PT1272489E - Processo para a preparacao da forma i cristalina de cabergolina - Google Patents

Processo para a preparacao da forma i cristalina de cabergolina

Info

Publication number
PT1272489E
PT1272489E PT01936098T PT01936098T PT1272489E PT 1272489 E PT1272489 E PT 1272489E PT 01936098 T PT01936098 T PT 01936098T PT 01936098 T PT01936098 T PT 01936098T PT 1272489 E PT1272489 E PT 1272489E
Authority
PT
Portugal
Prior art keywords
cabergolina
preparation
crystalline form
crystalline
Prior art date
Application number
PT01936098T
Other languages
English (en)
Inventor
Attilio Tomasi
Stefania Magenes
Mario Ungari
Giuliano Ramella
Gianfranco Pallanza
Original Assignee
Pharmacia Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9888433&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT1272489(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia Italia Spa filed Critical Pharmacia Italia Spa
Publication of PT1272489E publication Critical patent/PT1272489E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/04Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
    • C07D457/06Lysergic acid amides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/04Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16Masculine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
PT01936098T 2000-03-24 2001-03-19 Processo para a preparacao da forma i cristalina de cabergolina PT1272489E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0007308.0A GB0007308D0 (en) 2000-03-24 2000-03-24 Process for preparing crystalline form | of cabergoline

Publications (1)

Publication Number Publication Date
PT1272489E true PT1272489E (pt) 2004-02-27

Family

ID=9888433

Family Applications (1)

Application Number Title Priority Date Filing Date
PT01936098T PT1272489E (pt) 2000-03-24 2001-03-19 Processo para a preparacao da forma i cristalina de cabergolina

Country Status (31)

Country Link
US (2) US6727363B2 (pt)
EP (1) EP1272489B1 (pt)
JP (1) JP4184666B2 (pt)
KR (1) KR100827558B1 (pt)
CN (1) CN1188412C (pt)
AR (1) AR032449A1 (pt)
AT (1) ATE250601T1 (pt)
AU (2) AU780747B2 (pt)
BR (1) BR0109507A (pt)
CA (1) CA2402836A1 (pt)
CZ (1) CZ20023176A3 (pt)
DE (1) DE60100858T2 (pt)
DK (1) DK1272489T3 (pt)
EA (1) EA005928B1 (pt)
EE (1) EE05088B1 (pt)
ES (1) ES2208602T3 (pt)
GB (1) GB0007308D0 (pt)
HK (1) HK1052348B (pt)
HU (1) HUP0300591A3 (pt)
IL (2) IL150985A0 (pt)
MX (1) MXPA02009283A (pt)
MY (1) MY134189A (pt)
NO (1) NO20024321L (pt)
NZ (1) NZ521316A (pt)
PE (1) PE20011140A1 (pt)
PL (1) PL358253A1 (pt)
PT (1) PT1272489E (pt)
SI (1) SI1272489T1 (pt)
SK (1) SK13582002A3 (pt)
WO (1) WO2001070740A1 (pt)
ZA (1) ZA200206045B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0007307D0 (en) * 2000-03-24 2000-05-17 Pharmacia & Upjohn Spa Crystalline form || of cabergoline
GB0007308D0 (en) * 2000-03-24 2000-05-17 Pharmacia & Upjohn Spa Process for preparing crystalline form | of cabergoline
DE10053397A1 (de) * 2000-10-20 2002-05-02 Schering Ag Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen
DE10043321B4 (de) * 2000-08-24 2005-07-28 Neurobiotec Gmbh Verwendung eines transdermalen therapeutischen Systems zur Behandlung der Parkinsonschen Krankheit, zur Behandlung und Prävention des prämenstruellen Syndroms und zur Lactationshemmung
DE10064453A1 (de) * 2000-12-16 2002-07-04 Schering Ag Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen
AU2003218753A1 (en) * 2002-03-15 2003-09-29 Pharmacia Corporation Process for preparing crystalline form i of cabergoline
EP1507777A4 (en) * 2002-03-15 2007-03-07 Pharmacia Corp PROCESS FOR THE PREPARATION OF A CRYSTALLINE FORM I OF CABERGOLIN
IL155545A (en) * 2003-04-21 2009-12-24 Finetech Pharmaceutical Ltd Solvate form of cabergoline
CA2525104A1 (en) 2003-05-08 2004-11-25 Ivax Pharmaceuticals S.R.O. Polymorphs of cabergoline
GB0409785D0 (en) * 2004-04-30 2004-06-09 Resolution Chemicals Ltd Preparation of cabergoline
GB0515430D0 (en) * 2005-07-27 2005-08-31 Resolution Chemicals Ltd Preparation of cabergoline
US7339060B2 (en) * 2005-03-23 2008-03-04 Resolution Chemicals, Ltd. Preparation of cabergoline
GB0505965D0 (en) 2005-03-23 2005-04-27 Resolution Chemicals Ltd Preparation of cabergoline
EP1925616A1 (en) * 2006-10-26 2008-05-28 LEK Pharmaceuticals D.D. Process for the preparation of crystal forms of cabergoline via stable solvates of cabergoline
EP1953157A1 (en) 2007-01-31 2008-08-06 LEK Pharmaceuticals D.D. New crystal form of cabergoline
US8637099B2 (en) * 2007-08-29 2014-01-28 Max Zeller Sohne Ag Use of Vitex agnus castus extracts for preparing a medicament
EP4074552B1 (en) * 2021-04-16 2024-04-03 Thermo King LLC Electrical connection unit

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3019322A1 (de) 1980-05-21 1981-12-03 Merck Patent Gmbh, 6100 Darmstadt Psychopharmakon sowie verwendung von adenosinderivaten
US4526892A (en) * 1981-03-03 1985-07-02 Farmitalia Carlo Erba, S.P.A. Dimethylaminoalkyl-3-(ergoline-8'βcarbonyl)-ureas
GB2103603B (en) 1981-08-11 1985-04-11 Erba Farmitalia Ergoline derivatives
GB9205439D0 (en) 1992-03-12 1992-04-22 Erba Carlo Spa Process for the synthesis of ergoline derivatives
EP0664705B1 (en) 1993-08-18 2000-10-04 Alcon Laboratories, Inc. Compositions of ergoline derivatives for the treatment of glaucoma
EP1075278A1 (en) 1998-01-13 2001-02-14 AstraZeneca UK Limited PHARMACEUTICAL COMPOSITIONS COMPRISING A COMPOUND HAVING DOPAMINE (D 2?) RECEPTOR AGONIST ACTIVITY AND A COMPOUND (B) HAVING $g(b) 2?-ADRENORECEPTOR AGONIST ACTIVITY
BR9908953A (pt) 1998-03-27 2000-12-05 Upjohn Co Utilização de cabergolina no tratamento da sìndrome de pernas agitadas (sìndrome de ekbom)
GB0007309D0 (en) 2000-03-24 2000-05-17 Pharmacia & Upjohn Spa Crystalline form V|| of cabergoline
GB0007307D0 (en) 2000-03-24 2000-05-17 Pharmacia & Upjohn Spa Crystalline form || of cabergoline
GB0007308D0 (en) 2000-03-24 2000-05-17 Pharmacia & Upjohn Spa Process for preparing crystalline form | of cabergoline

Also Published As

Publication number Publication date
MY134189A (en) 2007-11-30
US6953854B2 (en) 2005-10-11
GB0007308D0 (en) 2000-05-17
MXPA02009283A (es) 2003-03-12
EA200201016A1 (ru) 2003-02-27
NO20024321D0 (no) 2002-09-10
CN1419554A (zh) 2003-05-21
NZ521316A (en) 2004-05-28
AU780747B2 (en) 2005-04-14
SI1272489T1 (en) 2004-02-29
EP1272489A1 (en) 2003-01-08
HK1052348B (zh) 2005-09-16
EA005928B1 (ru) 2005-08-25
ZA200206045B (en) 2003-07-29
CZ20023176A3 (cs) 2003-02-12
EE200200545A (et) 2004-04-15
US20030149067A1 (en) 2003-08-07
AU2005203071B2 (en) 2007-10-18
PL358253A1 (en) 2004-08-09
PE20011140A1 (es) 2001-11-01
AU2005203071A1 (en) 2005-08-11
AR032449A1 (es) 2003-11-12
DK1272489T3 (da) 2003-12-15
HUP0300591A3 (en) 2009-01-28
HUP0300591A2 (hu) 2003-07-28
JP2003528100A (ja) 2003-09-24
ES2208602T3 (es) 2004-06-16
SK13582002A3 (sk) 2003-04-01
JP4184666B2 (ja) 2008-11-19
US6727363B2 (en) 2004-04-27
HK1052348A1 (en) 2003-09-11
DE60100858T2 (de) 2004-07-29
AU6211001A (en) 2001-10-03
NO20024321L (no) 2002-09-10
EE05088B1 (et) 2008-10-15
KR20020081587A (ko) 2002-10-28
KR100827558B1 (ko) 2008-05-07
IL150985A (en) 2007-03-08
ATE250601T1 (de) 2003-10-15
IL150985A0 (en) 2003-02-12
US20040092744A1 (en) 2004-05-13
BR0109507A (pt) 2002-12-10
CA2402836A1 (en) 2001-09-27
CN1188412C (zh) 2005-02-09
WO2001070740A1 (en) 2001-09-27
EP1272489B1 (en) 2003-09-24
DE60100858D1 (de) 2003-10-30

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