DK0854879T3 - Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer - Google Patents

Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer

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Publication number
DK0854879T3
DK0854879T3 DK96933501T DK96933501T DK0854879T3 DK 0854879 T3 DK0854879 T3 DK 0854879T3 DK 96933501 T DK96933501 T DK 96933501T DK 96933501 T DK96933501 T DK 96933501T DK 0854879 T3 DK0854879 T3 DK 0854879T3
Authority
DK
Denmark
Prior art keywords
preparation
desosamiyl
erythronolide
methyl
biologically active
Prior art date
Application number
DK96933501T
Other languages
Danish (da)
English (en)
Inventor
Alain Bonnet
Bernadette Chappert
Jacques Lagouardat
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of DK0854879T3 publication Critical patent/DK0854879T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK96933501T 1995-10-09 1996-10-08 Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer DK0854879T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001567 WO1997013774A2 (fr) 1995-10-09 1996-10-08 Nouveaux derives de la 5-o-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
DK0854879T3 true DK0854879T3 (da) 2002-05-06

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96933501T DK0854879T3 (da) 1995-10-09 1996-10-08 Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer

Country Status (33)

Country Link
US (1) US6011142A (tr)
EP (1) EP0854879B1 (tr)
JP (1) JP4327248B2 (tr)
KR (1) KR100451063B1 (tr)
CN (1) CN1067401C (tr)
AP (1) AP888A (tr)
AR (1) AR004688A1 (tr)
AT (1) ATE212034T1 (tr)
AU (1) AU708351B2 (tr)
BG (1) BG63752B1 (tr)
BR (1) BR9610959A (tr)
CA (1) CA2231562C (tr)
CZ (1) CZ293430B6 (tr)
DE (1) DE69618607T2 (tr)
DK (1) DK0854879T3 (tr)
EA (1) EA000765B1 (tr)
EE (1) EE03878B1 (tr)
ES (1) ES2171722T3 (tr)
FR (1) FR2739620B1 (tr)
GE (1) GEP20032899B (tr)
HU (1) HUP9900136A3 (tr)
IL (1) IL123613A0 (tr)
MX (1) MX9802655A (tr)
NO (1) NO312592B1 (tr)
PL (1) PL183645B1 (tr)
PT (1) PT854879E (tr)
RO (1) RO118874B1 (tr)
SI (1) SI0854879T1 (tr)
SK (1) SK283619B6 (tr)
TR (1) TR199800624T1 (tr)
UA (1) UA52621C2 (tr)
WO (1) WO1997013774A2 (tr)
ZA (1) ZA966666B (tr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
ES2272273T3 (es) * 1999-04-16 2007-05-01 Kosan Biosciences, Inc. Agentes antiinfecciosos macrolidos.
AU4354900A (en) 1999-04-16 2000-11-02 Kosan Biosciences, Inc. Ketolide antibacterials
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
CA2529817C (en) 2003-03-10 2013-02-12 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
WO2010048599A1 (en) 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Methods for treating gastrointestinal diseases
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
JP5914335B2 (ja) 2009-09-10 2016-05-11 センプラ ファーマシューティカルズ，インコーポレイテッド マラリア、結核、及びｍａｃ病の治療方法
NZ602544A (en) 2010-03-22 2014-11-28 Cempra Pharmaceuticals Inc Crystalline forms of a macrolide, and uses therefor
US9051346B2 (en) 2010-05-20 2015-06-09 Cempra Pharmaceuticals, Inc. Process for preparing triazole-containing ketolide antibiotics
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
SG11201405895UA (en) 2012-03-27 2014-10-30 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
US9861616B2 (en) 2013-03-14 2018-01-09 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
JP6675973B2 (ja) 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ，インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
DK90788A (da) * 1987-02-24 1988-08-25 Beecham Group Plc Erythromycinderivater
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
WO1993021199A1 (en) * 1992-04-22 1993-10-28 Taisho Pharmaceutical Co., Ltd. 5-o-desosaminylerythronolide a derivative
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
CA2154550A1 (en) * 1993-01-26 1994-08-04 Yoko Misawa 5-o-desosaminylerythronolide derivatives

Also Published As

Publication number Publication date
DE69618607T2 (de) 2002-08-14
FR2739620B1 (fr) 1997-12-19
PT854879E (pt) 2002-07-31
CN1199403A (zh) 1998-11-18
AU708351B2 (en) 1999-08-05
EA000765B1 (ru) 2000-04-24
JP4327248B2 (ja) 2009-09-09
DE69618607D1 (de) 2002-02-21
SK283619B6 (sk) 2003-10-07
HUP9900136A1 (hu) 1999-05-28
CA2231562C (fr) 2006-11-28
CZ293430B6 (cs) 2004-04-14
NO312592B1 (no) 2002-06-03
EE9800109A (et) 1998-10-15
WO1997013774A2 (fr) 1997-04-17
UA52621C2 (uk) 2003-01-15
HUP9900136A3 (en) 2000-04-28
SK43198A3 (en) 1998-11-04
ES2171722T3 (es) 2002-09-16
AU7220896A (en) 1997-04-30
BG63752B1 (bg) 2002-11-29
PL183645B1 (pl) 2002-06-28
BG102350A (en) 1999-03-31
CZ105598A3 (cs) 1998-07-15
CA2231562A1 (fr) 1997-04-17
AP888A (en) 2000-11-10
FR2739620A1 (fr) 1997-04-11
ATE212034T1 (de) 2002-02-15
ZA966666B (en) 1997-08-06
TR199800624T1 (tr) 1998-06-22
EA199800280A1 (ru) 1998-10-29
PL326001A1 (en) 1998-08-17
US6011142A (en) 2000-01-04
EE03878B1 (et) 2002-10-15
GEP20032899B (en) 2003-02-25
KR19990064100A (ko) 1999-07-26
NO981630L (no) 1998-04-08
WO1997013774A3 (fr) 1997-05-29
JPH11513401A (ja) 1999-11-16
BR9610959A (pt) 1999-03-02
EP0854879A2 (fr) 1998-07-29
IL123613A0 (en) 1998-10-30
RO118874B1 (ro) 2003-12-30
CN1067401C (zh) 2001-06-20
MX9802655A (es) 1998-11-30
EP0854879B1 (fr) 2002-01-16
KR100451063B1 (ko) 2004-12-17
AR004688A1 (es) 1999-03-10
SI0854879T1 (en) 2002-08-31
NO981630D0 (no) 1998-04-08

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