PT96937A - Processo para a preparacao de derivados de n-(4-piperidinil) (di-hidro-benzofurano ou di-hidro-2h-benzopiran) carboxamida e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados de n-(4-piperidinil) (di-hidro-benzofurano ou di-hidro-2h-benzopiran) carboxamida e de composicoes farmaceuticas que os contem

Info

Publication number
PT96937A
PT96937A PT96937A PT9693791A PT96937A PT 96937 A PT96937 A PT 96937A PT 96937 A PT96937 A PT 96937A PT 9693791 A PT9693791 A PT 9693791A PT 96937 A PT96937 A PT 96937A
Authority
PT
Portugal
Prior art keywords
aryl
alkyl
dihydro
alk
cycloalkyl
Prior art date
Application number
PT96937A
Other languages
English (en)
Other versions
PT96937B (pt
Inventor
Georges Henri Paul Van Daele
Jean-Paul Rene Marie A Bosmans
Michel Anna Josef De Cleyn
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PT96937A publication Critical patent/PT96937A/pt
Publication of PT96937B publication Critical patent/PT96937B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10—Laxatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrane Compounds (AREA)
  • Cosmetics (AREA)
PT96937A 1990-03-06 1991-03-05 Processo para a preparacao de derivados de n-(4-piperidinil) (di-hidro-benzofurano ou di-hidro-2h-benzopiran) carboxamida e de composicoes farmaceuticas que os contem PT96937B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909005014A GB9005014D0 (en) 1990-03-06 1990-03-06 N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives

Publications (2)

Publication Number Publication Date
PT96937A true PT96937A (pt) 1991-10-31
PT96937B PT96937B (pt) 1998-07-31

Family

ID=10672103

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96937A PT96937B (pt) 1990-03-06 1991-03-05 Processo para a preparacao de derivados de n-(4-piperidinil) (di-hidro-benzofurano ou di-hidro-2h-benzopiran) carboxamida e de composicoes farmaceuticas que os contem

Country Status (39)

Country Link
US (2) US5185335A (pt)
EP (1) EP0445862B1 (pt)
JP (1) JP2601566B2 (pt)
KR (1) KR0177521B1 (pt)
CN (1) CN1038936C (pt)
AT (1) ATE191912T1 (pt)
AU (1) AU636012B2 (pt)
BG (1) BG60381B1 (pt)
CA (1) CA2037575C (pt)
CY (1) CY2235B1 (pt)
CZ (1) CZ286617B6 (pt)
DE (1) DE69132119T2 (pt)
DK (1) DK0445862T3 (pt)
ES (1) ES2147175T3 (pt)
FI (1) FI101622B (pt)
GB (1) GB9005014D0 (pt)
GR (1) GR3033461T3 (pt)
HK (1) HK1010727A1 (pt)
HR (1) HRP930483B1 (pt)
HU (2) HU221627B1 (pt)
IE (1) IE910710A1 (pt)
IL (1) IL97018A (pt)
LT (1) LT3708B (pt)
LV (1) LV10085B (pt)
MA (1) MA22076A1 (pt)
MY (1) MY108831A (pt)
NO (1) NO177424C (pt)
NZ (1) NZ237189A (pt)
PL (6) PL169238B1 (pt)
PT (1) PT96937B (pt)
RU (1) RU2070884C1 (pt)
SG (1) SG47482A1 (pt)
SI (1) SI9110396B (pt)
SK (2) SK282406B6 (pt)
TN (1) TNSN91010A1 (pt)
UA (1) UA25969A1 (pt)
YU (1) YU48854B (pt)
ZA (1) ZA911611B (pt)
ZW (1) ZW2391A1 (pt)

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JPH0873463A (ja) 1994-07-05 1996-03-19 Sanwa Kagaku Kenkyusho Co Ltd ベンゾピランカルボキサミド誘導体、その塩及び製法並びに用途
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TW548103B (en) * 1997-07-11 2003-08-21 Janssen Pharmaceutica Nv Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
EP1076055B1 (en) 1998-04-28 2004-11-24 Dainippon Pharmaceutical Co., Ltd. 1- (1-substituted-4-piperidinyl)methyl]-4-piperidine derivatives, process for producing the same, medicinal compositions containing the same and intermediates of these compounds
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EP1112270B1 (en) 1998-09-10 2007-03-21 F. Hoffmann-La Roche Ag Dihydrobenzodioxine carboxamide and ketone derivatives as 5-ht4 receptor antagonists
NZ511117A (en) * 1998-11-23 2002-11-26 Janssen Pharmaceutica Nv Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia
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SE9902987D0 (sv) 1999-08-24 1999-08-24 Astra Pharma Prod Novel compounds
CN1288730A (zh) * 1999-09-07 2001-03-28 麦克内尔-Ppc股份有限公司 轻泻组合物
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PL214274B1 (pl) * 2002-01-16 2013-07-31 Movetis N V N-Tlenek prukaloprydu, sposób jego wytwarzania i zastosowanie oraz zawierająca go kompozycja i sposób jej wytwarzania
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SE0301369D0 (sv) 2003-05-09 2003-05-09 Astrazeneca Ab Chemical compounds
DE10349113A1 (de) * 2003-10-17 2005-05-12 Boehringer Ingelheim Pharma Verfahren zur Herstellung von Aminocrotonylverbindungen
GB0525661D0 (en) * 2005-12-16 2006-01-25 Glaxo Group Ltd Novel compounds
PT2674428T (pt) * 2006-04-07 2016-07-14 Vertex Pharma Modeladores de transportadores de cassetes de ligação de atp
CN102477002B (zh) * 2010-11-26 2015-04-15 苏州凯达生物医药技术有限公司 3-氨基-2,2-双甲基丙酰胺的制备方法
HUE029988T2 (en) 2011-02-25 2017-04-28 Yuhan Corp Diaminopyrimidine derivatives and processes for their preparation
GB201103397D0 (pt) * 2011-02-28 2011-04-13 Shire Movetis N V
KR101256908B1 (ko) * 2011-04-28 2013-04-23 (주)에이치비메디컬스 주름제거용 충전체
CN102295594B (zh) * 2011-07-12 2016-01-20 上海医药工业研究院 4-n-取代-1-(3-甲氧基丙基)-4-哌啶胺类化合物及制备和应用
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Also Published As

Publication number Publication date
ATE191912T1 (de) 2000-05-15
UA25969A1 (uk) 1999-02-26
CS46091A3 (en) 1991-10-15
CY2235B1 (en) 2003-07-04
JPH04211685A (ja) 1992-08-03
RU2070884C1 (ru) 1996-12-27
NO910863L (no) 1991-09-09
LT3708B (en) 1996-02-26
HU211350A9 (en) 1995-11-28
GR3033461T3 (en) 2000-09-29
DE69132119D1 (de) 2000-05-25
SI9110396B (sl) 2000-06-30
LV10085B (en) 1995-02-20
EP0445862A2 (en) 1991-09-11
NZ237189A (en) 1992-11-25
ZW2391A1 (en) 1992-09-07
CA2037575A1 (en) 1991-09-07
MY108831A (en) 1996-11-30
HUT60733A (en) 1992-10-28
KR910016744A (ko) 1991-11-05
PL168686B1 (pl) 1996-03-29
EP0445862B1 (en) 2000-04-19
NO177424B (no) 1995-06-06
EP0445862A3 (en) 1992-05-20
CA2037575C (en) 2003-09-16
FI911096A (fi) 1991-09-07
TNSN91010A1 (fr) 1992-10-25
FI101622B1 (fi) 1998-07-31
SK282407B6 (sk) 2002-01-07
CN1038936C (zh) 1998-07-01
LTIP846A (en) 1995-02-27
US5185335A (en) 1993-02-09
HU910706D0 (en) 1991-09-30
FI911096A0 (fi) 1991-03-05
NO177424C (no) 1995-09-13
ES2147175T3 (es) 2000-09-01
PL169238B1 (pl) 1996-06-28
DE69132119T2 (de) 2000-12-21
DK0445862T3 (da) 2000-09-04
FI101622B (fi) 1998-07-31
CN1054598A (zh) 1991-09-18
MA22076A1 (fr) 1991-10-01
YU48854B (sh) 2002-06-19
HK1010727A1 (en) 1999-06-25
IL97018A (en) 1995-11-27
HRP930483A2 (en) 1995-12-31
PT96937B (pt) 1998-07-31
BG60381B1 (bg) 1995-01-31
PL168693B1 (pl) 1996-03-29
AU636012B2 (en) 1993-04-08
NO910863D0 (no) 1991-03-05
HRP930483B1 (en) 2001-04-30
SK282406B6 (sk) 2002-01-07
JP2601566B2 (ja) 1997-04-16
CZ286617B6 (cs) 2000-05-17
HU221627B1 (hu) 2002-12-28
AU7207991A (en) 1991-09-12
PL289323A1 (en) 1992-03-09
LV10085A (lv) 1994-05-10
SI9110396A (en) 1997-12-31
US5262418A (en) 1993-11-16
YU39691A (sh) 1994-06-10
PL168356B1 (pl) 1996-02-29
IE910710A1 (en) 1991-09-11
KR0177521B1 (ko) 1999-03-20
IL97018A0 (en) 1992-03-29
PL168811B1 (pl) 1996-04-30
SG47482A1 (en) 1998-04-17
PL168384B1 (en) 1996-02-29
GB9005014D0 (en) 1990-05-02
ZA911611B (en) 1992-11-25

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Effective date: 19980414

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Effective date: 20130415