SI2875011T1 - Antagonisti receptorja 5-HT3 - Google Patents

Antagonisti receptorja 5-HT3 Download PDF

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Publication number
SI2875011T1
SI2875011T1 SI201330981T SI201330981T SI2875011T1 SI 2875011 T1 SI2875011 T1 SI 2875011T1 SI 201330981 T SI201330981 T SI 201330981T SI 201330981 T SI201330981 T SI 201330981T SI 2875011 T1 SI2875011 T1 SI 2875011T1
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Slovenia
Prior art keywords
receptor antagonists
compounds
receptor
compound
disorders
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SI201330981T
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English (en)
Inventor
Stephen Hitchcock
Holger Monenschein
Holly Reichard
Huikai Sun
Shota Kikuchi
Todd Macklin
Maria Hopkins
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Takeda Pharmaceutical Company Limited
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48877569&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI2875011(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical Company Limited filed Critical Takeda Pharmaceutical Company Limited
Publication of SI2875011T1 publication Critical patent/SI2875011T1/sl

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  • Chemical & Material Sciences (AREA)
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Claims (3)

  1. Antagonisti receptorja 5-HT3 Patentni zahtevki
    1. Spojina 1 -(1 -metil-1 H-pirazol-4-il)-N-(( 1 R,5S,7S)-9-metil-3-oksa-9-azabiciklo[3.3.1]-nonan-7-il)-lH-indol-3-karboksamid ali njena farmacevtsko sprejemljiva sol.
  2. 2. Farmacevtski sestavek, ki vsebuje spojino po zahtevku 1 in farmacevtsko sprejemljiv ekscipient.
  3. 3. Spojina po zahtevku 1 za uporabo kot zdravilo.
SI201330981T 2012-07-17 2013-07-16 Antagonisti receptorja 5-HT3 SI2875011T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201261672709P 2012-07-17 2012-07-17
US201261708521P 2012-10-01 2012-10-01
PCT/US2013/050746 WO2014014951A1 (en) 2012-07-17 2013-07-16 5-ht3 receptor antagonists
EP13742355.4A EP2875011B1 (en) 2012-07-17 2013-07-16 5-ht3 receptor antagonists

Publications (1)

Publication Number Publication Date
SI2875011T1 true SI2875011T1 (sl) 2018-06-29

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SI201330981T SI2875011T1 (sl) 2012-07-17 2013-07-16 Antagonisti receptorja 5-HT3

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US (8) US9303045B2 (sl)
EP (3) EP2875012B1 (sl)
JP (5) JP5816400B2 (sl)
KR (1) KR102148969B1 (sl)
CN (2) CN106478662B (sl)
AP (1) AP2015008240A0 (sl)
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AU (1) AU2013290375B2 (sl)
BR (1) BR112015001028B1 (sl)
CA (1) CA2879115C (sl)
CL (1) CL2015000121A1 (sl)
CO (1) CO7280468A2 (sl)
CR (1) CR20150057A (sl)
CY (1) CY1120881T1 (sl)
DK (2) DK2875011T3 (sl)
DO (1) DOP2015000009A (sl)
EA (1) EA025986B1 (sl)
EC (1) ECSP15004780A (sl)
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IL (1) IL236702B (sl)
IN (1) IN2015DN00957A (sl)
JO (1) JOP20130213B1 (sl)
LT (1) LT2875011T (sl)
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MX (1) MX359733B (sl)
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PE (1) PE20150671A1 (sl)
PH (1) PH12015500085A1 (sl)
PL (2) PL2875011T3 (sl)
PT (2) PT3312169T (sl)
RS (1) RS57096B1 (sl)
SG (1) SG11201500302UA (sl)
SI (1) SI2875011T1 (sl)
TN (1) TN2015000018A1 (sl)
TW (1) TWI602821B (sl)
UY (1) UY34912A (sl)
WO (2) WO2014014962A1 (sl)
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Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JOP20130213B1 (ar) * 2012-07-17 2021-08-17 Takeda Pharmaceuticals Co معارضات لمستقبلht3-5
CN106414439B (zh) * 2014-03-06 2017-12-08 上海海雁医药科技有限公司 作为食欲素受体拮抗剂的哌啶衍生物
HUE055175T2 (hu) * 2014-09-29 2021-11-29 Takeda Pharmaceuticals Co Az 1-(1-metil-1H-pirazol-4-il)-N-((1R,5S,7S)-9-metil-3-oxa-9-azabiciklo[3.3.1] nonan-7-il)-1H-indol-3-karboxamid kristályos formája
EP3623371A1 (en) 2014-12-16 2020-03-18 Axovant Sciences GmbH Geminal substituted quinuclidine amide compounds as agonists of alpha-7 nicotinic acetylcholine receptors
KR20180044256A (ko) 2015-06-10 2018-05-02 엑소반트 사이언시즈 게엠베하 A7-니코틴성 아세틸콜린 수용체의 작용제로서의 아미노벤즈이소옥사졸 화합물
JP2018523707A (ja) 2015-08-12 2018-08-23 アクソバント サイエンシズ ゲーエムベーハー α７−ニコチン性アセチルコリン受容体のアゴニストとしてのジェミナル置換アミノベンゾイソオキサゾール化合物
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