PT1373255E - Processo para a preparacao de compostos de imidazole - Google Patents
Processo para a preparacao de compostos de imidazoleInfo
- Publication number
- PT1373255E PT1373255E PT02722184T PT02722184T PT1373255E PT 1373255 E PT1373255 E PT 1373255E PT 02722184 T PT02722184 T PT 02722184T PT 02722184 T PT02722184 T PT 02722184T PT 1373255 E PT1373255 E PT 1373255E
- Authority
- PT
- Portugal
- Prior art keywords
- preparation
- imidazole compounds
- imidazole
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epoxy Resins (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP01200928 | 2001-03-12 | ||
PCT/EP2002/002459 WO2002072574A1 (en) | 2001-03-12 | 2002-03-05 | Process for the preparation of imidazole compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1373255E true PT1373255E (pt) | 2005-05-31 |
Family
ID=8180004
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT02722184T PT1373255E (pt) | 2001-03-12 | 2002-03-05 | Processo para a preparacao de compostos de imidazole |
Country Status (32)
Country | Link |
---|---|
US (1) | US6844439B2 (pt) |
EP (1) | EP1373255B1 (pt) |
JP (1) | JP4257698B2 (pt) |
KR (1) | KR100849042B1 (pt) |
CN (1) | CN1246318C (pt) |
AR (1) | AR035944A1 (pt) |
AT (1) | ATE287882T1 (pt) |
AU (1) | AU2002253101B2 (pt) |
BR (1) | BRPI0208075B8 (pt) |
CA (1) | CA2438421C (pt) |
CZ (1) | CZ300622B6 (pt) |
DE (1) | DE60202755T2 (pt) |
DK (1) | DK1373255T3 (pt) |
EA (1) | EA006770B1 (pt) |
EE (1) | EE05247B1 (pt) |
ES (1) | ES2236505T3 (pt) |
HK (1) | HK1063315A1 (pt) |
HR (1) | HRP20030695B1 (pt) |
HU (1) | HU230282B1 (pt) |
IL (2) | IL157839A0 (pt) |
MX (1) | MXPA03008205A (pt) |
MY (1) | MY124838A (pt) |
NO (1) | NO324954B1 (pt) |
NZ (1) | NZ528620A (pt) |
PL (1) | PL208238B1 (pt) |
PT (1) | PT1373255E (pt) |
SI (1) | SI1373255T1 (pt) |
SK (1) | SK287807B6 (pt) |
TW (1) | TWI249532B (pt) |
UA (1) | UA74871C2 (pt) |
WO (1) | WO2002072574A1 (pt) |
ZA (1) | ZA200307117B (pt) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR0208010A (pt) | 2001-03-12 | 2004-12-21 | Avanir Pharmaceuticals | Composto de benzimidazol para modulação de ige e inibição de proliferação celular |
WO2004024655A2 (en) | 2002-09-12 | 2004-03-25 | Avanir Pharmaceuticals | Phenyl-indole compounds for modulating ige and inhibiting cellular proliferation |
TWI276631B (en) | 2002-09-12 | 2007-03-21 | Avanir Pharmaceuticals | Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation |
US20060106060A1 (en) * | 2004-03-18 | 2006-05-18 | The Brigham And Women's Hospital, Inc. | Methods for the treatment of synucleinopathies (Lansbury) |
CN100567291C (zh) * | 2004-05-03 | 2009-12-09 | 詹森药业有限公司 | 用6-溴-4-(3-氯苯基)-2-甲氧基喹啉进行的非对映选择性合成方法 |
DE602005007604D1 (de) | 2004-05-03 | 2008-07-31 | Janssen Pharmaceutica Nv | Diastereoselektive addition von lithiiertem n-methylimidazol an sulfinimine |
WO2005105784A1 (en) * | 2004-05-03 | 2005-11-10 | Janssen Pharmaceutica N.V. | Diastereoselective synthesis process for the preparation of imidazole compounds |
US20070213366A1 (en) | 2005-12-23 | 2007-09-13 | Justman Craig J | Treatment of Synucleinopathies |
WO2009151683A2 (en) * | 2008-03-12 | 2009-12-17 | Link Medicine Corporation | Quinolinone farnesyl transferase inhibitors for the treatment of synucleinopathies and other indications |
KR101044430B1 (ko) * | 2009-09-25 | 2011-06-27 | 듀오백코리아 주식회사 | 요추받이를 포함하는 의자의 등 지지 장치 |
KR101107900B1 (ko) * | 2009-10-21 | 2012-01-25 | 성용기업 주식회사 | 의자용 허리지지장치 |
KR101885361B1 (ko) | 2015-08-17 | 2018-08-06 | 쿠라 온콜로지, 인크. | 파르네실전달효소 억제제를 이용하여 암환자를 치료하는 방법 |
JP2019534290A (ja) | 2016-11-03 | 2019-11-28 | クラ オンコロジー, インコーポレイテッド | 癌の治療方法において使用するためのファルネシルトランスフェラーゼ阻害剤 |
WO2018103027A1 (zh) * | 2016-12-08 | 2018-06-14 | 杭州领业医药科技有限公司 | 替吡法尼的晶型及其制备方法及药物组合物 |
JP2021526513A (ja) * | 2018-05-18 | 2021-10-07 | クラ オンコロジー, インコーポレイテッド | ティピファニブの合成 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW349948B (en) | 1995-10-31 | 1999-01-11 | Janssen Pharmaceutica Nv | Farnesyl transferase inhibiting 2-quinolone derivatives |
EP1162201B1 (en) * | 1995-12-08 | 2006-03-29 | Janssen Pharmaceutica N.V. | Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives |
TW591030B (en) * | 1997-03-10 | 2004-06-11 | Janssen Pharmaceutica Nv | Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with N- or C-linked imidazoles |
IL130363A (en) * | 1997-04-25 | 2002-08-14 | Janssen Pharmaceutica Nv | Quinazolines that inhibit frenzyl transferase, their preparation and pharmaceutical preparations containing them |
NZ509372A (en) | 1998-08-27 | 2003-08-29 | Pfizer Prod Inc | Substituted quinolin-2-one derivatives, pharmaceuticals thereof and their use for treating abnormal cell growth (e.g. cancer) |
ATE289602T1 (de) | 1998-08-27 | 2005-03-15 | Pfizer Prod Inc | Quinolin-2-on-derivate verwendbar als antikrebsmittel |
-
2002
- 2002-03-05 EE EEP200300442A patent/EE05247B1/xx unknown
- 2002-03-05 AU AU2002253101A patent/AU2002253101B2/en not_active Expired
- 2002-03-05 PT PT02722184T patent/PT1373255E/pt unknown
- 2002-03-05 CZ CZ20032704A patent/CZ300622B6/cs not_active IP Right Cessation
- 2002-03-05 US US10/471,215 patent/US6844439B2/en not_active Expired - Lifetime
- 2002-03-05 AT AT02722184T patent/ATE287882T1/de active
- 2002-03-05 CA CA2438421A patent/CA2438421C/en not_active Expired - Lifetime
- 2002-03-05 SK SK1246-2003A patent/SK287807B6/sk unknown
- 2002-03-05 DE DE60202755T patent/DE60202755T2/de not_active Expired - Lifetime
- 2002-03-05 BR BR0208075-3 patent/BRPI0208075B8/pt not_active IP Right Cessation
- 2002-03-05 HU HU0303443A patent/HU230282B1/hu unknown
- 2002-03-05 NZ NZ528620A patent/NZ528620A/en not_active IP Right Cessation
- 2002-03-05 WO PCT/EP2002/002459 patent/WO2002072574A1/en active IP Right Grant
- 2002-03-05 ES ES02722184T patent/ES2236505T3/es not_active Expired - Lifetime
- 2002-03-05 EP EP02722184A patent/EP1373255B1/en not_active Expired - Lifetime
- 2002-03-05 PL PL363263A patent/PL208238B1/pl unknown
- 2002-03-05 MX MXPA03008205A patent/MXPA03008205A/es active IP Right Grant
- 2002-03-05 CN CNB02806335XA patent/CN1246318C/zh not_active Expired - Lifetime
- 2002-03-05 DK DK02722184T patent/DK1373255T3/da active
- 2002-03-05 IL IL15783902A patent/IL157839A0/xx unknown
- 2002-03-05 EA EA200300998A patent/EA006770B1/ru not_active IP Right Cessation
- 2002-03-05 KR KR1020037010091A patent/KR100849042B1/ko active IP Right Grant
- 2002-03-05 JP JP2002571490A patent/JP4257698B2/ja not_active Expired - Lifetime
- 2002-03-05 SI SI200230100T patent/SI1373255T1/xx unknown
- 2002-03-11 AR ARP020100873A patent/AR035944A1/es active IP Right Grant
- 2002-03-11 MY MYPI20020866A patent/MY124838A/en unknown
- 2002-03-11 TW TW091104444A patent/TWI249532B/zh not_active IP Right Cessation
- 2002-05-03 UA UA2003087776A patent/UA74871C2/uk unknown
-
2003
- 2003-09-01 HR HR20030695A patent/HRP20030695B1/xx not_active IP Right Cessation
- 2003-09-10 NO NO20034003A patent/NO324954B1/no not_active IP Right Cessation
- 2003-09-10 IL IL157839A patent/IL157839A/en unknown
- 2003-09-11 ZA ZA200307117A patent/ZA200307117B/en unknown
-
2004
- 2004-08-12 HK HK04106065A patent/HK1063315A1/xx not_active IP Right Cessation
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