status (33)

Country Link
US (1) US6011142A (es)
EP (1) EP0854879B1 (es)
JP (1) JP4327248B2 (es)
KR (1) KR100451063B1 (es)
CN (1) CN1067401C (es)
AP (1) AP888A (es)
AR (1) AR004688A1 (es)
AT (1) ATE212034T1 (es)
AU (1) AU708351B2 (es)
BG (1) BG63752B1 (es)
BR (1) BR9610959A (es)
CA (1) CA2231562C (es)
CZ (1) CZ293430B6 (es)
DE (1) DE69618607T2 (es)
DK (1) DK0854879T3 (es)
EA (1) EA000765B1 (es)
EE (1) EE03878B1 (es)
ES (1) ES2171722T3 (es)
FR (1) FR2739620B1 (es)
GE (1) GEP20032899B (es)
HU (1) HUP9900136A3 (es)
IL (1) IL123613A0 (es)
MX (1) MX9802655A (es)
NO (1) NO312592B1 (es)
PL (1) PL183645B1 (es)
PT (1) PT854879E (es)
RO (1) RO118874B1 (es)
SI (1) SI0854879T1 (es)
SK (1) SK283619B6 (es)
TR (1) TR199800624T1 (es)
UA (1) UA52621C2 (es)
WO (1) WO1997013774A2 (es)
ZA (1) ZA966666B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
MXPA01010521A (es) 1999-04-16 2003-08-19 Johnson & Johnson Antibacteriales de cetolidos.
AU775637B2 (en) * 1999-04-16 2004-08-12 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
WO2004080391A2 (en) 2003-03-10 2004-09-23 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
US9453042B2 (en) 2007-10-25 2016-09-27 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2010048600A1 (en) * 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Methods for treating resistant diseases using triazole containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
WO2011032052A1 (en) 2009-09-10 2011-03-17 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and mac diseases
DK2550286T3 (en) 2010-03-22 2016-02-29 Cempra Pharmaceuticals Inc CRYSTALLINE FORMS OF A MACROLID AND APPLICATIONS THEREOF
EP2571506B1 (en) 2010-05-20 2017-05-10 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
WO2012034058A1 (en) 2010-09-10 2012-03-15 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
RU2658050C2 (ru) 2012-03-27 2018-06-19 Семпра Фармасьютикалз, Инк. Парентеральные составы для введения макролидных антибиотиков
AU2014239959A1 (en) 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
US9751908B2 (en) 2013-03-15 2017-09-05 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
DK90788A (da) * 1987-02-24 1988-08-25 Beecham Group Plc Erythromycinderivater
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
ATE145212T1 (de) * 1992-04-22 1996-11-15 Taisho Pharmaceutical Co Ltd 5-0-desosaminylerythronolide a derivate
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
AU671899B2 (en) * 1993-01-26 1996-09-12 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivative

Also Published As

Publication number Publication date
HUP9900136A1 (hu) 1999-05-28
SK43198A3 (en) 1998-11-04
PT854879E (pt) 2002-07-31
AU708351B2 (en) 1999-08-05
SK283619B6 (sk) 2003-10-07
DE69618607T2 (de) 2002-08-14
IL123613A0 (en) 1998-10-30
EE03878B1 (et) 2002-10-15
AR004688A1 (es) 1999-03-10
EA199800280A1 (ru) 1998-10-29
ATE212034T1 (de) 2002-02-15
CZ105598A3 (cs) 1998-07-15
NO981630L (no) 1998-04-08
EE9800109A (et) 1998-10-15
WO1997013774A2 (fr) 1997-04-17
PL326001A1 (en) 1998-08-17
ZA966666B (en) 1997-08-06
AU7220896A (en) 1997-04-30
CA2231562A1 (fr) 1997-04-17
DK0854879T3 (da) 2002-05-06
NO312592B1 (no) 2002-06-03
EP0854879A2 (fr) 1998-07-29
PL183645B1 (pl) 2002-06-28
CZ293430B6 (cs) 2004-04-14
JPH11513401A (ja) 1999-11-16
NO981630D0 (no) 1998-04-08
ES2171722T3 (es) 2002-09-16
AP888A (en) 2000-11-10
FR2739620A1 (fr) 1997-04-11
FR2739620B1 (fr) 1997-12-19
BR9610959A (pt) 1999-03-02
SI0854879T1 (en) 2002-08-31
EP0854879B1 (fr) 2002-01-16
EA000765B1 (ru) 2000-04-24
WO1997013774A3 (fr) 1997-05-29
BG102350A (en) 1999-03-31
JP4327248B2 (ja) 2009-09-09
RO118874B1 (ro) 2003-12-30
GEP20032899B (en) 2003-02-25
TR199800624T1 (xx) 1998-06-22
KR19990064100A (ko) 1999-07-26
KR100451063B1 (ko) 2004-12-17
CN1067401C (zh) 2001-06-20
DE69618607D1 (de) 2002-02-21
CA2231562C (fr) 2006-11-28
HUP9900136A3 (en) 2000-04-28
UA52621C2 (uk) 2003-01-15
CN1199403A (zh) 1998-11-18
BG63752B1 (bg) 2002-11-29
US6011142A (en) 2000-01-04

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