ES2154761T3 - Mejora de la tolerancia de beta-aminoacidos farmaceuticamente activos. - Google Patents
Mejora de la tolerancia de beta-aminoacidos farmaceuticamente activos.Info
- Publication number
- ES2154761T3 ES2154761T3 ES96110967T ES96110967T ES2154761T3 ES 2154761 T3 ES2154761 T3 ES 2154761T3 ES 96110967 T ES96110967 T ES 96110967T ES 96110967 T ES96110967 T ES 96110967T ES 2154761 T3 ES2154761 T3 ES 2154761T3
- Authority
- ES
- Spain
- Prior art keywords
- aminoacidos
- beta
- improvement
- pharmaceutically active
- cyclopentane
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
- C07C237/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
- C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Gastroenterology & Hepatology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Communicable Diseases (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pyrrole Compounds (AREA)
Abstract
LA PRESENTE INVENCION TRATA DE MEZCLAS DE AL -AMINOACIDOS Y/O SUS DERIVADOS, Y CICLOPENTANO-{BE}-AMINOACIDOS Y/O SUS DERIVADOS, DIPEPTIDOS DE LOS {AL}-AMINOACIDOS Y CICLOPENTANO-{BE}AMINOACIDOS ANTES CITADOS, Y MEZCLAS DE LAS MEZCLAS Y DIPEPTIDOS ANTES CITADOS, QUE EN COMPARACION CON LOS CICLOPENTANO-{BE}AMINOACIDOS PUROS TIENEN UNA MEJOR ACEPTACION POR LOS ANIMALES DE SANGRE CALIENTE.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19526274A DE19526274A1 (de) | 1995-07-19 | 1995-07-19 | Verbesserung der Verträglichkeit von pharmazeutisch wirksamen beta-Aminosäuren |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2154761T3 true ES2154761T3 (es) | 2001-04-16 |
Family
ID=7767189
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES00110958T Expired - Lifetime ES2275460T3 (es) | 1995-07-19 | 1996-07-08 | Dipeptidos que contienen ciclopentano-beta-aminoacidos. |
ES96110967T Expired - Lifetime ES2154761T3 (es) | 1995-07-19 | 1996-07-08 | Mejora de la tolerancia de beta-aminoacidos farmaceuticamente activos. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES00110958T Expired - Lifetime ES2275460T3 (es) | 1995-07-19 | 1996-07-08 | Dipeptidos que contienen ciclopentano-beta-aminoacidos. |
Country Status (45)
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6191306B1 (en) * | 1999-08-03 | 2001-02-20 | Eastman Chemical Company | Process for the preparation of cyclopropylglycine |
KR20010073441A (ko) * | 2000-01-14 | 2001-08-01 | 최인도 | 패류종묘 착상판의 제조방법 |
US8394813B2 (en) | 2000-11-14 | 2013-03-12 | Shire Llc | Active agent delivery systems and methods for protecting and administering active agents |
US20060014697A1 (en) | 2001-08-22 | 2006-01-19 | Travis Mickle | Pharmaceutical compositions for prevention of overdose or abuse |
US7169752B2 (en) | 2003-09-30 | 2007-01-30 | New River Pharmaceuticals Inc. | Compounds and compositions for prevention of overdose of oxycodone |
US7659253B2 (en) * | 2002-02-22 | 2010-02-09 | Shire Llc | Abuse-resistant amphetamine prodrugs |
US7105486B2 (en) * | 2002-02-22 | 2006-09-12 | New River Pharmaceuticals Inc. | Abuse-resistant amphetamine compounds |
US7700561B2 (en) * | 2002-02-22 | 2010-04-20 | Shire Llc | Abuse-resistant amphetamine prodrugs |
KR101159477B1 (ko) * | 2003-05-29 | 2012-07-02 | 샤이어 엘엘씨 | 남용 방지성 암페타민 화합물 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8716278D0 (en) * | 1987-07-10 | 1987-08-19 | Fujisawa Pharmaceutical Co | Antimicrobial agent |
JPH02174753A (ja) * | 1988-08-25 | 1990-07-06 | Fujisawa Pharmaceut Co Ltd | シス―2―アミノシクロペンタンカルボン酸誘導体およびその製法ならびに抗菌剤 |
DE4302155A1 (de) * | 1993-01-27 | 1994-07-28 | Bayer Ag | Verwendung von Cyclopentan- und -penten-beta-Aminosäuren |
AU673824B2 (en) * | 1992-05-29 | 1996-11-28 | Bayer Aktiengesellschaft | Cyclopentane- and -pentene-beta-amino acids |
US5631291A (en) * | 1992-05-29 | 1997-05-20 | Bayer Aktiengesellschaft | Cyclopentane- and -pentene-β-amino acids |
GB9216441D0 (en) * | 1992-08-03 | 1992-09-16 | Ici Plc | Fungicidal process |
WO1995007022A1 (en) * | 1993-09-07 | 1995-03-16 | Zeneca Limited | Fungicides |
DE19548825C2 (de) * | 1995-12-27 | 1999-03-25 | Rolf Dr Hermann | Neue, substituierte Cyclopentylaminderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
DE19604225A1 (de) * | 1996-02-06 | 1997-08-07 | Bayer Ag | Stoffzusammensetzungen aus alpha-Aminosäuren und Cyclohexen-beta-aminosäuren |
-
1995
- 1995-07-19 DE DE19526274A patent/DE19526274A1/de not_active Withdrawn
-
1996
- 1996-06-28 HR HR960303A patent/HRP960303B1/xx not_active IP Right Cessation
- 1996-07-08 SI SI9630749T patent/SI1043332T1/sl unknown
- 1996-07-08 EP EP00110958A patent/EP1043332B1/de not_active Expired - Lifetime
- 1996-07-08 DK DK96110967T patent/DK0754678T3/da active
- 1996-07-08 PT PT96110967T patent/PT754678E/pt unknown
- 1996-07-08 DE DE59611398T patent/DE59611398D1/de not_active Expired - Fee Related
- 1996-07-08 EP EP96110967A patent/EP0754678B1/de not_active Expired - Lifetime
- 1996-07-08 PT PT00110958T patent/PT1043332E/pt unknown
- 1996-07-08 DE DE59606266T patent/DE59606266D1/de not_active Expired - Fee Related
- 1996-07-08 AT AT96110967T patent/ATE198469T1/de not_active IP Right Cessation
- 1996-07-08 ES ES00110958T patent/ES2275460T3/es not_active Expired - Lifetime
- 1996-07-08 ES ES96110967T patent/ES2154761T3/es not_active Expired - Lifetime
- 1996-07-08 DK DK00110958T patent/DK1043332T3/da active
- 1996-07-08 SI SI9630243T patent/SI0754678T1/xx unknown
- 1996-07-08 AT AT00110958T patent/ATE344274T1/de not_active IP Right Cessation
- 1996-07-12 CU CU1996063A patent/CU22820A3/es unknown
- 1996-07-12 US US08/679,027 patent/US5935988A/en not_active Expired - Fee Related
- 1996-07-12 YU YU20050685A patent/YU20050685A/sh unknown
- 1996-07-12 RS YU41796A patent/RS49520B/sr unknown
- 1996-07-12 AU AU59488/96A patent/AU713555B2/en not_active Ceased
- 1996-07-16 NZ NZ299008A patent/NZ299008A/en unknown
- 1996-07-16 TR TR96/00583A patent/TR199600583A2/xx unknown
- 1996-07-16 CA CA002181308A patent/CA2181308A1/en not_active Abandoned
- 1996-07-16 RO RO96-01451A patent/RO118656B1/ro unknown
- 1996-07-16 MA MA24315A patent/MA23940A1/fr unknown
- 1996-07-16 TW TW085108582A patent/TW496737B/zh not_active IP Right Cessation
- 1996-07-16 IL IL11886996A patent/IL118869A/en not_active IP Right Cessation
- 1996-07-17 SG SG1996010277A patent/SG47158A1/en unknown
- 1996-07-17 BG BG100716A patent/BG62134B1/bg unknown
- 1996-07-17 DZ DZ960117A patent/DZ2073A1/fr active
- 1996-07-17 UA UA96072884A patent/UA46725C2/uk unknown
- 1996-07-18 ZA ZA9606111A patent/ZA966111B/xx unknown
- 1996-07-18 EE EE9600109A patent/EE03803B1/xx not_active IP Right Cessation
- 1996-07-18 CO CO96037937A patent/CO4700525A1/es unknown
- 1996-07-18 MX MX9602836A patent/MX9602836A/es not_active IP Right Cessation
- 1996-07-18 NO NO19963000A patent/NO315926B1/no unknown
- 1996-07-18 PE PE1996000543A patent/PE9398A1/es not_active Application Discontinuation
- 1996-07-18 KR KR1019960028961A patent/KR100433968B1/ko not_active IP Right Cessation
- 1996-07-18 SK SK947-96A patent/SK281850B6/sk unknown
- 1996-07-18 TN TNTNSN96100A patent/TNSN96100A1/fr unknown
- 1996-07-18 CZ CZ19962143A patent/CZ287896B6/cs not_active IP Right Cessation
- 1996-07-18 PL PL96315330A patent/PL184861B1/pl not_active IP Right Cessation
- 1996-07-18 BR BR9603124A patent/BR9603124A/pt active Search and Examination
- 1996-07-18 JP JP20641096A patent/JP3891503B2/ja not_active Expired - Fee Related
- 1996-07-18 SK SK1421-2000A patent/SK284733B6/sk unknown
- 1996-07-19 CN CN96108880A patent/CN1115145C/zh not_active Expired - Fee Related
- 1996-07-19 SV SV1996000062A patent/SV1996000062A/es not_active Application Discontinuation
- 1996-07-19 AR ARP960103667A patent/AR003465A1/es unknown
- 1996-07-19 RU RU96115341/04A patent/RU2181123C2/ru not_active IP Right Cessation
- 1996-07-19 HU HU9601977A patent/HUP9601977A3/hu unknown
- 1996-12-11 SA SA96170491A patent/SA96170491B1/ar unknown
-
1998
- 1998-05-18 HK HK98104267A patent/HK1005131A1/xx not_active IP Right Cessation
-
2000
- 2000-07-10 CZ CZ20002554A patent/CZ288204B6/cs not_active IP Right Cessation
-
2001
- 2001-03-20 GR GR20010400447T patent/GR3035601T3/el not_active IP Right Cessation
-
2006
- 2006-09-27 JP JP2006263475A patent/JP2007056026A/ja active Pending
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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