PT1345939E - Processo para a preparacao de imidazotriazinonas substituidas por sulfonamida - Google Patents

Processo para a preparacao de imidazotriazinonas substituidas por sulfonamida

Info

Publication number
PT1345939E
PT1345939E PT01271374T PT01271374T PT1345939E PT 1345939 E PT1345939 E PT 1345939E PT 01271374 T PT01271374 T PT 01271374T PT 01271374 T PT01271374 T PT 01271374T PT 1345939 E PT1345939 E PT 1345939E
Authority
PT
Portugal
Prior art keywords
sulfonamide
preparation
substituted imidazotriazinones
imidazotriazinones
substituted
Prior art date
Application number
PT01271374T
Other languages
English (en)
Inventor
Marc Nowakowski
Gehring Reinhold
Heilmann Werner
Wahl Karl-Heinz
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of PT1345939E publication Critical patent/PT1345939E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
PT01271374T 2000-12-18 2001-12-05 Processo para a preparacao de imidazotriazinonas substituidas por sulfonamida PT1345939E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10063108A DE10063108A1 (de) 2000-12-18 2000-12-18 Verfahren zur Herstellung von Sulfonamid-substituierten Imidazotriazinonen

Publications (1)

Publication Number Publication Date
PT1345939E true PT1345939E (pt) 2006-08-31

Family

ID=7667666

Family Applications (1)

Application Number Title Priority Date Filing Date
PT01271374T PT1345939E (pt) 2000-12-18 2001-12-05 Processo para a preparacao de imidazotriazinonas substituidas por sulfonamida

Country Status (43)

Country Link
US (3) US6777551B2 (pt)
EP (1) EP1345939B1 (pt)
JP (1) JP4441175B2 (pt)
KR (1) KR100787288B1 (pt)
CN (1) CN1227253C (pt)
AR (1) AR032775A1 (pt)
AT (1) ATE328885T1 (pt)
AU (2) AU1708902A (pt)
BG (1) BG66142B1 (pt)
BR (1) BRPI0116227B8 (pt)
CA (1) CA2431933C (pt)
CU (2) CU23341B7 (pt)
CY (1) CY1105197T1 (pt)
CZ (1) CZ297005B6 (pt)
DE (2) DE10063108A1 (pt)
DK (1) DK1345939T3 (pt)
DO (1) DOP2001000295A (pt)
EC (1) ECSP034657A (pt)
EE (1) EE05308B1 (pt)
ES (1) ES2266098T3 (pt)
GT (1) GT200100251A (pt)
HK (1) HK1063799A1 (pt)
HN (1) HN2001000278A (pt)
HR (1) HRP20030583B1 (pt)
HU (1) HU229296B1 (pt)
IL (2) IL156278A0 (pt)
MA (1) MA25927A1 (pt)
MX (1) MXPA03005429A (pt)
MY (1) MY126689A (pt)
NO (1) NO325398B1 (pt)
NZ (1) NZ526477A (pt)
PE (1) PE20020590A1 (pt)
PL (1) PL207294B1 (pt)
PT (1) PT1345939E (pt)
RU (1) RU2299211C2 (pt)
SI (1) SI1345939T1 (pt)
SK (1) SK286894B6 (pt)
SV (1) SV2003000766A (pt)
TW (1) TWI289562B (pt)
UA (1) UA75109C2 (pt)
UY (2) UY27070A1 (pt)
WO (1) WO2002050076A2 (pt)
ZA (1) ZA200304705B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10063108A1 (de) * 2000-12-18 2002-06-20 Bayer Ag Verfahren zur Herstellung von Sulfonamid-substituierten Imidazotriazinonen
DE10107639A1 (de) * 2001-02-15 2002-08-22 Bayer Ag 2-Alkoxyphenyl-substituierte Imidazotriazinone
DE10232113A1 (de) 2002-07-16 2004-01-29 Bayer Ag Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel
DE202004006552U1 (de) * 2004-04-26 2004-07-08 Knürr AG Kühlungssystem für Geräte- und Netzwerkschränke
DE102004023069A1 (de) 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil
US7977478B2 (en) * 2006-03-13 2011-07-12 Dr. Reddy's Laboratories Limited Polymorphic forms of vardenafil
WO2009030095A1 (en) * 2007-09-06 2009-03-12 Topharman Shanghai Co., Ltd. Process for preparing vardenafil and its intermediates
WO2009082845A1 (en) 2007-12-28 2009-07-09 Topharman Shanghai Co., Ltd. N-{1-[3-(2-ethoxy-5-(4-ethylpiperazinyl)benzenesulfonyl)-4,5-dihydro-5-oxo-1,2,4-triazin-6-yl]ethyl}butyramide, the preparation method and use thereof
CA2770471A1 (en) 2009-08-07 2011-02-10 Ranbaxy Laboratories Limited Processes for the preparation of vardenafil
PL390079A1 (pl) * 2009-12-30 2011-07-04 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Sposób otrzymywania wardenafilu i jego izolacji jako soli z kwasem cytrynowym oraz krystaliczna postać tej soli
CN102134242B (zh) 2011-01-21 2013-08-28 浙江大德药业集团有限公司 一种用于治疗阳痿的快速长效的化合物
CZ2011767A3 (cs) * 2011-11-24 2013-06-05 Zentiva, K.S. Zpusob prípravy a izolace solí vardenafilu s kyselinami
WO2015089105A1 (en) 2013-12-09 2015-06-18 Respira Therapeutics, Inc. Pde5 inhibitor powder formulations and methods relating thereto
PL223869B1 (pl) 2013-12-16 2016-11-30 Starogardzkie Zakłady Farm Polpharma Spółka Akcyjna Sposób otrzymywania wardenafilu i jego soli
CN107383020A (zh) * 2017-07-29 2017-11-24 合肥创新医药技术有限公司 一种伐地那非杂质的制备方法
CA3085219A1 (en) 2017-12-20 2019-06-27 Klaria Pharma Holding Ab Film formulation comprising vardenafil, method for its preparation, and use thereof
CN115043757B (zh) * 2022-07-27 2023-08-08 南京桦冠生物技术有限公司 一种连续化制备苄脒盐酸盐的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9301192D0 (en) * 1993-06-09 1993-06-09 Trott Francis W Flower shaped mechanised table
CH693954A5 (de) 1997-11-12 2004-05-14 Bayer Ag 2-Phenyl-substituierte Imidazotriazinone als Phosphodiesterase Inhibitoren.
DE10063108A1 (de) * 2000-12-18 2002-06-20 Bayer Ag Verfahren zur Herstellung von Sulfonamid-substituierten Imidazotriazinonen
DE10107639A1 (de) * 2001-02-15 2002-08-22 Bayer Ag 2-Alkoxyphenyl-substituierte Imidazotriazinone

Also Published As

Publication number Publication date
HUP0302467A3 (en) 2004-11-29
SK286894B6 (sk) 2009-07-06
DOP2001000295A (es) 2002-12-15
CZ297005B6 (cs) 2006-08-16
US20020137930A1 (en) 2002-09-26
JP2004517849A (ja) 2004-06-17
HK1063799A1 (en) 2005-01-14
NO325398B1 (no) 2008-04-21
CU23873B1 (es) 2013-04-19
UA75109C2 (en) 2006-03-15
CA2431933A1 (en) 2002-06-27
SV2003000766A (es) 2003-01-13
HU229296B1 (en) 2013-10-28
BR0116227B1 (pt) 2014-08-26
ATE328885T1 (de) 2006-06-15
WO2002050076A2 (de) 2002-06-27
UY27070A1 (es) 2002-07-31
NO20032731L (no) 2003-06-16
MA25927A1 (fr) 2003-10-01
HN2001000278A (es) 2002-01-30
HUP0302467A2 (hu) 2003-11-28
UY37172A (es) 2017-06-30
PE20020590A1 (es) 2002-07-13
NZ526477A (en) 2004-12-24
DE50110080D1 (de) 2006-07-20
RU2299211C2 (ru) 2007-05-20
DE10063108A1 (de) 2002-06-20
KR100787288B1 (ko) 2007-12-20
EP1345939B1 (de) 2006-06-07
SK7502003A3 (en) 2003-10-07
BRPI0116227B8 (pt) 2021-05-25
CY1105197T1 (el) 2010-03-03
TWI289562B (en) 2007-11-11
CN1481386A (zh) 2004-03-10
BG107892A (bg) 2004-08-31
CA2431933C (en) 2009-12-01
AU2002217089B2 (en) 2006-01-12
SI1345939T1 (sl) 2006-10-31
MXPA03005429A (es) 2004-05-04
US20050203298A1 (en) 2005-09-15
BG66142B1 (bg) 2011-07-29
HRP20030583A2 (en) 2005-06-30
ECSP034657A (es) 2003-07-25
US6777551B2 (en) 2004-08-17
ES2266098T3 (es) 2007-03-01
US20050014756A1 (en) 2005-01-20
BR0116227A (pt) 2003-12-30
EE05308B1 (et) 2010-06-15
US6998483B2 (en) 2006-02-14
WO2002050076A3 (de) 2002-08-29
MY126689A (en) 2006-10-31
AR032775A1 (es) 2003-11-26
CN1227253C (zh) 2005-11-16
CU23341B7 (es) 2009-02-20
DK1345939T3 (da) 2006-09-25
AU1708902A (en) 2002-07-01
KR20030063430A (ko) 2003-07-28
IL156278A (en) 2009-06-15
HRP20030583B1 (en) 2011-09-30
JP4441175B2 (ja) 2010-03-31
CZ20031692A3 (cs) 2003-10-15
PL207294B1 (pl) 2010-11-30
EP1345939A2 (de) 2003-09-24
CU20080213A7 (es) 2012-06-21
ZA200304705B (en) 2004-08-12
PL365310A1 (en) 2004-12-27
IL156278A0 (en) 2004-01-04
EE200300294A (et) 2003-10-15
NO20032731D0 (no) 2003-06-16
GT200100251A (es) 2002-10-01

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