PT1373255E - Processo para a preparacao de compostos de imidazole - Google Patents

Processo para a preparacao de compostos de imidazole

Info

Publication number
PT1373255E
PT1373255E PT02722184T PT02722184T PT1373255E PT 1373255 E PT1373255 E PT 1373255E PT 02722184 T PT02722184 T PT 02722184T PT 02722184 T PT02722184 T PT 02722184T PT 1373255 E PT1373255 E PT 1373255E
Authority
PT
Portugal
Prior art keywords
preparation
imidazole compounds
imidazole
compounds
Prior art date
Application number
PT02722184T
Other languages
English (en)
Inventor
Walter Ferdinand Mari Filliers
Rudy Laurent Maria Broeckx
Stefan Marcel Herman Leurs
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PT1373255E publication Critical patent/PT1373255E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epoxy Resins (AREA)
PT02722184T 2001-03-12 2002-03-05 Processo para a preparacao de compostos de imidazole PT1373255E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01200928 2001-03-12
PCT/EP2002/002459 WO2002072574A1 (en) 2001-03-12 2002-03-05 Process for the preparation of imidazole compounds

Publications (1)

Publication Number Publication Date
PT1373255E true PT1373255E (pt) 2005-05-31

Family

ID=8180004

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02722184T PT1373255E (pt) 2001-03-12 2002-03-05 Processo para a preparacao de compostos de imidazole

Country Status (32)

Country Link
US (1) US6844439B2 (pt)
EP (1) EP1373255B1 (pt)
JP (1) JP4257698B2 (pt)
KR (1) KR100849042B1 (pt)
CN (1) CN1246318C (pt)
AR (1) AR035944A1 (pt)
AT (1) ATE287882T1 (pt)
AU (1) AU2002253101B2 (pt)
BR (1) BRPI0208075B8 (pt)
CA (1) CA2438421C (pt)
CZ (1) CZ300622B6 (pt)
DE (1) DE60202755T2 (pt)
DK (1) DK1373255T3 (pt)
EA (1) EA006770B1 (pt)
EE (1) EE05247B1 (pt)
ES (1) ES2236505T3 (pt)
HK (1) HK1063315A1 (pt)
HR (1) HRP20030695B1 (pt)
HU (1) HU230282B1 (pt)
IL (2) IL157839A0 (pt)
MX (1) MXPA03008205A (pt)
MY (1) MY124838A (pt)
NO (1) NO324954B1 (pt)
NZ (1) NZ528620A (pt)
PL (1) PL208238B1 (pt)
PT (1) PT1373255E (pt)
SI (1) SI1373255T1 (pt)
SK (1) SK287807B6 (pt)
TW (1) TWI249532B (pt)
UA (1) UA74871C2 (pt)
WO (1) WO2002072574A1 (pt)
ZA (1) ZA200307117B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0208010A (pt) 2001-03-12 2004-12-21 Avanir Pharmaceuticals Composto de benzimidazol para modulação de ige e inibição de proliferação celular
WO2004024655A2 (en) 2002-09-12 2004-03-25 Avanir Pharmaceuticals Phenyl-indole compounds for modulating ige and inhibiting cellular proliferation
TWI276631B (en) 2002-09-12 2007-03-21 Avanir Pharmaceuticals Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
US20060106060A1 (en) * 2004-03-18 2006-05-18 The Brigham And Women's Hospital, Inc. Methods for the treatment of synucleinopathies (Lansbury)
CN100567291C (zh) * 2004-05-03 2009-12-09 詹森药业有限公司 用6-溴-4-(3-氯苯基)-2-甲氧基喹啉进行的非对映选择性合成方法
DE602005007604D1 (de) 2004-05-03 2008-07-31 Janssen Pharmaceutica Nv Diastereoselektive addition von lithiiertem n-methylimidazol an sulfinimine
WO2005105784A1 (en) * 2004-05-03 2005-11-10 Janssen Pharmaceutica N.V. Diastereoselective synthesis process for the preparation of imidazole compounds
US20070213366A1 (en) 2005-12-23 2007-09-13 Justman Craig J Treatment of Synucleinopathies
WO2009151683A2 (en) * 2008-03-12 2009-12-17 Link Medicine Corporation Quinolinone farnesyl transferase inhibitors for the treatment of synucleinopathies and other indications
KR101044430B1 (ko) * 2009-09-25 2011-06-27 듀오백코리아 주식회사 요추받이를 포함하는 의자의 등 지지 장치
KR101107900B1 (ko) * 2009-10-21 2012-01-25 성용기업 주식회사 의자용 허리지지장치
KR101885361B1 (ko) 2015-08-17 2018-08-06 쿠라 온콜로지, 인크. 파르네실전달효소 억제제를 이용하여 암환자를 치료하는 방법
JP2019534290A (ja) 2016-11-03 2019-11-28 クラ オンコロジー, インコーポレイテッド 癌の治療方法において使用するためのファルネシルトランスフェラーゼ阻害剤
WO2018103027A1 (zh) * 2016-12-08 2018-06-14 杭州领业医药科技有限公司 替吡法尼的晶型及其制备方法及药物组合物
JP2021526513A (ja) * 2018-05-18 2021-10-07 クラ オンコロジー, インコーポレイテッド ティピファニブの合成

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW349948B (en) 1995-10-31 1999-01-11 Janssen Pharmaceutica Nv Farnesyl transferase inhibiting 2-quinolone derivatives
EP1162201B1 (en) * 1995-12-08 2006-03-29 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
TW591030B (en) * 1997-03-10 2004-06-11 Janssen Pharmaceutica Nv Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with N- or C-linked imidazoles
IL130363A (en) * 1997-04-25 2002-08-14 Janssen Pharmaceutica Nv Quinazolines that inhibit frenzyl transferase, their preparation and pharmaceutical preparations containing them
NZ509372A (en) 1998-08-27 2003-08-29 Pfizer Prod Inc Substituted quinolin-2-one derivatives, pharmaceuticals thereof and their use for treating abnormal cell growth (e.g. cancer)
ATE289602T1 (de) 1998-08-27 2005-03-15 Pfizer Prod Inc Quinolin-2-on-derivate verwendbar als antikrebsmittel

Also Published As

Publication number Publication date
ATE287882T1 (de) 2005-02-15
BRPI0208075B1 (pt) 2018-02-14
DE60202755D1 (de) 2005-03-03
ES2236505T3 (es) 2005-07-16
ZA200307117B (en) 2004-09-13
IL157839A0 (en) 2004-03-28
HK1063315A1 (en) 2004-12-24
US6844439B2 (en) 2005-01-18
PL208238B1 (pl) 2011-04-29
MXPA03008205A (es) 2004-01-29
US20040138256A1 (en) 2004-07-15
CN1496363A (zh) 2004-05-12
CZ300622B6 (cs) 2009-07-01
NO324954B1 (no) 2008-01-14
TWI249532B (en) 2006-02-21
CA2438421C (en) 2010-05-18
EE05247B1 (et) 2009-12-15
KR100849042B1 (ko) 2008-07-29
BR0208075A (pt) 2004-03-02
EP1373255B1 (en) 2005-01-26
SK12462003A3 (sk) 2004-06-08
EE200300442A (et) 2003-12-15
HUP0303443A2 (hu) 2004-01-28
CN1246318C (zh) 2006-03-22
CA2438421A1 (en) 2002-09-19
CZ20032704A3 (en) 2004-03-17
PL363263A1 (en) 2004-11-15
AU2002253101B2 (en) 2007-08-09
NO20034003L (no) 2003-10-22
EA200300998A1 (ru) 2004-02-26
EA006770B1 (ru) 2006-04-28
HU230282B1 (hu) 2015-12-28
BRPI0208075B8 (pt) 2021-05-25
JP4257698B2 (ja) 2009-04-22
NO20034003D0 (no) 2003-09-10
WO2002072574A1 (en) 2002-09-19
NZ528620A (en) 2005-01-28
IL157839A (en) 2008-07-08
KR20030079971A (ko) 2003-10-10
SI1373255T1 (pt) 2005-08-31
AR035944A1 (es) 2004-07-28
HRP20030695B1 (en) 2011-07-31
HUP0303443A3 (en) 2012-09-28
SK287807B6 (sk) 2011-10-04
EP1373255A1 (en) 2004-01-02
UA74871C2 (en) 2006-02-15
MY124838A (en) 2006-07-31
JP2004523575A (ja) 2004-08-05
DE60202755T2 (de) 2006-03-30
HRP20030695A2 (en) 2005-02-28
DK1373255T3 (da) 2005-05-23

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