NO996483L - Imidasopyrimidiner og imidasopyridiner for behandling av neurologiske lidelser - Google Patents
Imidasopyrimidiner og imidasopyridiner for behandling av neurologiske lidelserInfo
- Publication number
- NO996483L NO996483L NO996483A NO996483A NO996483L NO 996483 L NO996483 L NO 996483L NO 996483 A NO996483 A NO 996483A NO 996483 A NO996483 A NO 996483A NO 996483 L NO996483 L NO 996483L
- Authority
- NO
- Norway
- Prior art keywords
- imidazopyrimidines
- imidazopyridines
- treatment
- neurological disorders
- neurological
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5162897P | 1997-07-03 | 1997-07-03 | |
US8066598P | 1998-04-03 | 1998-04-03 | |
PCT/US1998/013913 WO1999001454A1 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Publications (3)
Publication Number | Publication Date |
---|---|
NO996483D0 NO996483D0 (no) | 1999-12-27 |
NO996483L true NO996483L (no) | 2000-03-02 |
NO316119B1 NO316119B1 (no) | 2003-12-15 |
Family
ID=26729655
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO19996483A NO316119B1 (no) | 1997-07-03 | 1999-12-27 | Imidasopyrimidiner og imidasopyridiner, farmasöytisk sammensetning inneholdende samme og anvendelse av samme for fremstilling av medikamentet |
Country Status (20)
Country | Link |
---|---|
US (3) | US6143743A (no) |
EP (1) | EP0994877A1 (no) |
JP (1) | JP2002507996A (no) |
KR (1) | KR20010014431A (no) |
CN (1) | CN1268137A (no) |
AR (1) | AR016307A1 (no) |
AU (1) | AU746706B2 (no) |
BR (1) | BR9810508A (no) |
CA (1) | CA2294117A1 (no) |
EE (1) | EE04280B1 (no) |
HR (1) | HRP980375A2 (no) |
HU (1) | HUP0100179A3 (no) |
IL (1) | IL133800A0 (no) |
MY (1) | MY132871A (no) |
NO (1) | NO316119B1 (no) |
NZ (1) | NZ502642A (no) |
PL (1) | PL337888A1 (no) |
SK (1) | SK179899A3 (no) |
TW (1) | TW589309B (no) |
WO (1) | WO1999001454A1 (no) |
Families Citing this family (74)
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BR9713705A (pt) * | 1996-12-11 | 2000-05-09 | Rhone Poulenc Rorer Pharma | Composto, e, processo para a preparação do mesmo |
US6365589B1 (en) * | 1998-07-02 | 2002-04-02 | Bristol-Myers Squibb Pharma Company | Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists |
US6124463A (en) * | 1998-07-02 | 2000-09-26 | Dupont Pharmaceuticals | Benzimidazoles as corticotropin release factor antagonists |
BR9917080A (pt) * | 1998-12-23 | 2002-03-12 | Du Pont Pharm Co | Composto, composição farmacêutica, uso do composto e método de tratamento ou prevenção de uma disfunção tromboembólica |
US6271380B1 (en) * | 1998-12-30 | 2001-08-07 | Dupont Pharmaceuticals Company | 1H-imidazo[4,5-d]pyridazin-7-ones, 3H-imidazo-[4,5-c]pyridin-4-ones and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands |
WO2000059908A2 (en) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines as crf antagonists |
AU4331500A (en) | 1999-04-06 | 2000-10-23 | Du Pont Pharmaceuticals Company | Pyrazolotriazines as crf antagonists |
US6432989B1 (en) * | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
EP1244666A1 (en) * | 1999-12-17 | 2002-10-02 | Bristol-Myers Squibb Pharma Company | Imidazopyrimidinyl and imidazopyridinyl derivatives |
CA2398956A1 (en) * | 2000-02-14 | 2001-08-16 | Japan Tobacco Inc. | A pharmaceutical composition for prophylaxis or therapy of a postoperative stress |
US20040077605A1 (en) * | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
AR028782A1 (es) | 2000-07-05 | 2003-05-21 | Taisho Pharmaceutical Co Ltd | Derivados heterociclicos tetrahidropiridino o piperidino |
CA2419626A1 (en) | 2000-07-14 | 2002-01-24 | Rajagopal Bakthavatachalam | Imidazo¬1,2-a|pyrazines for the treatment of neurological disorders |
EP1854798A3 (en) | 2000-09-19 | 2007-11-28 | Bristol-Myers Squibb Company | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
GB0100623D0 (en) | 2001-01-10 | 2001-02-21 | Vernalis Res Ltd | Chemical compounds IV |
RU2003126188A (ru) | 2001-01-26 | 2005-03-27 | Бристол-Маерс Сквибб Компани (Us) | Имидазолильные производные как ингибиторы кортикотропин-рилизинг фактора |
TWI312347B (en) | 2001-02-08 | 2009-07-21 | Eisai R&D Man Co Ltd | Bicyclic nitrogen-containing condensed ring compounds |
US20040087548A1 (en) | 2001-02-27 | 2004-05-06 | Salvati Mark E. | Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
US20030125330A1 (en) | 2001-03-13 | 2003-07-03 | Gilligan Paul J. | 4 - (2-butylamino) - 2, 7-dimethyl-8- (2-methyl-6-methoxypyrid-3-yl) pyrazolo- [1,5-A] - 1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands |
CA2443802C (en) | 2001-04-27 | 2010-04-13 | Eisai Co., Ltd. | Pyrazolo[1,5-a]pyridines and medicines containing the same |
CN1527710A (zh) | 2001-05-14 | 2004-09-08 | ����˹�ж�-����˹˹����ҩƷ��˾ | 作为促肾上腺皮质激素释放因子配体的取代的吡嗪酮、吡啶和嘧啶 |
WO2003005969A2 (en) | 2001-07-12 | 2003-01-23 | Bristol-Myers Squibb Pharma Company | Tetrahydropurinones as corticotropin releasing factor |
US7276526B2 (en) | 2001-07-13 | 2007-10-02 | Bristol-Myers Squibb Pharma Company | Substituted thiazoles and oxazoles as corticotropin releasing hormone ligands |
AU2002343604C1 (en) | 2001-10-30 | 2009-09-17 | Conforma Therapeutics Corporation | Purine analogs having HSP90-inhibiting activity |
US20070129334A1 (en) * | 2001-10-30 | 2007-06-07 | Conforma Therapeutics Corporation | Orally Active Purine-Based Inhibitors of Heat Shock Protein 90 |
US20030119831A1 (en) | 2001-11-20 | 2003-06-26 | Hartz Richard A. | 3,7-dihydro-purine-2,6-dione derivatives as CRF receptor ligands |
NZ533958A (en) * | 2002-01-07 | 2007-09-28 | Eisai Co Ltd | Deazapurines and uses thereof |
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US7176216B2 (en) | 2002-10-22 | 2007-02-13 | Eisai Co., Ltd. | 7-phenylpyrazolopyridine compounds |
US7332508B2 (en) | 2002-12-18 | 2008-02-19 | Novo Nordisk A/S | Substituted homopiperidine, piperidine or pyrrolidine derivatives |
US7834014B2 (en) | 2003-04-09 | 2010-11-16 | Biogen Idec Ma Inc. | A2a adenosine receptor antagonists |
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US7674791B2 (en) | 2003-04-09 | 2010-03-09 | Biogen Idec Ma Inc. | Triazolopyrazines and methods of making and using the same |
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US7572805B2 (en) | 2004-07-14 | 2009-08-11 | Bristol-Myers Squibb Company | Pyrrolo(oxo)isoquinolines as 5HT ligands |
DE102004037554A1 (de) * | 2004-08-03 | 2006-03-16 | Sanofi-Aventis Deutschland Gmbh | Substituierte 8-Aminoalkylthio-xanthine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
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ATE421518T1 (de) * | 2005-02-10 | 2009-02-15 | Bristol Myers Squibb Co | Dihydrochinazolinone als 5ht-modulatoren |
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JP2010523663A (ja) * | 2007-04-11 | 2010-07-15 | メルク・シャープ・エンド・ドーム・コーポレイション | 第3級アミド、スルホンアミド、カルバミン酸及び尿素末端基をもつcgrp受容体アンタゴニスト |
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CA2721670C (en) | 2008-04-15 | 2013-09-10 | Eisai R&D Management Co., Ltd. | 3-phenylpyrazolo[5,1-b]thiazole compound |
US20110152313A1 (en) * | 2008-06-20 | 2011-06-23 | Macquarie University | Synthesis of ageladine a and analogs thereof |
FR2933982A1 (fr) * | 2008-07-18 | 2010-01-22 | Sanofi Aventis | Nouveaux derives imidazo°1,2-a!pyrimidine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met |
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-
1998
- 1998-07-02 AU AU81819/98A patent/AU746706B2/en not_active Ceased
- 1998-07-02 EE EEP199900607A patent/EE04280B1/xx not_active IP Right Cessation
- 1998-07-02 NZ NZ502642A patent/NZ502642A/en unknown
- 1998-07-02 JP JP50744099A patent/JP2002507996A/ja active Pending
- 1998-07-02 BR BR9810508-6A patent/BR9810508A/pt not_active IP Right Cessation
- 1998-07-02 PL PL98337888A patent/PL337888A1/xx unknown
- 1998-07-02 TW TW087110857A patent/TW589309B/zh active
- 1998-07-02 HR HR60/080,665A patent/HRP980375A2/hr not_active Application Discontinuation
- 1998-07-02 IL IL13380098A patent/IL133800A0/xx unknown
- 1998-07-02 SK SK1798-99A patent/SK179899A3/sk unknown
- 1998-07-02 CN CN98808584A patent/CN1268137A/zh active Pending
- 1998-07-02 MY MYPI98003027A patent/MY132871A/en unknown
- 1998-07-02 CA CA002294117A patent/CA2294117A1/en not_active Abandoned
- 1998-07-02 HU HU0100179A patent/HUP0100179A3/hu unknown
- 1998-07-02 US US09/109,877 patent/US6143743A/en not_active Expired - Lifetime
- 1998-07-02 KR KR1019997012619A patent/KR20010014431A/ko not_active Application Discontinuation
- 1998-07-02 WO PCT/US1998/013913 patent/WO1999001454A1/en not_active Application Discontinuation
- 1998-07-02 EP EP98931795A patent/EP0994877A1/en not_active Withdrawn
- 1998-07-03 AR ARP980103234A patent/AR016307A1/es not_active Application Discontinuation
- 1998-12-10 US US09/208,778 patent/US6362180B1/en not_active Expired - Lifetime
-
1999
- 1999-12-27 NO NO19996483A patent/NO316119B1/no not_active IP Right Cessation
-
2001
- 2001-11-07 US US10/053,475 patent/US6642230B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
HUP0100179A3 (en) | 2002-12-28 |
HRP980375A2 (en) | 1999-04-30 |
PL337888A1 (en) | 2000-09-11 |
MY132871A (en) | 2007-10-31 |
AR016307A1 (es) | 2001-07-04 |
JP2002507996A (ja) | 2002-03-12 |
US6362180B1 (en) | 2002-03-26 |
HUP0100179A2 (hu) | 2001-11-28 |
NZ502642A (en) | 2002-06-28 |
TW589309B (en) | 2004-06-01 |
EE04280B1 (et) | 2004-04-15 |
EP0994877A1 (en) | 2000-04-26 |
NO996483D0 (no) | 1999-12-27 |
US20030114468A1 (en) | 2003-06-19 |
KR20010014431A (ko) | 2001-02-26 |
EE9900607A (et) | 2000-08-15 |
IL133800A0 (en) | 2001-04-30 |
US6143743A (en) | 2000-11-07 |
WO1999001454A1 (en) | 1999-01-14 |
SK179899A3 (en) | 2001-12-03 |
BR9810508A (pt) | 2000-09-05 |
AU746706B2 (en) | 2002-05-02 |
CN1268137A (zh) | 2000-09-27 |
US6642230B2 (en) | 2003-11-04 |
NO316119B1 (no) | 2003-12-15 |
CA2294117A1 (en) | 1999-01-14 |
AU8181998A (en) | 1999-01-25 |
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