SK283385B6 - Deriváty piperazín-2,5-diónu, spôsob ich prípravy, ich použitie a farmaceutický alebo veterinárny prostriedok s ich obsahom - Google Patents
Deriváty piperazín-2,5-diónu, spôsob ich prípravy, ich použitie a farmaceutický alebo veterinárny prostriedok s ich obsahom Download PDFInfo
- Publication number
- SK283385B6 SK283385B6 SK835-97A SK83597A SK283385B6 SK 283385 B6 SK283385 B6 SK 283385B6 SK 83597 A SK83597 A SK 83597A SK 283385 B6 SK283385 B6 SK 283385B6
- Authority
- SK
- Slovakia
- Prior art keywords
- methyl
- benzylidene
- formula
- dioxo
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Electron Tubes For Measurement (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9426090.8A GB9426090D0 (en) | 1994-12-23 | 1994-12-23 | Pharmaceutical compounds |
| PCT/GB1995/003029 WO1996020180A1 (en) | 1994-12-23 | 1995-12-22 | Piperazine-2,5-dione derivatives as modulators of multidrug resistance |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SK83597A3 SK83597A3 (en) | 1998-04-08 |
| SK283385B6 true SK283385B6 (sk) | 2003-06-03 |
Family
ID=10766502
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK835-97A SK283385B6 (sk) | 1994-12-23 | 1995-12-22 | Deriváty piperazín-2,5-diónu, spôsob ich prípravy, ich použitie a farmaceutický alebo veterinárny prostriedok s ich obsahom |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US5935955A (cs) |
| EP (1) | EP0799210B1 (cs) |
| JP (1) | JPH10511385A (cs) |
| KR (1) | KR100412167B1 (cs) |
| CN (1) | CN1108294C (cs) |
| AT (1) | ATE204569T1 (cs) |
| AU (1) | AU700891B2 (cs) |
| BG (1) | BG63305B1 (cs) |
| BR (1) | BR9510429A (cs) |
| CA (1) | CA2207548A1 (cs) |
| CZ (1) | CZ288935B6 (cs) |
| DE (1) | DE69522342T2 (cs) |
| DK (1) | DK0799210T3 (cs) |
| ES (1) | ES2160726T3 (cs) |
| FI (1) | FI972661L (cs) |
| GB (2) | GB9426090D0 (cs) |
| HU (1) | HUT77740A (cs) |
| IL (1) | IL116526A (cs) |
| MY (1) | MY131762A (cs) |
| NO (1) | NO308532B1 (cs) |
| NZ (1) | NZ297849A (cs) |
| PL (1) | PL186851B1 (cs) |
| PT (1) | PT799210E (cs) |
| SK (1) | SK283385B6 (cs) |
| UA (1) | UA61879C2 (cs) |
| WO (1) | WO1996020180A1 (cs) |
| ZA (1) | ZA9510908B (cs) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9708805D0 (en) | 1997-05-01 | 1997-06-25 | Smithkline Beecham Plc | Compounds |
| GB9810876D0 (en) | 1998-05-20 | 1998-07-22 | Smithkline Beecham Plc | Compounds |
| SK4782001A3 (en) | 1998-10-08 | 2001-11-06 | Smithkline Beecham Plc | Tetrahydrobenzazepine derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents) |
| EP1210093A4 (en) * | 1999-09-03 | 2005-01-12 | Polytherics Ltd | DEGRADABLE POLYMERS |
| US6828412B1 (en) * | 1999-09-03 | 2004-12-07 | School Of Pharmacy, University Of London | Degradable polymers |
| EP2266607A3 (en) | 1999-10-01 | 2011-04-20 | Immunogen, Inc. | Immunoconjugates for treating cancer |
| US7220414B2 (en) | 2000-09-06 | 2007-05-22 | A.P. Pharma, Inc. | Degradable polyacetal polymers |
| US6693099B2 (en) | 2000-10-17 | 2004-02-17 | The Procter & Gamble Company | Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance |
| US6376514B1 (en) | 2000-10-17 | 2002-04-23 | The Procter & Gamble Co. | Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof |
| JP2005508990A (ja) * | 2001-11-07 | 2005-04-07 | ファルマシア・コーポレーション | 真核細胞におけるポリアミドの取込みおよび核蓄積を促進する方法 |
| US8710062B2 (en) * | 2011-03-11 | 2014-04-29 | Taipei Medical University | Piperazinedione compounds |
| CN103396372B (zh) * | 2013-08-09 | 2015-05-20 | 中国科学院南海海洋研究所 | 一类2,5-二酮哌嗪衍生物及其制备方法和在制备抗海洋污损生物防除剂中的应用 |
| BR112021012639A2 (pt) * | 2018-12-27 | 2021-09-28 | Holosmedic | Novo composto e composição farmacêutica compreendendo o mesmo para intensificar atividade anticâncer |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2103479T3 (es) * | 1992-07-10 | 1997-09-16 | Glaxo Lab Sa | Derivados de anilida. |
| GB9217331D0 (en) * | 1992-08-14 | 1992-09-30 | Xenova Ltd | Pharmaceutical compounds |
| AU664920B2 (en) * | 1992-08-14 | 1995-12-07 | Asahi Breweries, Ltd. | Peptide having allergenicity |
| GB9402807D0 (en) * | 1994-02-14 | 1994-04-06 | Xenova Ltd | Pharmaceutical compounds |
| GB9410387D0 (en) * | 1994-05-24 | 1994-07-13 | Xenova Ltd | Pharmaceutical compounds |
-
1994
- 1994-12-23 GB GBGB9426090.8A patent/GB9426090D0/en active Pending
-
1995
- 1995-12-21 ZA ZA9510908A patent/ZA9510908B/xx unknown
- 1995-12-22 PT PT95941799T patent/PT799210E/pt unknown
- 1995-12-22 PL PL95320915A patent/PL186851B1/pl not_active IP Right Cessation
- 1995-12-22 AT AT95941799T patent/ATE204569T1/de not_active IP Right Cessation
- 1995-12-22 ES ES95941799T patent/ES2160726T3/es not_active Expired - Lifetime
- 1995-12-22 CA CA002207548A patent/CA2207548A1/en not_active Abandoned
- 1995-12-22 FI FI972661A patent/FI972661L/fi not_active IP Right Cessation
- 1995-12-22 CZ CZ19971902A patent/CZ288935B6/cs not_active IP Right Cessation
- 1995-12-22 JP JP8520303A patent/JPH10511385A/ja not_active Ceased
- 1995-12-22 HU HU9800446A patent/HUT77740A/hu unknown
- 1995-12-22 UA UA97062956A patent/UA61879C2/uk unknown
- 1995-12-22 US US08/860,328 patent/US5935955A/en not_active Expired - Fee Related
- 1995-12-22 DE DE69522342T patent/DE69522342T2/de not_active Expired - Fee Related
- 1995-12-22 NZ NZ297849A patent/NZ297849A/en unknown
- 1995-12-22 AU AU43102/96A patent/AU700891B2/en not_active Ceased
- 1995-12-22 CN CN95197673A patent/CN1108294C/zh not_active Expired - Fee Related
- 1995-12-22 SK SK835-97A patent/SK283385B6/sk unknown
- 1995-12-22 GB GB9712179A patent/GB2311780B/en not_active Expired - Fee Related
- 1995-12-22 WO PCT/GB1995/003029 patent/WO1996020180A1/en not_active Ceased
- 1995-12-22 BR BR9510429A patent/BR9510429A/pt not_active Application Discontinuation
- 1995-12-22 DK DK95941799T patent/DK0799210T3/da active
- 1995-12-22 IL IL11652695A patent/IL116526A/xx not_active IP Right Cessation
- 1995-12-22 KR KR1019970704226A patent/KR100412167B1/ko not_active Expired - Fee Related
- 1995-12-22 EP EP95941799A patent/EP0799210B1/en not_active Expired - Lifetime
- 1995-12-23 MY MYPI95004072A patent/MY131762A/en unknown
-
1997
- 1997-06-11 BG BG101601A patent/BG63305B1/bg unknown
- 1997-06-23 NO NO972938A patent/NO308532B1/no not_active IP Right Cessation
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