SK179899A3 - Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders - Google Patents
Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders Download PDFInfo
- Publication number
- SK179899A3 SK179899A3 SK1798-99A SK179899A SK179899A3 SK 179899 A3 SK179899 A3 SK 179899A3 SK 179899 A SK179899 A SK 179899A SK 179899 A3 SK179899 A3 SK 179899A3
- Authority
- SK
- Slovakia
- Prior art keywords
- alkyl
- group
- cycloalkyl
- substituted
- cor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5162897P | 1997-07-03 | 1997-07-03 | |
US8066598P | 1998-04-03 | 1998-04-03 | |
PCT/US1998/013913 WO1999001454A1 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Publications (1)
Publication Number | Publication Date |
---|---|
SK179899A3 true SK179899A3 (en) | 2001-12-03 |
Family
ID=26729655
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK1798-99A SK179899A3 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Country Status (20)
Country | Link |
---|---|
US (3) | US6143743A (et) |
EP (1) | EP0994877A1 (et) |
JP (1) | JP2002507996A (et) |
KR (1) | KR20010014431A (et) |
CN (1) | CN1268137A (et) |
AR (1) | AR016307A1 (et) |
AU (1) | AU746706B2 (et) |
BR (1) | BR9810508A (et) |
CA (1) | CA2294117A1 (et) |
EE (1) | EE04280B1 (et) |
HR (1) | HRP980375A2 (et) |
HU (1) | HUP0100179A3 (et) |
IL (1) | IL133800A0 (et) |
MY (1) | MY132871A (et) |
NO (1) | NO316119B1 (et) |
NZ (1) | NZ502642A (et) |
PL (1) | PL337888A1 (et) |
SK (1) | SK179899A3 (et) |
TW (1) | TW589309B (et) |
WO (1) | WO1999001454A1 (et) |
Families Citing this family (74)
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PT946550E (pt) * | 1996-12-11 | 2005-09-30 | Aventis Pharma Inc | Preparacao de [1s-[1a,2b,3b,4a(s*)]]-4-[7-[1-(3-cloro-2-tienil)metil]propil]amino]-3h-imidazo[4,5-b]piridin-3-il]-n-etil-2,3-di-hidroxiciclopentanocarboxamida |
US6365589B1 (en) * | 1998-07-02 | 2002-04-02 | Bristol-Myers Squibb Pharma Company | Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists |
US6124463A (en) * | 1998-07-02 | 2000-09-26 | Dupont Pharmaceuticals | Benzimidazoles as corticotropin release factor antagonists |
JP2002533465A (ja) * | 1998-12-23 | 2002-10-08 | デュポン ファーマシューティカルズ カンパニー | Xa因子阻害剤としての窒素を含む複素二環類 |
US6271380B1 (en) * | 1998-12-30 | 2001-08-07 | Dupont Pharmaceuticals Company | 1H-imidazo[4,5-d]pyridazin-7-ones, 3H-imidazo-[4,5-c]pyridin-4-ones and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands |
WO2000059908A2 (en) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines as crf antagonists |
AU4331500A (en) | 1999-04-06 | 2000-10-23 | Du Pont Pharmaceuticals Company | Pyrazolotriazines as crf antagonists |
US6432989B1 (en) * | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
JP2003516992A (ja) * | 1999-12-17 | 2003-05-20 | デュポン ファーマシューティカルズ カンパニー | イミダゾピリミジニル誘導体およびイミダゾピリジニル誘導体 |
KR20030016222A (ko) * | 2000-02-14 | 2003-02-26 | 니뽄 다바코 산교 가부시키가이샤 | 수술후 스트레스 예방ㆍ치료제 |
US20040077605A1 (en) * | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
AR028782A1 (es) * | 2000-07-05 | 2003-05-21 | Taisho Pharmaceutical Co Ltd | Derivados heterociclicos tetrahidropiridino o piperidino |
EP1301511A2 (en) | 2000-07-14 | 2003-04-16 | Bristol-Myers Squibb Pharma Company | IMIDAZO 1,2-a]PYRAZINES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS |
EP1854798A3 (en) | 2000-09-19 | 2007-11-28 | Bristol-Myers Squibb Company | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
GB0100623D0 (en) | 2001-01-10 | 2001-02-21 | Vernalis Res Ltd | Chemical compounds IV |
EP1359916A4 (en) | 2001-01-26 | 2004-04-07 | Bristol Myers Squibb Co | IMIDAZOLYLATED DERIVATIVES AS INHIBITORS OF CORTICOTROPIN RELEASE FACTOR |
TWI312347B (en) | 2001-02-08 | 2009-07-21 | Eisai R&D Man Co Ltd | Bicyclic nitrogen-containing condensed ring compounds |
US20040087548A1 (en) | 2001-02-27 | 2004-05-06 | Salvati Mark E. | Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
HU229317B1 (en) | 2001-03-13 | 2013-10-28 | Bristol Myers Squibb Pharma Co | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine derivatives, and enantiomers of the same az cortikotropine releasing factor (cfr) ligands |
CZ301491B6 (cs) | 2001-04-27 | 2010-03-24 | Eisai R&D Management Co., Ltd. | Pyrazolo[1,5-a]pyridiny a léciva s jejich obsahem |
RU2003135424A (ru) | 2001-05-14 | 2005-05-20 | Бристол-Маерс Сквибб Фарма Компани (Us) | Замещенные пиразиноны, пиридины и пиримидины в качестве лигандов кортикотропин высвобождающего фактора |
WO2003005969A2 (en) | 2001-07-12 | 2003-01-23 | Bristol-Myers Squibb Pharma Company | Tetrahydropurinones as corticotropin releasing factor |
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US20070129334A1 (en) * | 2001-10-30 | 2007-06-07 | Conforma Therapeutics Corporation | Orally Active Purine-Based Inhibitors of Heat Shock Protein 90 |
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JP4322211B2 (ja) | 2002-10-22 | 2009-08-26 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 7−フェニルピラゾロピリジン化合物 |
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-
1998
- 1998-07-02 HU HU0100179A patent/HUP0100179A3/hu unknown
- 1998-07-02 NZ NZ502642A patent/NZ502642A/en unknown
- 1998-07-02 US US09/109,877 patent/US6143743A/en not_active Expired - Lifetime
- 1998-07-02 CA CA002294117A patent/CA2294117A1/en not_active Abandoned
- 1998-07-02 WO PCT/US1998/013913 patent/WO1999001454A1/en not_active Application Discontinuation
- 1998-07-02 HR HR60/080,665A patent/HRP980375A2/hr not_active Application Discontinuation
- 1998-07-02 AU AU81819/98A patent/AU746706B2/en not_active Ceased
- 1998-07-02 EP EP98931795A patent/EP0994877A1/en not_active Withdrawn
- 1998-07-02 TW TW087110857A patent/TW589309B/zh active
- 1998-07-02 BR BR9810508-6A patent/BR9810508A/pt not_active IP Right Cessation
- 1998-07-02 IL IL13380098A patent/IL133800A0/xx unknown
- 1998-07-02 SK SK1798-99A patent/SK179899A3/sk unknown
- 1998-07-02 CN CN98808584A patent/CN1268137A/zh active Pending
- 1998-07-02 MY MYPI98003027A patent/MY132871A/en unknown
- 1998-07-02 JP JP50744099A patent/JP2002507996A/ja active Pending
- 1998-07-02 EE EEP199900607A patent/EE04280B1/et not_active IP Right Cessation
- 1998-07-02 KR KR1019997012619A patent/KR20010014431A/ko not_active Application Discontinuation
- 1998-07-02 PL PL98337888A patent/PL337888A1/xx unknown
- 1998-07-03 AR ARP980103234A patent/AR016307A1/es not_active Application Discontinuation
- 1998-12-10 US US09/208,778 patent/US6362180B1/en not_active Expired - Lifetime
-
1999
- 1999-12-27 NO NO19996483A patent/NO316119B1/no not_active IP Right Cessation
-
2001
- 2001-11-07 US US10/053,475 patent/US6642230B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
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PL337888A1 (en) | 2000-09-11 |
MY132871A (en) | 2007-10-31 |
EE9900607A (et) | 2000-08-15 |
NO316119B1 (no) | 2003-12-15 |
AU746706B2 (en) | 2002-05-02 |
CN1268137A (zh) | 2000-09-27 |
EE04280B1 (et) | 2004-04-15 |
NO996483D0 (no) | 1999-12-27 |
AR016307A1 (es) | 2001-07-04 |
JP2002507996A (ja) | 2002-03-12 |
AU8181998A (en) | 1999-01-25 |
NZ502642A (en) | 2002-06-28 |
KR20010014431A (ko) | 2001-02-26 |
CA2294117A1 (en) | 1999-01-14 |
US20030114468A1 (en) | 2003-06-19 |
HUP0100179A2 (hu) | 2001-11-28 |
NO996483L (no) | 2000-03-02 |
HRP980375A2 (en) | 1999-04-30 |
US6642230B2 (en) | 2003-11-04 |
EP0994877A1 (en) | 2000-04-26 |
US6362180B1 (en) | 2002-03-26 |
IL133800A0 (en) | 2001-04-30 |
US6143743A (en) | 2000-11-07 |
WO1999001454A1 (en) | 1999-01-14 |
BR9810508A (pt) | 2000-09-05 |
HUP0100179A3 (en) | 2002-12-28 |
TW589309B (en) | 2004-06-01 |
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