SE5292304T3 - - Google Patents

Info

Publication number
SE5292304T3
SE5292304T3 SE01930705T SE01930705T SE5292304T3 SE 5292304 T3 SE5292304 T3 SE 5292304T3 SE 01930705 T SE01930705 T SE 01930705T SE 01930705 T SE01930705 T SE 01930705T SE 5292304 T3 SE5292304 T3 SE 5292304T3
Authority
SE
Sweden
Prior art keywords
polymorphs
preparation
provides
present
zolpidem hemitartrate
Prior art date
Application number
SE01930705T
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27394001&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE5292304(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of SE5292304T3 publication Critical patent/SE5292304T3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Other Liquid Machine Or Engine Such As Wave Power Use (AREA)
  • Supply Devices, Intensifiers, Converters, And Telemotors (AREA)
  • Suspension Of Electric Lines Or Cables (AREA)
  • Amplifiers (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SE01930705T 2000-04-24 2001-04-24 SE5292304T3 (xx)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19929800P 2000-04-24 2000-04-24
US20602500P 2000-05-22 2000-05-22
US22536400P 2000-08-14 2000-08-14

Publications (1)

Publication Number Publication Date
SE5292304T3 true SE5292304T3 (xx) 2005-11-02

Family

ID=27394001

Family Applications (1)

Application Number Title Priority Date Filing Date
SE01930705T SE5292304T3 (xx) 2000-04-24 2001-04-24

Country Status (21)

Country Link
US (8) US20020077332A1 (xx)
EP (1) EP1292304B1 (xx)
JP (3) JP2003531173A (xx)
KR (1) KR20030069796A (xx)
AT (4) ATE338550T1 (xx)
AU (2) AU5721301A (xx)
CA (1) CA2406982A1 (xx)
CZ (1) CZ20023775A3 (xx)
DE (7) DE60122216T2 (xx)
DK (1) DK1292304T3 (xx)
ES (4) ES2248321T3 (xx)
HR (1) HRP20020909A2 (xx)
HU (1) HUP0300701A2 (xx)
IL (1) IL152411A0 (xx)
NZ (1) NZ522015A (xx)
PL (1) PL358548A1 (xx)
PT (3) PT1473036E (xx)
SE (1) SE5292304T3 (xx)
SK (1) SK16372002A3 (xx)
WO (1) WO2001080857A1 (xx)
YU (1) YU79402A (xx)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6921839B2 (en) 2000-08-29 2005-07-26 Ranbaxy Laboratories Limited Synthesis of N,N-dimethyl-3-(4-methyl) benzoyl propionamide a key intermediate of zolpidem
US6869970B2 (en) 2002-02-04 2005-03-22 Novartis Ag Crystalline salt forms of valsartan
CN100398539C (zh) 2002-12-18 2008-07-02 马林克罗特公司 杂芳基乙酰胺的合成
WO2004087703A1 (en) * 2003-03-12 2004-10-14 Sun Pharmaceutical Industries Limited Process for the preparation of n,n,6-trimethyl-2-(4-methylphenyl)-imidazo[1,2-a]pyridine-3-acetamide
EP1660496A1 (en) * 2003-07-31 2006-05-31 Ranbaxy Laboratories Limited Process for the synthesis of zolpidem
US7658945B2 (en) * 2004-02-17 2010-02-09 Transcept Pharmaceuticals, Inc. Compositions for delivering hypnotic agents across the oral mucosa and methods of use thereof
WO2006008636A2 (en) * 2004-07-16 2006-01-26 Ranbaxy Laboratories Limited Processes for the preparation of zolpidem and its hemitartrate
US20070287740A1 (en) * 2005-05-25 2007-12-13 Transcept Pharmaceuticals, Inc. Compositions and methods of treating middle-of-the night insomnia
US20070225322A1 (en) * 2005-05-25 2007-09-27 Transoral Pharmaceuticals, Inc. Compositions and methods for treating middle-of-the night insomnia
BRPI0609984A2 (pt) * 2005-05-25 2010-05-18 Transcept Pharmaceuticals Inc uso de zolpidem ou um sal do mesmo
RU2008110498A (ru) * 2005-08-19 2009-09-27 Авентис Фармасьютикалз Инк. (Us) Комбинация снотворного средства и замещенного соединения бис арила и гетероарила и ее терапевтическое применение
CN101247810A (zh) * 2005-08-19 2008-08-20 安万特药物公司 催眠药与R(+)-α-(2,3-二甲氧基-苯基)-1-[2-(4-氟苯基)乙基]-4-哌啶甲醇的组合及其治疗应用
AU2006297475A1 (en) * 2005-10-03 2007-04-12 Mallinckrodt Inc. Process for preparing zolpidem hemitartrate and tartrate polymorphs
WO2007047047A2 (en) * 2005-10-17 2007-04-26 Mallinckrodt Inc. Polymorph transformation of zolpidem in tablet matrix
US20070098788A1 (en) * 2005-10-28 2007-05-03 Gore Subhash P Non-benzodiazepine hypnotic compositions
TWI400234B (zh) 2006-03-31 2013-07-01 Janssen Pharmaceutica Nv 作為組織胺ｈ4受體調節劑之苯并咪唑-２-基嘧啶類及吡類
WO2008067549A2 (en) * 2006-11-30 2008-06-05 Transcept Pharmaceuticals, Inc. Stabilized zolpidem pharmaceutical compositions
US20080145425A1 (en) * 2006-12-15 2008-06-19 Pliva Research & Development Limited Pharmaceutical composition of zolpidem
US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
EA020090B1 (ru) * 2008-06-30 2014-08-29 Янссен Фармацевтика Нв Способ получения и рекристаллизации кристаллического гемитартрата бензоимидазол-2-илпиримидинового производного
BR112012012947B8 (pt) 2009-11-27 2021-05-25 Genzyme Corp sal de hemitartarato e composição farmacêutica compreendendo o mesmo
WO2011115069A1 (ja) * 2010-03-19 2011-09-22 第一三共株式会社 結晶の網羅的探索
PL2964229T3 (pl) 2013-03-06 2020-05-18 Janssen Pharmaceutica Nv Benzoimidazol-2-ilo pirymidynowe modulatory receptora histaminowego H<sub>4</sub>

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4151273A (en) * 1974-10-31 1979-04-24 The Regents Of The University Of California Increasing the absorption rate of insoluble drugs
FR2408345A1 (fr) * 1976-11-30 1979-06-08 Besins Jean Louis Nouvelle composition a action anti-conceptionnelle
US4302446A (en) * 1979-10-02 1981-11-24 Bristol-Myers Company Pharmaceutical compositions
IT1130924B (it) * 1980-03-06 1986-06-18 Secifarma Spa Procedimento per la preparazione di spironolattone micronizzato
DE3018940A1 (de) * 1980-05-17 1981-11-26 Hoechst Ag, 6000 Frankfurt Verwendung eines vinylchlorid-pfropf-copolymerisates in der plastisolverarbeitung
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
FR2525601A1 (fr) * 1982-04-21 1983-10-28 Synthelabo Derives d'imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
US4675323A (en) * 1985-08-06 1987-06-23 Synthelabo Imidazo(1,2-a)quinoline derivatives useful as anxiolytic agents
SE457326B (sv) * 1986-02-14 1988-12-19 Lejus Medical Ab Foerfarande foer framstaellning av en snabbt soenderfallande kaerna innehaallande bl a mikrokristallin cellulosa
FR2600650B1 (fr) * 1986-06-27 1988-09-09 Synthelabo Procede de preparation d'imidazopyridines et composes intermediaires
FR2606410B1 (fr) * 1986-11-07 1989-02-24 Synthelabo Imidazopyridines, leur preparation et leur application en therapeutique
ES2026666T3 (es) * 1987-03-27 1992-05-01 Synthelabo Procedimiento para preparar derivados de imidazopiridinas.
US5271944A (en) * 1991-04-05 1993-12-21 Biofor, Ltd. Pharmacologically enhanced formulations
IT1276522B1 (it) * 1995-04-07 1997-10-31 Elena Benincasa Uso dello zolpidem per il trattamento terapeudico di sindromi neuropsichiatriche associate a disfunsione e di circuiti neurali dei
DK1163241T3 (da) * 1999-03-25 2005-10-10 Synthon Bv Zolpidemsalte
DE69908546T2 (de) * 1999-03-25 2004-04-29 Synthon B.V. Imidazopyridinderivate und Verfahren zu ihrer Herstellung
AU6474200A (en) * 1999-12-13 2001-06-18 Sumika Fine Chemicals Co., Ltd. Process for the preparation of a pyridinemethanol compound

Also Published As

Publication number Publication date
DK1292304T3 (da) 2005-12-19
DE60122944T2 (de) 2007-04-12
EP1292304A1 (en) 2003-03-19
WO2001080857A1 (en) 2001-11-01
HRP20020909A2 (en) 2004-08-31
DE60122216T2 (de) 2007-08-30
US20040214859A1 (en) 2004-10-28
ATE308324T1 (de) 2005-11-15
US20020077332A1 (en) 2002-06-20
ES2239558T1 (es) 2005-10-01
JP2003531173A (ja) 2003-10-21
US20040220210A1 (en) 2004-11-04
DE04010435T1 (de) 2005-09-01
PT1473036E (pt) 2006-10-31
WO2001080857A9 (en) 2002-06-27
NZ522015A (en) 2004-08-27
US20040220213A1 (en) 2004-11-04
US20040220212A1 (en) 2004-11-04
ES2248321T3 (es) 2006-03-16
YU79402A (sh) 2006-03-03
EP1292304B1 (en) 2005-11-02
KR20030069796A (ko) 2003-08-27
ES2238941T1 (es) 2005-09-16
CZ20023775A3 (cs) 2003-10-15
SK16372002A3 (sk) 2003-04-01
ES2238941T3 (es) 2007-04-01
EP1292304A4 (en) 2003-07-23
DE60122216D1 (de) 2006-09-21
DE60122944D1 (de) 2006-10-19
DE04010651T1 (de) 2005-09-01
ATE335481T1 (de) 2006-09-15
PT1541146E (pt) 2007-01-31
ATE338550T1 (de) 2006-09-15
DE60125429D1 (de) 2007-02-01
DE20122435U1 (de) 2005-10-06
JP2006249105A (ja) 2006-09-21
CA2406982A1 (en) 2001-11-01
IL152411A0 (en) 2003-05-29
DE60114617T2 (de) 2006-07-27
AU5721301A (en) 2001-11-07
ES2277301T3 (es) 2007-07-01
JP2006137778A (ja) 2006-06-01
PL358548A1 (en) 2004-08-09
ATE348613T1 (de) 2007-01-15
DE60114617D1 (de) 2005-12-08
AU2001257213B2 (en) 2005-09-29
ES2239558T3 (es) 2007-04-01
US20040220211A1 (en) 2004-11-04
DE60125429T2 (de) 2007-09-27
HUP0300701A2 (hu) 2003-07-28
PT1475093E (pt) 2006-11-30
US20070037843A1 (en) 2007-02-15
US20040214858A1 (en) 2004-10-28

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