RS49520B - Antimikrobno aktivne smeše - Google Patents

Antimikrobno aktivne smeše

Info

Publication number
RS49520B
RS49520B YU41796A YU41796A RS49520B RS 49520 B RS49520 B RS 49520B YU 41796 A YU41796 A YU 41796A YU 41796 A YU41796 A YU 41796A RS 49520 B RS49520 B RS 49520B
Authority
RS
Serbia
Prior art keywords
amino
carboxylic acid
active mixtures
antimicrobially active
methylenecyclopentane
Prior art date
Application number
YU41796A
Other languages
English (en)
Inventor
Dr. Michael Matzke
Dr. Hans-Christian MILITZER
Dr. Joachim Mittendorf
Dr. Franz Kunisch
Dr. Axel SCHMIDT
Dr. Wolfgang Schonfeld
Dr. Karl ZIEGELBAUER
Original Assignee
Bayer Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag. filed Critical Bayer Ag.
Publication of YU41796A publication Critical patent/YU41796A/sh
Publication of RS49520B publication Critical patent/RS49520B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05—Dipeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Abstract

Antimikrobno aktivne smeše, koje sadrže α-amino kiseline i ciklopentan--amino kiseline iz grupe koju sačinjavaju "(S)-izoleucin sa 2-amino-4-metilenciklopentan-1-karbonskom kiselinom, (S)-alanin sa 2-amino-4-metilenciklopentan-1-karbonskom kiselinom, (S)-prolin sa 1,2-cis-amino-ciklopentan-1-karbonskom kiselinom" ili njihove izomerne oblike i, u datom slučaju, jedan ili više farmaceutski prihvatljivih ekscipijenata. Prijava sadrži još 3 zavisna patentna zahteva.
YU41796A 1995-07-19 1996-07-12 Antimikrobno aktivne smeše RS49520B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19526274A DE19526274A1 (de) 1995-07-19 1995-07-19 Verbesserung der Verträglichkeit von pharmazeutisch wirksamen beta-Aminosäuren

Publications (2)

Publication Number Publication Date
YU41796A YU41796A (sh) 1999-06-15
RS49520B true RS49520B (sr) 2006-10-27

Family

ID=7767189

Family Applications (1)

Application Number Title Priority Date Filing Date
YU41796A RS49520B (sr) 1995-07-19 1996-07-12 Antimikrobno aktivne smeše

Country Status (45)

Country Link
US (1) US5935988A (sr)
EP (2) EP0754678B1 (sr)
JP (2) JP3891503B2 (sr)
KR (1) KR100433968B1 (sr)
CN (1) CN1115145C (sr)
AR (1) AR003465A1 (sr)
AT (2) ATE344274T1 (sr)
AU (1) AU713555B2 (sr)
BG (1) BG62134B1 (sr)
BR (1) BR9603124A (sr)
CA (1) CA2181308A1 (sr)
CO (1) CO4700525A1 (sr)
CU (1) CU22820A3 (sr)
CZ (2) CZ287896B6 (sr)
DE (3) DE19526274A1 (sr)
DK (2) DK1043332T3 (sr)
DZ (1) DZ2073A1 (sr)
EE (1) EE03803B1 (sr)
ES (2) ES2154761T3 (sr)
GR (1) GR3035601T3 (sr)
HK (1) HK1005131A1 (sr)
HR (1) HRP960303B1 (sr)
HU (1) HUP9601977A3 (sr)
IL (1) IL118869A (sr)
MA (1) MA23940A1 (sr)
MX (1) MX9602836A (sr)
NO (1) NO315926B1 (sr)
NZ (1) NZ299008A (sr)
PE (1) PE9398A1 (sr)
PL (1) PL184861B1 (sr)
PT (2) PT754678E (sr)
RO (1) RO118656B1 (sr)
RS (1) RS49520B (sr)
RU (1) RU2181123C2 (sr)
SA (1) SA96170491B1 (sr)
SG (1) SG47158A1 (sr)
SI (2) SI0754678T1 (sr)
SK (2) SK281850B6 (sr)
SV (1) SV1996000062A (sr)
TN (1) TNSN96100A1 (sr)
TR (1) TR199600583A2 (sr)
TW (1) TW496737B (sr)
UA (1) UA46725C2 (sr)
YU (1) YU20050685A (sr)
ZA (1) ZA966111B (sr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6191306B1 (en) * 1999-08-03 2001-02-20 Eastman Chemical Company Process for the preparation of cyclopropylglycine
KR20010073441A (ko) * 2000-01-14 2001-08-01 최인도 패류종묘 착상판의 제조방법
US8394813B2 (en) 2000-11-14 2013-03-12 Shire Llc Active agent delivery systems and methods for protecting and administering active agents
US20060014697A1 (en) 2001-08-22 2006-01-19 Travis Mickle Pharmaceutical compositions for prevention of overdose or abuse
US7169752B2 (en) 2003-09-30 2007-01-30 New River Pharmaceuticals Inc. Compounds and compositions for prevention of overdose of oxycodone
US7105486B2 (en) * 2002-02-22 2006-09-12 New River Pharmaceuticals Inc. Abuse-resistant amphetamine compounds
US7659253B2 (en) * 2002-02-22 2010-02-09 Shire Llc Abuse-resistant amphetamine prodrugs
US7700561B2 (en) * 2002-02-22 2010-04-20 Shire Llc Abuse-resistant amphetamine prodrugs
SI1644019T2 (en) 2003-05-29 2018-04-30 Shire Llc AMPHETAMINE COMPOUNDS COMPOUNDS TO ABUSE

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8716278D0 (en) * 1987-07-10 1987-08-19 Fujisawa Pharmaceutical Co Antimicrobial agent
JPH02174753A (ja) * 1988-08-25 1990-07-06 Fujisawa Pharmaceut Co Ltd シス―２―アミノシクロペンタンカルボン酸誘導体およびその製法ならびに抗菌剤
AU673824B2 (en) * 1992-05-29 1996-11-28 Bayer Aktiengesellschaft Cyclopentane- and -pentene-beta-amino acids
US5631291A (en) * 1992-05-29 1997-05-20 Bayer Aktiengesellschaft Cyclopentane- and -pentene-β-amino acids
DE4302155A1 (de) * 1993-01-27 1994-07-28 Bayer Ag Verwendung von Cyclopentan- und -penten-beta-Aminosäuren
GB9216441D0 (en) * 1992-08-03 1992-09-16 Ici Plc Fungicidal process
WO1995007022A1 (en) * 1993-09-07 1995-03-16 Zeneca Limited Fungicides
DE19548825C2 (de) * 1995-12-27 1999-03-25 Rolf Dr Hermann Neue, substituierte Cyclopentylaminderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE19604225A1 (de) * 1996-02-06 1997-08-07 Bayer Ag Stoffzusammensetzungen aus alpha-Aminosäuren und Cyclohexen-beta-aminosäuren

Also Published As

Publication number Publication date
AU5948896A (en) 1997-01-23
HK1005131A1 (en) 1998-12-24
HRP960303B1 (en) 2001-08-31
CN1143496A (zh) 1997-02-26
GR3035601T3 (en) 2001-06-29
DZ2073A1 (fr) 2002-07-22
CN1115145C (zh) 2003-07-23
NZ299008A (en) 1998-05-27
CZ288204B6 (en) 2001-05-16
EP1043332A1 (de) 2000-10-11
DK0754678T3 (da) 2001-02-05
HUP9601977A2 (en) 1997-05-28
EE03803B1 (et) 2002-08-15
KR970006312A (ko) 1997-02-19
JP2007056026A (ja) 2007-03-08
YU20050685A (sh) 2006-08-17
IL118869A0 (en) 1996-10-31
SK281850B6 (sk) 2001-08-06
NO963000D0 (no) 1996-07-18
ATE344274T1 (de) 2006-11-15
JPH09202761A (ja) 1997-08-05
EP0754678B1 (de) 2001-01-03
EP0754678A2 (de) 1997-01-22
SV1996000062A (es) 1997-06-26
SK94796A3 (en) 1997-02-05
EP1043332B1 (de) 2006-11-02
ATE198469T1 (de) 2001-01-15
PT754678E (pt) 2001-04-30
NO315926B1 (no) 2003-11-17
KR100433968B1 (ko) 2004-08-30
SA96170491B1 (ar) 2006-09-20
CA2181308A1 (en) 1997-01-20
PE9398A1 (es) 1998-04-15
TR199600583A2 (tr) 1997-02-21
TW496737B (en) 2002-08-01
ZA966111B (en) 1997-02-03
UA46725C2 (uk) 2002-06-17
CO4700525A1 (es) 1998-12-29
MA23940A1 (fr) 1997-04-01
BG62134B1 (bg) 1999-03-31
EE9600109A (et) 1997-02-17
PT1043332E (pt) 2007-01-31
BG100716A (bg) 1997-04-30
PL184861B1 (pl) 2003-01-31
CU22820A3 (es) 2003-01-29
CZ214396A3 (en) 1997-02-12
JP3891503B2 (ja) 2007-03-14
HUP9601977A3 (en) 1998-04-28
DE59611398D1 (de) 2006-12-14
DE19526274A1 (de) 1997-01-23
SG47158A1 (en) 1998-03-20
RU2181123C2 (ru) 2002-04-10
PL315330A1 (en) 1997-01-20
RO118656B1 (ro) 2003-08-29
DK1043332T3 (da) 2007-03-12
AR003465A1 (es) 1998-08-05
ES2275460T3 (es) 2007-06-16
EP0754678A3 (de) 1997-12-17
HRP960303A2 (en) 1998-02-28
SI1043332T1 (sl) 2007-04-30
BR9603124A (pt) 1998-04-22
SK284733B6 (sk) 2005-10-06
ES2154761T3 (es) 2001-04-16
HU9601977D0 (en) 1996-09-30
SI0754678T1 (en) 2001-04-30
TNSN96100A1 (fr) 2005-03-15
DE59606266D1 (de) 2001-02-08
AU713555B2 (en) 1999-12-02
IL118869A (en) 2002-03-10
YU41796A (sh) 1999-06-15
MX9602836A (es) 1997-01-31
CZ287896B6 (cs) 2001-03-14
US5935988A (en) 1999-08-10
NO963000L (no) 1997-01-20

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