BR9603124A - Dipeptídeo processo para preparação do mesmo mistura e medicamentos - Google Patents

Dipeptídeo processo para preparação do mesmo mistura e medicamentos

Info

Publication number
BR9603124A
BR9603124A BR9603124A BR9603124A BR9603124A BR 9603124 A BR9603124 A BR 9603124A BR 9603124 A BR9603124 A BR 9603124A BR 9603124 A BR9603124 A BR 9603124A BR 9603124 A BR9603124 A BR 9603124A
Authority
BR
Brazil
Prior art keywords
dipeptide
drugs
preparing
same mixture
mixture
Prior art date
Application number
BR9603124A
Other languages
English (en)
Inventor
Wolfgang Schoenfeld
Karl Ziegelbauer
Axel Schmidt
Hans-Christian Militzer
Michael Matzke
Joachim Mittendorf
Franz Kunisch
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of BR9603124A publication Critical patent/BR9603124A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyrrole Compounds (AREA)
BR9603124A 1995-07-19 1996-07-18 Dipeptídeo processo para preparação do mesmo mistura e medicamentos BR9603124A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19526274A DE19526274A1 (de) 1995-07-19 1995-07-19 Verbesserung der Verträglichkeit von pharmazeutisch wirksamen beta-Aminosäuren

Publications (1)

Publication Number Publication Date
BR9603124A true BR9603124A (pt) 1998-04-22

Family

ID=7767189

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9603124A BR9603124A (pt) 1995-07-19 1996-07-18 Dipeptídeo processo para preparação do mesmo mistura e medicamentos

Country Status (45)

Country Link
US (1) US5935988A (pt)
EP (2) EP0754678B1 (pt)
JP (2) JP3891503B2 (pt)
KR (1) KR100433968B1 (pt)
CN (1) CN1115145C (pt)
AR (1) AR003465A1 (pt)
AT (2) ATE344274T1 (pt)
AU (1) AU713555B2 (pt)
BG (1) BG62134B1 (pt)
BR (1) BR9603124A (pt)
CA (1) CA2181308A1 (pt)
CO (1) CO4700525A1 (pt)
CU (1) CU22820A3 (pt)
CZ (2) CZ287896B6 (pt)
DE (3) DE19526274A1 (pt)
DK (2) DK1043332T3 (pt)
DZ (1) DZ2073A1 (pt)
EE (1) EE03803B1 (pt)
ES (2) ES2275460T3 (pt)
GR (1) GR3035601T3 (pt)
HK (1) HK1005131A1 (pt)
HR (1) HRP960303B1 (pt)
HU (1) HUP9601977A3 (pt)
IL (1) IL118869A (pt)
MA (1) MA23940A1 (pt)
MX (1) MX9602836A (pt)
NO (1) NO315926B1 (pt)
NZ (1) NZ299008A (pt)
PE (1) PE9398A1 (pt)
PL (1) PL184861B1 (pt)
PT (2) PT1043332E (pt)
RO (1) RO118656B1 (pt)
RS (1) RS49520B (pt)
RU (1) RU2181123C2 (pt)
SA (1) SA96170491B1 (pt)
SG (1) SG47158A1 (pt)
SI (2) SI0754678T1 (pt)
SK (2) SK284733B6 (pt)
SV (1) SV1996000062A (pt)
TN (1) TNSN96100A1 (pt)
TR (1) TR199600583A2 (pt)
TW (1) TW496737B (pt)
UA (1) UA46725C2 (pt)
YU (1) YU20050685A (pt)
ZA (1) ZA966111B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6191306B1 (en) * 1999-08-03 2001-02-20 Eastman Chemical Company Process for the preparation of cyclopropylglycine
KR20010073441A (ko) * 2000-01-14 2001-08-01 최인도 패류종묘 착상판의 제조방법
US8394813B2 (en) 2000-11-14 2013-03-12 Shire Llc Active agent delivery systems and methods for protecting and administering active agents
US20060014697A1 (en) 2001-08-22 2006-01-19 Travis Mickle Pharmaceutical compositions for prevention of overdose or abuse
US7169752B2 (en) 2003-09-30 2007-01-30 New River Pharmaceuticals Inc. Compounds and compositions for prevention of overdose of oxycodone
US7659253B2 (en) * 2002-02-22 2010-02-09 Shire Llc Abuse-resistant amphetamine prodrugs
US7105486B2 (en) * 2002-02-22 2006-09-12 New River Pharmaceuticals Inc. Abuse-resistant amphetamine compounds
US7700561B2 (en) * 2002-02-22 2010-04-20 Shire Llc Abuse-resistant amphetamine prodrugs
PT1644019E (pt) * 2003-05-29 2012-05-23 Shire Llc Compostos de anfetamina resistentes ao abuso

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8716278D0 (en) * 1987-07-10 1987-08-19 Fujisawa Pharmaceutical Co Antimicrobial agent
JPH02174753A (ja) * 1988-08-25 1990-07-06 Fujisawa Pharmaceut Co Ltd シス―2―アミノシクロペンタンカルボン酸誘導体およびその製法ならびに抗菌剤
DE4302155A1 (de) * 1993-01-27 1994-07-28 Bayer Ag Verwendung von Cyclopentan- und -penten-beta-Aminosäuren
US5631291A (en) * 1992-05-29 1997-05-20 Bayer Aktiengesellschaft Cyclopentane- and -pentene-β-amino acids
AU673824B2 (en) * 1992-05-29 1996-11-28 Bayer Aktiengesellschaft Cyclopentane- and -pentene-beta-amino acids
GB9216441D0 (en) * 1992-08-03 1992-09-16 Ici Plc Fungicidal process
WO1995007022A1 (en) * 1993-09-07 1995-03-16 Zeneca Limited Fungicides
DE19548825C2 (de) * 1995-12-27 1999-03-25 Rolf Dr Hermann Neue, substituierte Cyclopentylaminderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE19604225A1 (de) * 1996-02-06 1997-08-07 Bayer Ag Stoffzusammensetzungen aus alpha-Aminosäuren und Cyclohexen-beta-aminosäuren

Also Published As

Publication number Publication date
CN1115145C (zh) 2003-07-23
JPH09202761A (ja) 1997-08-05
EE03803B1 (et) 2002-08-15
ES2154761T3 (es) 2001-04-16
AU5948896A (en) 1997-01-23
MA23940A1 (fr) 1997-04-01
NO963000L (no) 1997-01-20
RU2181123C2 (ru) 2002-04-10
YU20050685A (sh) 2006-08-17
RO118656B1 (ro) 2003-08-29
CZ287896B6 (cs) 2001-03-14
TW496737B (en) 2002-08-01
US5935988A (en) 1999-08-10
IL118869A (en) 2002-03-10
GR3035601T3 (en) 2001-06-29
YU41796A (sh) 1999-06-15
SI1043332T1 (sl) 2007-04-30
MX9602836A (es) 1997-01-31
UA46725C2 (uk) 2002-06-17
TNSN96100A1 (fr) 2005-03-15
DZ2073A1 (fr) 2002-07-22
TR199600583A2 (tr) 1997-02-21
SK284733B6 (sk) 2005-10-06
EP1043332A1 (de) 2000-10-11
PL315330A1 (en) 1997-01-20
CA2181308A1 (en) 1997-01-20
CU22820A3 (es) 2003-01-29
DK0754678T3 (da) 2001-02-05
HUP9601977A2 (en) 1997-05-28
JP2007056026A (ja) 2007-03-08
AR003465A1 (es) 1998-08-05
CZ288204B6 (en) 2001-05-16
IL118869A0 (en) 1996-10-31
NO963000D0 (no) 1996-07-18
SA96170491B1 (ar) 2006-09-20
EE9600109A (et) 1997-02-17
JP3891503B2 (ja) 2007-03-14
ZA966111B (en) 1997-02-03
NO315926B1 (no) 2003-11-17
DK1043332T3 (da) 2007-03-12
EP1043332B1 (de) 2006-11-02
HRP960303B1 (en) 2001-08-31
DE59611398D1 (de) 2006-12-14
PL184861B1 (pl) 2003-01-31
SK281850B6 (sk) 2001-08-06
ATE344274T1 (de) 2006-11-15
EP0754678B1 (de) 2001-01-03
PT1043332E (pt) 2007-01-31
RS49520B (sr) 2006-10-27
KR970006312A (ko) 1997-02-19
PE9398A1 (es) 1998-04-15
EP0754678A3 (de) 1997-12-17
DE59606266D1 (de) 2001-02-08
PT754678E (pt) 2001-04-30
HRP960303A2 (en) 1998-02-28
SK94796A3 (en) 1997-02-05
CO4700525A1 (es) 1998-12-29
ATE198469T1 (de) 2001-01-15
SG47158A1 (en) 1998-03-20
HK1005131A1 (en) 1998-12-24
BG100716A (bg) 1997-04-30
EP0754678A2 (de) 1997-01-22
HUP9601977A3 (en) 1998-04-28
SI0754678T1 (en) 2001-04-30
HU9601977D0 (en) 1996-09-30
CN1143496A (zh) 1997-02-26
NZ299008A (en) 1998-05-27
CZ214396A3 (en) 1997-02-12
BG62134B1 (bg) 1999-03-31
DE19526274A1 (de) 1997-01-23
SV1996000062A (es) 1997-06-26
AU713555B2 (en) 1999-12-02
ES2275460T3 (es) 2007-06-16
KR100433968B1 (ko) 2004-08-30

Similar Documents

Publication Publication Date Title
BR9600148A (pt) Quinazolinonas 2,8-dissubstituídas processo para sua preparação medicamentos e uso
BR9610988A (pt) Composto uso do mesmo fomulação farmacêutica e processo para produção do composto
BR9612204A (pt) Composto uso do composto composição farmacêutica e processo para preparação do composto e para o tratamento de dor
EE9900014A (et) Erütromütsiinid ja nende valmistamise protsess
BR9612135A (pt) Taxóides processo para sua preparação e composiç o farmacêutica
BR9611198A (pt) Composto processo de preparação do mesmo e composição farmacêutica
BR9607721A (pt) Processo para preparar compostos ciclo-hexapeptídeo
BR9408463A (pt) Novos derivados de ginkgolide e processo para sua preparação
BR9605354A (pt) Composto composição farmacêutica processo para a produção do composto e uso
BR9601093A (pt) Pirido(3,2-E)pirazinoas processo para sua preparação medicamentos processo para sua preparação e utilização
BR9606782A (pt) Processo para preparar ciclopilacetileno
BR9606396A (pt) Derivados de camptotecin substituídos e processo para sua preparação
BR9600147A (pt) Purin-6-onas 2,9-DI-substituidas processo para sua preparação medicamentos e uso
BR9602983A (pt) Gel e processo para sua preparação
BR9601294A (pt) Composto e processo para preparação do mesmo
BR9704986A (pt) Processo de síntese de uréia aperfeiçoado e aparelho para o mesmo
BR9303456A (pt) Compostos,processo para sua preparacao,medicamentos,processo para sua preparacao e emprego
BR9800557A (pt) Processo contínuo para preparação de 4-aminopiperidinas
BR9602337A (pt) Composto processo para sua preparação usos do mesmo processo para tratamento de arritmias e medicamento
BR9603124A (pt) Dipeptídeo processo para preparação do mesmo mistura e medicamentos
BR9400338A (pt) Processo para preparação de 1,1,1,2-tetrafluoro-2-cloroetano e de pentafluoretano
BR9600778A (pt) Benzenossulfoniluréia e - tiouréla substituida processo para sua preparação seu uso e medicamento
BR9601193A (pt) Vacina de múltiplos componentes e processos para preparar e administrar a vacina
NO962534D0 (no) Polyorganosiloksanforbindelser, fremgangsmåte for fremstilling derav, samt anvendelse og blanding
BR9611010A (pt) Processo para preparação de medicamento antimalária

Legal Events

Date Code Title Description
FB34 Technical and formal requirements: requirement - article 34 of industrial property law
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B11D Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time
B15K Others concerning applications: alteration of classification

Ipc: C07C 237/04 (2006.01), A61K 31/195 (2006.0