SI0854879T1 - Novel 5-o-deosaminyl 6-o-methyl erythronolide a derivatives, preparation method therefor and use thereof for preparing biologically active materials - Google Patents

Novel 5-o-deosaminyl 6-o-methyl erythronolide a derivatives, preparation method therefor and use thereof for preparing biologically active materials

Info

Publication number
SI0854879T1
SI0854879T1 SI9630452T SI9630452T SI0854879T1 SI 0854879 T1 SI0854879 T1 SI 0854879T1 SI 9630452 T SI9630452 T SI 9630452T SI 9630452 T SI9630452 T SI 9630452T SI 0854879 T1 SI0854879 T1 SI 0854879T1
Authority
SI
Slovenia
Prior art keywords
deosaminyl
derivatives
novel
preparation
biologically active
Prior art date
Application number
SI9630452T
Other languages
English (en)
Slovenian (sl)
Inventor
Alain Bonnet
Bernadette Chappert
Jacques Lagouardat
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of SI0854879T1 publication Critical patent/SI0854879T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
SI9630452T 1995-10-09 1996-10-08 Novel 5-o-deosaminyl 6-o-methyl erythronolide a derivatives, preparation method therefor and use thereof for preparing biologically active materials SI0854879T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
EP96933501A EP0854879B1 (fr) 1995-10-09 1996-10-08 Nouveaux derives de la 5-o-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001567 WO1997013774A2 (fr) 1995-10-09 1996-10-08 Nouveaux derives de la 5-o-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
SI0854879T1 true SI0854879T1 (en) 2002-08-31

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9630452T SI0854879T1 (en) 1995-10-09 1996-10-08 Novel 5-o-deosaminyl 6-o-methyl erythronolide a derivatives, preparation method therefor and use thereof for preparing biologically active materials

Country Status (33)

Country Link
US (1) US6011142A (tr)
EP (1) EP0854879B1 (tr)
JP (1) JP4327248B2 (tr)
KR (1) KR100451063B1 (tr)
CN (1) CN1067401C (tr)
AP (1) AP888A (tr)
AR (1) AR004688A1 (tr)
AT (1) ATE212034T1 (tr)
AU (1) AU708351B2 (tr)
BG (1) BG63752B1 (tr)
BR (1) BR9610959A (tr)
CA (1) CA2231562C (tr)
CZ (1) CZ293430B6 (tr)
DE (1) DE69618607T2 (tr)
DK (1) DK0854879T3 (tr)
EA (1) EA000765B1 (tr)
EE (1) EE03878B1 (tr)
ES (1) ES2171722T3 (tr)
FR (1) FR2739620B1 (tr)
GE (1) GEP20032899B (tr)
HU (1) HUP9900136A3 (tr)
IL (1) IL123613A0 (tr)
MX (1) MX9802655A (tr)
NO (1) NO312592B1 (tr)
PL (1) PL183645B1 (tr)
PT (1) PT854879E (tr)
RO (1) RO118874B1 (tr)
SI (1) SI0854879T1 (tr)
SK (1) SK283619B6 (tr)
TR (1) TR199800624T1 (tr)
UA (1) UA52621C2 (tr)
WO (1) WO1997013774A2 (tr)
ZA (1) ZA966666B (tr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
ES2272273T3 (es) * 1999-04-16 2007-05-01 Kosan Biosciences, Inc. Agentes antiinfecciosos macrolidos.
AU4354900A (en) 1999-04-16 2000-11-02 Kosan Biosciences, Inc. Ketolide antibacterials
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
CA2529817C (en) 2003-03-10 2013-02-12 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
WO2010048599A1 (en) 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Methods for treating gastrointestinal diseases
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
JP5914335B2 (ja) 2009-09-10 2016-05-11 センプラ ファーマシューティカルズ，インコーポレイテッド マラリア、結核、及びｍａｃ病の治療方法
NZ602544A (en) 2010-03-22 2014-11-28 Cempra Pharmaceuticals Inc Crystalline forms of a macrolide, and uses therefor
US9051346B2 (en) 2010-05-20 2015-06-09 Cempra Pharmaceuticals, Inc. Process for preparing triazole-containing ketolide antibiotics
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
SG11201405895UA (en) 2012-03-27 2014-10-30 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
US9861616B2 (en) 2013-03-14 2018-01-09 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
JP6675973B2 (ja) 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ，インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
DK90788A (da) * 1987-02-24 1988-08-25 Beecham Group Plc Erythromycinderivater
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
WO1993021199A1 (en) * 1992-04-22 1993-10-28 Taisho Pharmaceutical Co., Ltd. 5-o-desosaminylerythronolide a derivative
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
CA2154550A1 (en) * 1993-01-26 1994-08-04 Yoko Misawa 5-o-desosaminylerythronolide derivatives

Also Published As

Publication number Publication date
DE69618607T2 (de) 2002-08-14
FR2739620B1 (fr) 1997-12-19
PT854879E (pt) 2002-07-31
CN1199403A (zh) 1998-11-18
AU708351B2 (en) 1999-08-05
EA000765B1 (ru) 2000-04-24
JP4327248B2 (ja) 2009-09-09
DE69618607D1 (de) 2002-02-21
SK283619B6 (sk) 2003-10-07
HUP9900136A1 (hu) 1999-05-28
CA2231562C (fr) 2006-11-28
CZ293430B6 (cs) 2004-04-14
NO312592B1 (no) 2002-06-03
EE9800109A (et) 1998-10-15
WO1997013774A2 (fr) 1997-04-17
UA52621C2 (uk) 2003-01-15
HUP9900136A3 (en) 2000-04-28
SK43198A3 (en) 1998-11-04
ES2171722T3 (es) 2002-09-16
AU7220896A (en) 1997-04-30
BG63752B1 (bg) 2002-11-29
PL183645B1 (pl) 2002-06-28
BG102350A (en) 1999-03-31
CZ105598A3 (cs) 1998-07-15
CA2231562A1 (fr) 1997-04-17
AP888A (en) 2000-11-10
FR2739620A1 (fr) 1997-04-11
ATE212034T1 (de) 2002-02-15
ZA966666B (en) 1997-08-06
TR199800624T1 (tr) 1998-06-22
EA199800280A1 (ru) 1998-10-29
PL326001A1 (en) 1998-08-17
US6011142A (en) 2000-01-04
EE03878B1 (et) 2002-10-15
GEP20032899B (en) 2003-02-25
KR19990064100A (ko) 1999-07-26
NO981630L (no) 1998-04-08
WO1997013774A3 (fr) 1997-05-29
JPH11513401A (ja) 1999-11-16
BR9610959A (pt) 1999-03-02
EP0854879A2 (fr) 1998-07-29
IL123613A0 (en) 1998-10-30
RO118874B1 (ro) 2003-12-30
DK0854879T3 (da) 2002-05-06
CN1067401C (zh) 2001-06-20
MX9802655A (es) 1998-11-30
EP0854879B1 (fr) 2002-01-16
KR100451063B1 (ko) 2004-12-17
AR004688A1 (es) 1999-03-10
NO981630D0 (no) 1998-04-08

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