SMT201400154B - Composti di triazolopiridina come inibitori di chinasi pim - Google Patents
Composti di triazolopiridina come inibitori di chinasi pimInfo
- Publication number
- SMT201400154B SMT201400154B SM201400154T SM201400154T SMT201400154B SM T201400154 B SMT201400154 B SM T201400154B SM 201400154 T SM201400154 T SM 201400154T SM 201400154 T SM201400154 T SM 201400154T SM T201400154 B SMT201400154 B SM T201400154B
- Authority
- SM
- San Marino
- Prior art keywords
- kinase inhibitors
- pim kinase
- triazolopyridine compounds
- triazolopyridine
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Transplantation (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8995208P | 2008-08-19 | 2008-08-19 | |
US17527709P | 2009-05-04 | 2009-05-04 | |
PCT/US2009/054193 WO2010022076A1 (en) | 2008-08-19 | 2009-08-18 | Triazolopyridine compounds as pim kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
SMT201400154B true SMT201400154B (it) | 2015-01-15 |
Family
ID=41227138
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SM201400154T SMT201400154B (it) | 2008-08-19 | 2014-10-21 | Composti di triazolopiridina come inibitori di chinasi pim |
Country Status (17)
Country | Link |
---|---|
US (1) | US8575145B2 (de) |
EP (1) | EP2334677B1 (de) |
JP (2) | JP5518072B2 (de) |
CN (1) | CN102186851B (de) |
AR (1) | AR073079A1 (de) |
CA (1) | CA2734831C (de) |
DK (1) | DK2334677T3 (de) |
ES (1) | ES2439501T3 (de) |
HR (1) | HRP20131140T1 (de) |
PL (1) | PL2334677T3 (de) |
PT (1) | PT2334677E (de) |
RS (1) | RS53079B (de) |
SI (1) | SI2334677T1 (de) |
SM (1) | SMT201400154B (de) |
TW (1) | TWI496779B (de) |
UY (1) | UY32057A (de) |
WO (1) | WO2010022076A1 (de) |
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EA019085B1 (ru) | 2007-09-14 | 2014-01-30 | Янссен Фармасьютикалз, Инк. | 1',3-двузамещенные 4-(арил-х-фенил)-1н-пиридин-2-оны |
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JP5357763B2 (ja) | 2006-11-06 | 2013-12-04 | トレロ ファーマシューティカルズ, インコーポレイテッド | イミダゾ[1,2−b]ピリダジン誘導体およびピラゾロ[1,5−a]ピリダジン誘導体およびプロテインキナーゼインヒビターとしてのこれらの使用 |
WO2008082839A2 (en) | 2006-12-29 | 2008-07-10 | Abbott Laboratories | Pim kinase inhibitors as cancer chemotherapeutics |
JP2010522765A (ja) * | 2007-03-28 | 2010-07-08 | アレイ バイオファーマ、インコーポレイテッド | 受容体チロシンキナーゼとしてのイミダゾ[1,2−a]ピリジン化合物 |
-
2009
- 2009-08-14 TW TW098127485A patent/TWI496779B/zh not_active IP Right Cessation
- 2009-08-18 SI SI200930782T patent/SI2334677T1/sl unknown
- 2009-08-18 JP JP2011523939A patent/JP5518072B2/ja not_active Expired - Fee Related
- 2009-08-18 US US13/059,902 patent/US8575145B2/en active Active
- 2009-08-18 CN CN2009801413028A patent/CN102186851B/zh not_active Expired - Fee Related
- 2009-08-18 EP EP09791625.8A patent/EP2334677B1/de active Active
- 2009-08-18 DK DK09791625.8T patent/DK2334677T3/da active
- 2009-08-18 RS RS20130557A patent/RS53079B/en unknown
- 2009-08-18 UY UY0001032057A patent/UY32057A/es active IP Right Grant
- 2009-08-18 WO PCT/US2009/054193 patent/WO2010022076A1/en active Application Filing
- 2009-08-18 PT PT97916258T patent/PT2334677E/pt unknown
- 2009-08-18 AR ARP090103170A patent/AR073079A1/es active IP Right Grant
- 2009-08-18 CA CA2734831A patent/CA2734831C/en not_active Expired - Fee Related
- 2009-08-18 PL PL09791625T patent/PL2334677T3/pl unknown
- 2009-08-18 ES ES09791625.8T patent/ES2439501T3/es active Active
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2013
- 2013-11-28 HR HRP20131140AT patent/HRP20131140T1/hr unknown
-
2014
- 2014-03-07 JP JP2014044674A patent/JP2014129409A/ja not_active Withdrawn
- 2014-10-21 SM SM201400154T patent/SMT201400154B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
JP2012500277A (ja) | 2012-01-05 |
RS53079B (en) | 2014-06-30 |
AR073079A1 (es) | 2010-10-13 |
EP2334677B1 (de) | 2013-10-09 |
EP2334677A1 (de) | 2011-06-22 |
US20110144085A1 (en) | 2011-06-16 |
JP2014129409A (ja) | 2014-07-10 |
HRP20131140T1 (hr) | 2014-01-03 |
WO2010022076A1 (en) | 2010-02-25 |
DK2334677T3 (da) | 2013-11-18 |
PL2334677T3 (pl) | 2014-03-31 |
SI2334677T1 (sl) | 2013-12-31 |
CA2734831A1 (en) | 2010-02-25 |
CN102186851B (zh) | 2013-06-12 |
JP5518072B2 (ja) | 2014-06-11 |
US8575145B2 (en) | 2013-11-05 |
CA2734831C (en) | 2017-04-18 |
ES2439501T3 (es) | 2014-01-23 |
CN102186851A (zh) | 2011-09-14 |
PT2334677E (pt) | 2013-11-26 |
TWI496779B (zh) | 2015-08-21 |
UY32057A (es) | 2011-01-31 |
TW201008940A (en) | 2010-03-01 |
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