CZ105598A3 - Deriváty 5-O-desoaminyl 6-O-methyl erytronolidu A, způsob jejich přípravy a použití při přípravě biologicky aktivních produktů - Google Patents

Deriváty 5-O-desoaminyl 6-O-methyl erytronolidu A, způsob jejich přípravy a použití při přípravě biologicky aktivních produktů

Info

Publication number
CZ105598A3
CZ105598A3 CZ981055A CZ105598A CZ105598A3 CZ 105598 A3 CZ105598 A3 CZ 105598A3 CZ 981055 A CZ981055 A CZ 981055A CZ 105598 A CZ105598 A CZ 105598A CZ 105598 A3 CZ105598 A3 CZ 105598A3
Authority
CZ
Czechia
Prior art keywords
desoaminyl
derivatives
preparation
biologically active
active products
Prior art date
Application number
CZ981055A
Other languages
English (en)
Other versions
CZ293430B6 (cs
Inventor
Alain Bonnet
Bernadette Chappert
Jaques Lagouardat
Original Assignee
Hoechst Marion Roussel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel filed Critical Hoechst Marion Roussel
Publication of CZ105598A3 publication Critical patent/CZ105598A3/cs
Publication of CZ293430B6 publication Critical patent/CZ293430B6/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
CZ19981055A 1995-10-09 1996-10-08 Sloučeniny 5-O-desoaminyl 6-O-methylerytronolidu A a způsob jejich přípravy CZ293430B6 (cs)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (2)

Publication Number Publication Date
CZ105598A3 true CZ105598A3 (cs) 1998-07-15
CZ293430B6 CZ293430B6 (cs) 2004-04-14

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ19981055A CZ293430B6 (cs) 1995-10-09 1996-10-08 Sloučeniny 5-O-desoaminyl 6-O-methylerytronolidu A a způsob jejich přípravy

Country Status (33)

Country Link
US (1) US6011142A (cs)
EP (1) EP0854879B1 (cs)
JP (1) JP4327248B2 (cs)
KR (1) KR100451063B1 (cs)
CN (1) CN1067401C (cs)
AP (1) AP888A (cs)
AR (1) AR004688A1 (cs)
AT (1) ATE212034T1 (cs)
AU (1) AU708351B2 (cs)
BG (1) BG63752B1 (cs)
BR (1) BR9610959A (cs)
CA (1) CA2231562C (cs)
CZ (1) CZ293430B6 (cs)
DE (1) DE69618607T2 (cs)
DK (1) DK0854879T3 (cs)
EA (1) EA000765B1 (cs)
EE (1) EE03878B1 (cs)
ES (1) ES2171722T3 (cs)
FR (1) FR2739620B1 (cs)
GE (1) GEP20032899B (cs)
HU (1) HUP9900136A3 (cs)
IL (1) IL123613A0 (cs)
MX (1) MX9802655A (cs)
NO (1) NO312592B1 (cs)
PL (1) PL183645B1 (cs)
PT (1) PT854879E (cs)
RO (1) RO118874B1 (cs)
SI (1) SI0854879T1 (cs)
SK (1) SK283619B6 (cs)
TR (1) TR199800624T1 (cs)
UA (1) UA52621C2 (cs)
WO (1) WO1997013774A2 (cs)
ZA (1) ZA966666B (cs)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
JP2002542197A (ja) 1999-04-16 2002-12-10 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド ケトライド抗菌剤
DE60030847T2 (de) * 1999-04-16 2007-04-19 Kosan Biosciences, Inc., Hayward Antiinfektiöse makrolidderivate
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
ES2552682T3 (es) 2003-03-10 2015-12-01 Merck Sharp & Dohme Corp. Agentes antibacterianos novedosos
EP2214484A4 (en) 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
EP2358379B1 (en) * 2008-10-24 2015-12-16 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
US9480679B2 (en) 2009-09-10 2016-11-01 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and MAC diseases
DK2550286T3 (en) 2010-03-22 2016-02-29 Cempra Pharmaceuticals Inc CRYSTALLINE FORMS OF A MACROLID AND APPLICATIONS THEREOF
EP2571506B1 (en) 2010-05-20 2017-05-10 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
EP2613630A4 (en) 2010-09-10 2014-01-15 Cempra Pharmaceuticals Inc FLUOROCETOLIDES FORMING HYDROGEN LINKS TO TREAT DISEASES
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
JP6426696B2 (ja) 2013-03-14 2018-11-21 センプラ ファーマシューティカルズ,インコーポレイテッド 呼吸器疾患の治療のための方法および製剤
EP2968384A4 (en) 2013-03-15 2017-02-15 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
PT86800B (pt) * 1987-02-24 1992-05-29 Beecham Group Plc Processo para a preparacao de derivados de eritromicina
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
DK0638584T3 (da) * 1992-04-22 1996-04-15 Taisho Pharmaceutical Co Ltd 5-O-desosaminyl-erythronolid-A-derivat
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
KR960700258A (ko) * 1993-01-26 1996-01-19 우에하라 아키라 5-0-데소사미닐에리쓰로노라이드 유도체

Also Published As

Publication number Publication date
UA52621C2 (uk) 2003-01-15
SI0854879T1 (en) 2002-08-31
NO981630D0 (no) 1998-04-08
EP0854879B1 (fr) 2002-01-16
CA2231562C (fr) 2006-11-28
CZ293430B6 (cs) 2004-04-14
EE9800109A (et) 1998-10-15
KR19990064100A (ko) 1999-07-26
DE69618607D1 (de) 2002-02-21
DE69618607T2 (de) 2002-08-14
MX9802655A (es) 1998-11-30
SK283619B6 (sk) 2003-10-07
TR199800624T1 (xx) 1998-06-22
JP4327248B2 (ja) 2009-09-09
AU708351B2 (en) 1999-08-05
JPH11513401A (ja) 1999-11-16
PT854879E (pt) 2002-07-31
NO312592B1 (no) 2002-06-03
US6011142A (en) 2000-01-04
EA000765B1 (ru) 2000-04-24
ATE212034T1 (de) 2002-02-15
EA199800280A1 (ru) 1998-10-29
HUP9900136A3 (en) 2000-04-28
SK43198A3 (en) 1998-11-04
AU7220896A (en) 1997-04-30
RO118874B1 (ro) 2003-12-30
NO981630L (no) 1998-04-08
PL326001A1 (en) 1998-08-17
WO1997013774A2 (fr) 1997-04-17
EE03878B1 (et) 2002-10-15
AR004688A1 (es) 1999-03-10
GEP20032899B (en) 2003-02-25
PL183645B1 (pl) 2002-06-28
EP0854879A2 (fr) 1998-07-29
AP888A (en) 2000-11-10
HUP9900136A1 (hu) 1999-05-28
BG102350A (en) 1999-03-31
CN1199403A (zh) 1998-11-18
ZA966666B (en) 1997-08-06
BR9610959A (pt) 1999-03-02
CA2231562A1 (fr) 1997-04-17
WO1997013774A3 (fr) 1997-05-29
CN1067401C (zh) 2001-06-20
IL123613A0 (en) 1998-10-30
ES2171722T3 (es) 2002-09-16
FR2739620A1 (fr) 1997-04-11
DK0854879T3 (da) 2002-05-06
KR100451063B1 (ko) 2004-12-17
FR2739620B1 (fr) 1997-12-19
BG63752B1 (bg) 2002-11-29

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Legal Events

Date Code Title Description
PD00 Pending as of 2000-06-30 in czech republic
MM4A Patent lapsed due to non-payment of fee

Effective date: 20051008