SK10772002A3 - Pyridopyrimidinónové deriváty na liečbu neurodegeneratívnych ochorení - Google Patents

Pyridopyrimidinónové deriváty na liečbu neurodegeneratívnych ochorení Download PDF

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Publication number
SK10772002A3
SK10772002A3 SK1077-2002A SK10772002A SK10772002A3 SK 10772002 A3 SK10772002 A3 SK 10772002A3 SK 10772002 A SK10772002 A SK 10772002A SK 10772002 A3 SK10772002 A3 SK 10772002A3
Authority
SK
Slovakia
Prior art keywords
pyrimidin
pyrido
phenylamino
ethyl
propyl
Prior art date
Application number
SK1077-2002A
Other languages
English (en)
Slovak (sk)
Inventor
Richard John Booth
Arindam Chatterjee
Thomas Charles Malone
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of SK10772002A3 publication Critical patent/SK10772002A3/sk

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SK1077-2002A 2000-01-27 2000-11-30 Pyridopyrimidinónové deriváty na liečbu neurodegeneratívnych ochorení SK10772002A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17840000P 2000-01-27 2000-01-27
PCT/US2000/032572 WO2001055148A1 (en) 2000-01-27 2000-11-30 Pyridopyrimidinone derivatives for treatment of neurodegenerative disease

Publications (1)

Publication Number Publication Date
SK10772002A3 true SK10772002A3 (sk) 2004-01-08

Family

ID=22652409

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1077-2002A SK10772002A3 (sk) 2000-01-27 2000-11-30 Pyridopyrimidinónové deriváty na liečbu neurodegeneratívnych ochorení

Country Status (22)

Country Link
US (1) US20040224958A1 (es)
EP (1) EP1255755A1 (es)
JP (1) JP2003523358A (es)
KR (1) KR20020070520A (es)
CN (1) CN1433417A (es)
AR (1) AR029437A1 (es)
AU (1) AU1808601A (es)
BR (1) BR0017075A (es)
CA (1) CA2394525A1 (es)
CO (1) CO5280216A1 (es)
CZ (1) CZ20022521A3 (es)
GT (1) GT200100005A (es)
HN (1) HN2001000012A (es)
HU (1) HUP0203803A3 (es)
IL (1) IL150742A0 (es)
PA (1) PA8510801A1 (es)
PE (1) PE20011228A1 (es)
PL (1) PL357634A1 (es)
SK (1) SK10772002A3 (es)
SV (1) SV2002000287A (es)
TN (1) TNSN01018A1 (es)
WO (1) WO2001055148A1 (es)

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Also Published As

Publication number Publication date
AU1808601A (en) 2001-08-07
CZ20022521A3 (cs) 2003-02-12
EP1255755A1 (en) 2002-11-13
CN1433417A (zh) 2003-07-30
PA8510801A1 (es) 2002-12-11
HN2001000012A (es) 2001-07-09
US20040224958A1 (en) 2004-11-11
CA2394525A1 (en) 2001-08-02
AR029437A1 (es) 2003-06-25
KR20020070520A (ko) 2002-09-09
WO2001055148A1 (en) 2001-08-02
BR0017075A (pt) 2002-11-05
JP2003523358A (ja) 2003-08-05
PE20011228A1 (es) 2002-01-18
PL357634A1 (en) 2004-07-26
HUP0203803A3 (en) 2004-09-28
SV2002000287A (es) 2002-01-08
HUP0203803A2 (hu) 2003-02-28
GT200100005A (es) 2002-02-05
TNSN01018A1 (en) 2005-11-10
IL150742A0 (en) 2003-02-12
CO5280216A1 (es) 2003-05-30

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