BR9303456A - Compostos,processo para sua preparacao,medicamentos,processo para sua preparacao e emprego - Google Patents

Compostos,processo para sua preparacao,medicamentos,processo para sua preparacao e emprego

Info

Publication number
BR9303456A
BR9303456A BR9303456A BR9303456A BR9303456A BR 9303456 A BR9303456 A BR 9303456A BR 9303456 A BR9303456 A BR 9303456A BR 9303456 A BR9303456 A BR 9303456A BR 9303456 A BR9303456 A BR 9303456A
Authority
BR
Brazil
Prior art keywords
preparation
employment
drugs
compounds
Prior art date
Application number
BR9303456A
Other languages
English (en)
Inventor
Hans-Reinhold Dr Dieter
Juergen Dr Engel
Karl-Heinz Dr Klinger
Bernhard Dr Kutscher
Stefan Dr Szelenyi
Ute Dr Achterrath-Tuckermann
Juergen Dr Schmidt
Peter Dr Metzenauer
Original Assignee
Asta Medica Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asta Medica Ag filed Critical Asta Medica Ag
Publication of BR9303456A publication Critical patent/BR9303456A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
BR9303456A 1992-08-24 1993-08-23 Compostos,processo para sua preparacao,medicamentos,processo para sua preparacao e emprego BR9303456A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4228095A DE4228095A1 (de) 1992-08-24 1992-08-24 Neue 4,5-Dihydro-4-oxo-pyrrolo[1,2-a]chinoxaline und entsprechende Aza-analoga und Verfahren zu deren Herstellung

Publications (1)

Publication Number Publication Date
BR9303456A true BR9303456A (pt) 1994-03-22

Family

ID=6466304

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9303456A BR9303456A (pt) 1992-08-24 1993-08-23 Compostos,processo para sua preparacao,medicamentos,processo para sua preparacao e emprego

Country Status (18)

Country Link
US (1) US5405847A (pt)
EP (1) EP0584487A3 (pt)
JP (1) JPH06184155A (pt)
KR (1) KR940003957A (pt)
CN (1) CN1088928A (pt)
AU (1) AU661408B2 (pt)
BR (1) BR9303456A (pt)
CA (1) CA2104653A1 (pt)
CZ (1) CZ170693A3 (pt)
DE (1) DE4228095A1 (pt)
FI (1) FI933705A (pt)
HU (1) HUT70165A (pt)
IL (1) IL106761A0 (pt)
MX (1) MX9305092A (pt)
NO (1) NO932998L (pt)
PH (1) PH30110A (pt)
SK (1) SK89693A3 (pt)
ZA (1) ZA936169B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2704547B1 (fr) * 1993-04-30 1995-06-09 Adir Nouveaux composés pyrrolopyraziniques, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
DE19510965A1 (de) * 1995-03-24 1996-09-26 Asta Medica Ag Neue Pyrido/3,2-e/pyrazinone mit antiasthmatischer Wirksamkeit und Verfahren zu deren Herstellung
US6465465B1 (en) 2000-03-14 2002-10-15 Arzneimittelwerk Dresden Gmbh Process for the treatment of erectile dysfunction and product therefor
DE10012373A1 (de) * 2000-03-14 2001-09-20 Dresden Arzneimittel Verwendung von Pyrido[3,2-e]-pyrazinonen als Inhibitoren der Phosphodiesterase 5 zur Therapie von erektiler Dysfunktion
EP1312363A1 (en) * 2001-09-28 2003-05-21 Pfizer Products Inc. Methods of treatment and kits comprising a growth hormone secretagogue
US7550459B2 (en) 2001-12-28 2009-06-23 Acadia Pharmaceuticals, Inc. Tetrahydroquinoline analogues as muscarinic agonists
WO2003057672A2 (en) 2001-12-28 2003-07-17 Acadia Pharmaceuticals, Inc. Tetrahydroquinoline analogues as muscarinic agonists
US7342884B2 (en) * 2002-03-13 2008-03-11 Harmonic, Inc. Method and apparatus for one directional communications in bidirectional communications channel
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
CN101616919B (zh) * 2006-12-28 2012-10-10 雅培制药有限公司 聚(adp核糖)聚合酶抑制剂
EP2389379A1 (en) 2009-01-23 2011-11-30 Takeda Pharmaceutical Company Limited Poly (ADP-Ribose) Polymerase (PARP) Inhibitors
US8541417B2 (en) 2009-07-30 2013-09-24 Takeda Pharmaceutical Company Limited Poly (ADP-ribose) polymerase (PARP) inhibitors
WO2011081915A2 (en) * 2009-12-15 2011-07-07 Cebix Inc. Methods for treating erectile dysfunction in patients with insulin-dependent diabetes
JP6076913B2 (ja) * 2010-12-07 2017-02-08 ドレクセル ユニバーシティ 癌からの転移を阻害する方法
WO2018204370A1 (en) 2017-05-02 2018-11-08 Drexel University Cx3cr1 small molecule antagonists, and methods using same
MX2022015829A (es) 2020-06-11 2023-04-05 Chdi Foundation Inc Compuestos heterocíclicos y agentes formadores de imágenes para formar la imagen de la proteína huntingtina.
CN114560862A (zh) * 2022-03-08 2022-05-31 山东龙辰药业有限公司 一种吡咯并[1,2-a]喹喔啉-4(5h)-酮及其衍生物的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1576077A (en) * 1977-04-13 1980-10-01 Roussel Lab Ltd 4,5-dihydro-4-oxophyrrolo(1,2-)-quinoxaline-2-carboxylic acids and derivatives
GB2043637B (en) * 1979-02-09 1983-03-16 Roussel Lab Ltd Heterotricyclic derivatives
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
US4446323A (en) * 1983-05-23 1984-05-01 American Home Products Corporation Tetra- and hexa-hydropyrrolo(1,2-a)quinoxaline and azaquinoxaline derivatives
IL90315A0 (en) * 1988-06-01 1989-12-15 Ferrosan As Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them
DK626288D0 (da) * 1988-11-10 1988-11-10 Ferrosan As Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen
US5055465A (en) * 1989-05-31 1991-10-08 Berlex Laboratories, Inc. Imidazoquinoxalinones, their aza analogs and process for their preparation
US5306819A (en) * 1992-08-27 1994-04-26 Neurogen Corporation Certain aryl a cycloalkyl fused imidazopyrazinols; and new class of GABA brain receptor ligands

Also Published As

Publication number Publication date
EP0584487A2 (de) 1994-03-02
SK89693A3 (en) 1994-03-09
AU4483393A (en) 1994-03-03
MX9305092A (es) 1994-02-28
CN1088928A (zh) 1994-07-06
HU9302397D0 (en) 1993-11-29
FI933705A (fi) 1994-02-25
DE4228095A1 (de) 1994-03-03
JPH06184155A (ja) 1994-07-05
CA2104653A1 (en) 1994-02-25
CZ170693A3 (en) 1994-03-16
PH30110A (en) 1996-12-27
US5405847A (en) 1995-04-11
HUT70165A (en) 1995-09-28
FI933705A0 (fi) 1993-08-23
EP0584487A3 (en) 1994-07-06
NO932998L (no) 1994-02-25
KR940003957A (ko) 1994-03-14
ZA936169B (en) 1994-03-17
AU661408B2 (en) 1995-07-20
NO932998D0 (no) 1993-08-23
IL106761A0 (en) 1993-12-08

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Legal Events

Date Code Title Description
EE Request for examination
EG Technical examination (opinion): publication of technical examination (opinion)
FC Decision: refusal
FC Decision: refusal
B15K Others concerning applications: alteration of classification

Ipc: C07D 471/14 (2006.01), C07D 487/04 (2006.0