SK413591A3 - Substituted androsta-1,4-diene 3,17-diones,method of their production and use and pharmaceutical agent - Google Patents

Substituted androsta-1,4-diene 3,17-diones,method of their production and use and pharmaceutical agent Download PDF

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Publication number
SK413591A3
SK413591A3 SK4135-91A SK413591A SK413591A3 SK 413591 A3 SK413591 A3 SK 413591A3 SK 413591 A SK413591 A SK 413591A SK 413591 A3 SK413591 A3 SK 413591A3
Authority
SK
Slovakia
Prior art keywords
compound
formula
diene
dione
hydrogen
Prior art date
Application number
SK4135-91A
Other languages
English (en)
Slovak (sk)
Inventor
Franco Buzzetti
Natale Barbugian
Paolo Lombardi
Salle Enrico Di
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10582036&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK413591(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of SK413591A3 publication Critical patent/SK413591A3/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SK4135-91A 1985-07-09 1991-12-30 Substituted androsta-1,4-diene 3,17-diones,method of their production and use and pharmaceutical agent SK413591A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858517360A GB8517360D0 (en) 1985-07-09 1985-07-09 Substituted androsta-1,4-diene-3,17-diones

Publications (1)

Publication Number Publication Date
SK413591A3 true SK413591A3 (en) 1995-07-11

Family

ID=10582036

Family Applications (1)

Application Number Title Priority Date Filing Date
SK4135-91A SK413591A3 (en) 1985-07-09 1991-12-30 Substituted androsta-1,4-diene 3,17-diones,method of their production and use and pharmaceutical agent

Country Status (38)

Country Link
US (2) US4808616A (cg-RX-API-DMAC7.html)
JP (1) JPS6212797A (cg-RX-API-DMAC7.html)
KR (1) KR950003614B1 (cg-RX-API-DMAC7.html)
CN (1) CN86104664B (cg-RX-API-DMAC7.html)
AT (1) AT395157B (cg-RX-API-DMAC7.html)
AU (1) AU578840B2 (cg-RX-API-DMAC7.html)
BE (1) BE905067A (cg-RX-API-DMAC7.html)
BG (1) BG61370B2 (cg-RX-API-DMAC7.html)
BR (1) BR1100240A (cg-RX-API-DMAC7.html)
CA (1) CA1277656C (cg-RX-API-DMAC7.html)
CH (1) CH668599A5 (cg-RX-API-DMAC7.html)
CS (2) CS257794B2 (cg-RX-API-DMAC7.html)
CZ (1) CZ413591A3 (cg-RX-API-DMAC7.html)
DE (1) DE10199030I1 (cg-RX-API-DMAC7.html)
DK (1) DK163520C (cg-RX-API-DMAC7.html)
ES (2) ES8801304A1 (cg-RX-API-DMAC7.html)
FI (1) FI83424C (cg-RX-API-DMAC7.html)
FR (1) FR2584725B1 (cg-RX-API-DMAC7.html)
GB (2) GB8517360D0 (cg-RX-API-DMAC7.html)
GR (1) GR861780B (cg-RX-API-DMAC7.html)
HK (1) HK94190A (cg-RX-API-DMAC7.html)
HU (1) HU194274B (cg-RX-API-DMAC7.html)
IE (1) IE58949B1 (cg-RX-API-DMAC7.html)
IL (1) IL79336A (cg-RX-API-DMAC7.html)
IT (1) IT1196436B (cg-RX-API-DMAC7.html)
MY (1) MY102294A (cg-RX-API-DMAC7.html)
NL (2) NL193616C (cg-RX-API-DMAC7.html)
NO (2) NO165547C (cg-RX-API-DMAC7.html)
NZ (1) NZ216763A (cg-RX-API-DMAC7.html)
PH (1) PH21785A (cg-RX-API-DMAC7.html)
PT (1) PT82944B (cg-RX-API-DMAC7.html)
SE (1) SE468988B (cg-RX-API-DMAC7.html)
SG (1) SG80490G (cg-RX-API-DMAC7.html)
SK (1) SK413591A3 (cg-RX-API-DMAC7.html)
SU (2) SU1442077A3 (cg-RX-API-DMAC7.html)
UA (1) UA6046A1 (cg-RX-API-DMAC7.html)
YU (2) YU44585B (cg-RX-API-DMAC7.html)
ZA (1) ZA865079B (cg-RX-API-DMAC7.html)

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GB8617107D0 (en) * 1986-07-14 1986-08-20 Erba Farmitalia 6-/7-methylenandrosta-1 4-diene-3 17-dione derivatives
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GB8801697D0 (en) * 1988-01-26 1988-02-24 Erba Farmitalia Improvements in synthesis of 6-methylene derivatives of androsta-1 4-diene-3 17-dione
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US6511970B1 (en) 1996-09-13 2003-01-28 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of products that induce transforming growth factor-beta and/or apoptosis in the ovarian epithelium
US6765002B2 (en) 2000-03-21 2004-07-20 Gustavo Rodriguez Prevention of ovarian cancer by administration of products that induce transforming growth factor-β and/or apoptosis in the ovarian epithelium
US6034074A (en) 1996-09-13 2000-03-07 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of a Vitamin D compound
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WO2001004342A1 (en) * 1999-07-07 2001-01-18 Pharmacia & Upjohn Company Process to prepare exemestane
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US20040082557A1 (en) * 2001-01-26 2004-04-29 Wajszczuk Charles Paul Methods for treating estrogen-dependent disorders
JP2004519490A (ja) * 2001-01-26 2004-07-02 フアルマシア・イタリア・エツセ・ピー・アー エキセメスタンによるホルモン依存性異常症の組合せ治療方法
PL231418B1 (pl) 2001-02-19 2019-02-28 Novartis Ag 40-O-( 2-hydroksyetylo)- rapamycyna do zastosowania w leczeniu guzów litych płuc, innych niż nowotwór tkanki limfatycznej
KR20080091866A (ko) 2001-05-16 2008-10-14 노파르티스 아게 Ν-｛5-[4-(4-메틸-피페라지노-메틸)-벤조일아미도]-2-메틸페닐｝-4-(3-피리딜)-2-피리미딘-아민 및 화학치료제를 포함하는 배합물
GB0120147D0 (en) * 2001-08-17 2001-10-10 Metris Therapeutics Ltd Treatment method
US20040043938A1 (en) * 2001-11-06 2004-03-04 Dinesh Purandare Combination therapy for estrogen-dependent disorders
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CN1304413C (zh) * 2002-10-24 2007-03-14 上海华拓医药科技发展有限公司 一种抗癌药物依西美坦制备方法
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US10174070B2 (en) * 2005-09-30 2019-01-08 Endece Llc 6-substituted estradiol derivatives and methods of use
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CN101443002B (zh) 2006-05-09 2012-03-21 诺瓦提斯公司 包含铁螯合剂和抗肿瘤药的组合及其用途
US20080161324A1 (en) * 2006-09-14 2008-07-03 Johansen Lisa M Compositions and methods for treatment of viral diseases
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Also Published As

Publication number Publication date
BG61370B2 (bg) 1997-06-30
JPH0443919B2 (cg-RX-API-DMAC7.html) 1992-07-20
FR2584725B1 (fr) 1988-05-13
MY102294A (en) 1992-05-15
IE861821L (en) 1987-01-09
DK324386A (da) 1987-01-10
AU578840B2 (en) 1988-11-03
FI862871A7 (fi) 1987-01-10
FR2584725A1 (fr) 1987-01-16
AT395157B (de) 1992-10-12
GR861780B (en) 1986-11-11
PT82944A (en) 1986-08-01
KR950003614B1 (ko) 1995-04-17
ES8801304A1 (es) 1987-12-16
BR1100240A (pt) 1999-12-28
ATA181986A (de) 1992-02-15
GB2177700A (en) 1987-01-28
BE905067A (fr) 1987-01-08
ES556550A0 (es) 1987-12-16
CN86104664A (zh) 1987-02-18
YU44628B (en) 1990-10-31
ZA865079B (en) 1987-03-25
CS258498B2 (en) 1988-08-16
GB2177700B (en) 1988-12-07
UA6046A1 (uk) 1994-12-29
NO165547B (no) 1990-11-19
FI83424C (fi) 1991-07-10
NO165547C (no) 1991-02-27
CH668599A5 (de) 1989-01-13
US4808616A (en) 1989-02-28
NL193616B (nl) 1999-12-01
KR870001140A (ko) 1987-03-11
HUT42780A (en) 1987-08-28
FI862871A0 (fi) 1986-07-07
NL300017I1 (nl) 2000-11-01
IL79336A (en) 1991-06-10
PH21785A (en) 1988-02-24
YU44585B (en) 1990-10-31
AU5979986A (en) 1987-01-15
US4904650A (en) 1990-02-27
SU1501923A3 (ru) 1989-08-15
DK324386D0 (da) 1986-07-08
YU103687A (en) 1988-08-31
HK94190A (en) 1990-11-23
GB8616585D0 (en) 1986-08-13
GB8517360D0 (en) 1985-08-14
DK163520B (da) 1992-03-09
DE10199030I1 (de) 2001-10-04
NO2000009I1 (no) 2000-10-05
IE58949B1 (en) 1993-12-01
DK163520C (da) 1992-07-27
SU1442077A3 (ru) 1988-11-30
CS257794B2 (en) 1988-06-15
NL300017I2 (nl) 2001-01-02
NO862753L (no) 1987-01-12
HU194274B (en) 1988-01-28
SE8603046L (sv) 1987-01-10
CZ413591A3 (en) 1994-03-16
NL193616C (nl) 2000-04-04
NL8601785A (nl) 1987-02-02
IT1196436B (it) 1988-11-16
JPS6212797A (ja) 1987-01-21
ES557466A0 (es) 1988-06-01
YU120186A (en) 1988-02-29
IT8621004A0 (it) 1986-07-02
CS521486A2 (en) 1987-09-17
FI83424B (fi) 1991-03-28
CA1277656C (en) 1990-12-11
SE468988B (sv) 1993-04-26
SE8603046D0 (sv) 1986-07-08
NO862753D0 (no) 1986-07-08
CN86104664B (zh) 1988-06-29
IL79336A0 (en) 1986-10-31
PT82944B (pt) 1989-01-30
NZ216763A (en) 1988-05-30
ES8802429A1 (es) 1988-06-01
SG80490G (en) 1990-11-23

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