SI2193131T1 - Imidazo(1,2-A)pirazin spojine za zdravljenje virusnih okuĹľb kot je hepatitis - Google Patents

Imidazo(1,2-A)pirazin spojine za zdravljenje virusnih okuĹľb kot je hepatitis

Info

Publication number
SI2193131T1
SI2193131T1 SI200830948T SI200830948T SI2193131T1 SI 2193131 T1 SI2193131 T1 SI 2193131T1 SI 200830948 T SI200830948 T SI 200830948T SI 200830948 T SI200830948 T SI 200830948T SI 2193131 T1 SI2193131 T1 SI 2193131T1
Authority
SI
Slovenia
Prior art keywords
imidazos1
acpyrazine
hepatitis
compounds
treatment
Prior art date
Application number
SI200830948T
Other languages
English (en)
Inventor
Angus Macleod
Dale Robert Mitchell
Nicholas John Palmer
Christophe Claude Parsy
Michael Daniel Goldsmith
Clifford John Harris
Original Assignee
Biofocus Dpi Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biofocus Dpi Limited filed Critical Biofocus Dpi Limited
Publication of SI2193131T1 publication Critical patent/SI2193131T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI200830948T 2007-08-21 2008-08-20 Imidazo(1,2-A)pirazin spojine za zdravljenje virusnih okuĹľb kot je hepatitis SI2193131T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0716292.8A GB0716292D0 (en) 2007-08-21 2007-08-21 Imidazopyrazine compounds
PCT/EP2008/060896 WO2009024585A2 (en) 2007-08-21 2008-08-20 Imidazo [1,2-a] pyrazine compounds for treatment of viral infections such as hepatitis
EP08787346A EP2193131B1 (en) 2007-08-21 2008-08-20 Imidazo[1,2-a]pyrazine compounds for treatment of viral infections such as hepatitis

Publications (1)

Publication Number Publication Date
SI2193131T1 true SI2193131T1 (sl) 2013-06-28

Family

ID=38566736

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200830948T SI2193131T1 (sl) 2007-08-21 2008-08-20 Imidazo(1,2-A)pirazin spojine za zdravljenje virusnih okuĹľb kot je hepatitis

Country Status (21)

Country Link
US (1) US8362018B2 (sl)
EP (2) EP2193131B1 (sl)
JP (1) JP2010536825A (sl)
KR (1) KR20100081294A (sl)
CN (1) CN101835780B (sl)
AU (1) AU2008290531A1 (sl)
BR (1) BRPI0815717A2 (sl)
CA (1) CA2707521A1 (sl)
CY (1) CY1113872T1 (sl)
DK (1) DK2193131T3 (sl)
ES (1) ES2404415T3 (sl)
GB (1) GB0716292D0 (sl)
HK (1) HK1143810A1 (sl)
HR (1) HRP20130202T1 (sl)
MX (1) MX2010001733A (sl)
NZ (1) NZ584108A (sl)
PL (1) PL2193131T3 (sl)
PT (1) PT2193131E (sl)
SI (1) SI2193131T1 (sl)
WO (1) WO2009024585A2 (sl)
ZA (1) ZA201002009B (sl)

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JP5822944B2 (ja) * 2010-12-17 2015-11-25 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 過剰増殖性障害の治療におけるｍｐｓ−１およびｔｋｋ阻害剤として使用するための２置換イミダゾピラジン
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EP2651950A1 (en) 2010-12-17 2013-10-23 Bayer Intellectual Property GmbH 6 substituted imidazopyrazines for use as mps-1 and tkk inhibitors in the treatment of hyperproliferative disorders
JP5684406B2 (ja) 2010-12-23 2015-03-11 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｃｒ１受容体アンタゴニストとしてのピラゾロピペリジン化合物
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KR102171706B1 (ko) 2012-07-09 2020-10-30 얀센 파마슈티카 엔.브이. 포스포디에스테라아제 10 효소의 억제제
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TW201817714A (zh) 2016-08-30 2018-05-16 英商葛蘭素史密斯克藍智慧財產權有限公司 抑制3c及3cl蛋白酶之化合物及其使用方法
SI3697789T1 (sl) 2017-10-18 2022-04-29 Incyte Corporation Kondenzirani imidazolni derivati, substituirani s terciarnimi hidroksi skupinami, kot zaviralci PI3K-gama
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Also Published As

Publication number Publication date
CN101835780B (zh) 2013-09-18
WO2009024585A2 (en) 2009-02-26
ES2404415T3 (es) 2013-05-27
EP2567960A3 (en) 2013-06-05
KR20100081294A (ko) 2010-07-14
PL2193131T3 (pl) 2013-07-31
MX2010001733A (es) 2010-07-06
CN101835780A (zh) 2010-09-15
CY1113872T1 (el) 2016-07-27
EP2567960A2 (en) 2013-03-13
NZ584108A (en) 2012-06-29
JP2010536825A (ja) 2010-12-02
HRP20130202T1 (hr) 2013-04-30
HK1143810A1 (en) 2011-01-14
EP2193131B1 (en) 2013-01-30
ZA201002009B (en) 2010-12-29
GB0716292D0 (en) 2007-09-26
AU2008290531A1 (en) 2009-02-26
EP2193131A2 (en) 2010-06-09
BRPI0815717A2 (pt) 2015-02-10
PT2193131E (pt) 2013-04-04
US20110166147A1 (en) 2011-07-07
CA2707521A1 (en) 2009-02-26
DK2193131T3 (da) 2013-04-22
US8362018B2 (en) 2013-01-29
WO2009024585A3 (en) 2009-08-06

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