RS53176B - Inhibitori kinaze 1 koja reguliše signale u apoptozi - Google Patents

Inhibitori kinaze 1 koja reguliše signale u apoptozi

Info

Publication number
RS53176B
RS53176B RS20140066A RSP20140066A RS53176B RS 53176 B RS53176 B RS 53176B RS 20140066 A RS20140066 A RS 20140066A RS P20140066 A RSP20140066 A RS P20140066A RS 53176 B RS53176 B RS 53176B
Authority
RS
Serbia
Prior art keywords
alkyl
pyrrolo
hydroxy
group
hetero
Prior art date
Application number
RS20140066A
Other languages
English (en)
Serbian (sr)
Inventor
Edcon Chang
Original Assignee
Takeda Pharmaceutical Company Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical Company Limited filed Critical Takeda Pharmaceutical Company Limited
Publication of RS53176B publication Critical patent/RS53176B/sr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • AHUMAN NECESSITIES
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    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • A61P9/12Antihypertensives

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Communicable Diseases (AREA)
RS20140066A 2010-02-03 2011-01-21 Inhibitori kinaze 1 koja reguliše signale u apoptozi RS53176B (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30086910P 2010-02-03 2010-02-03
PCT/US2011/022137 WO2011097079A1 (en) 2010-02-03 2011-01-21 Apoptosis signal-regulating kinase 1 inhibitors

Publications (1)

Publication Number Publication Date
RS53176B true RS53176B (sr) 2014-06-30

Family

ID=43645892

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20140066A RS53176B (sr) 2010-02-03 2011-01-21 Inhibitori kinaze 1 koja reguliše signale u apoptozi

Country Status (14)

Country Link
US (2) US8802695B2 (https=)
EP (1) EP2531501B1 (https=)
JP (1) JP5711270B2 (https=)
CN (1) CN102834393B (https=)
CA (1) CA2787360C (https=)
DK (1) DK2531501T3 (https=)
ES (1) ES2445917T3 (https=)
HR (1) HRP20140114T1 (https=)
PL (1) PL2531501T3 (https=)
PT (1) PT2531501E (https=)
RS (1) RS53176B (https=)
SI (1) SI2531501T1 (https=)
SM (1) SMT201400012B (https=)
WO (1) WO2011097079A1 (https=)

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CN110770233B (zh) * 2017-06-19 2022-07-26 广东东阳光药业有限公司 稠合双环类化合物及其在药物中的应用
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US9403819B2 (en) 2016-08-02
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US20120316194A1 (en) 2012-12-13
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EP2531501A1 (en) 2012-12-12
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