PT1281707E - Processo para a preparacao de isobenzofuranos 5-substituidos - Google Patents

Processo para a preparacao de isobenzofuranos 5-substituidos

Info

Publication number
PT1281707E
PT1281707E PT01830517T PT01830517T PT1281707E PT 1281707 E PT1281707 E PT 1281707E PT 01830517 T PT01830517 T PT 01830517T PT 01830517 T PT01830517 T PT 01830517T PT 1281707 E PT1281707 E PT 1281707E
Authority
PT
Portugal
Prior art keywords
isobenzofuranes
substituted
preparation
substituted isobenzofuranes
Prior art date
Application number
PT01830517T
Other languages
English (en)
Inventor
Giovanni Cotticelli
Dall Asta Leone
Original Assignee
Infosint Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Infosint Sa filed Critical Infosint Sa
Publication of PT1281707E publication Critical patent/PT1281707E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32Oximes
    • C07C251/34Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT01830517T 2001-08-02 2001-08-02 Processo para a preparacao de isobenzofuranos 5-substituidos PT1281707E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01830517A EP1281707B1 (en) 2001-08-02 2001-08-02 Process for the preparation of 5-subtituted isobenzofurans

Publications (1)

Publication Number Publication Date
PT1281707E true PT1281707E (pt) 2005-04-29

Family

ID=8184643

Family Applications (1)

Application Number Title Priority Date Filing Date
PT01830517T PT1281707E (pt) 2001-08-02 2001-08-02 Processo para a preparacao de isobenzofuranos 5-substituidos

Country Status (23)

Country Link
US (1) US7166729B2 (pt)
EP (1) EP1281707B1 (pt)
JP (1) JP2005501056A (pt)
KR (1) KR20040043176A (pt)
CN (1) CN1298713C (pt)
AR (1) AR036212A1 (pt)
AT (1) ATE286037T1 (pt)
AU (1) AU2002325385B2 (pt)
BG (1) BG108554A (pt)
BR (1) BR0211858A (pt)
CA (1) CA2456004A1 (pt)
DE (1) DE60108105T2 (pt)
DK (1) DK1281707T3 (pt)
ES (1) ES2234797T3 (pt)
HK (1) HK1070357A1 (pt)
HU (1) HUP0401166A3 (pt)
MX (1) MXPA04001030A (pt)
PL (1) PL368320A1 (pt)
PT (1) PT1281707E (pt)
RO (1) RO122147B1 (pt)
TW (1) TWI225055B (pt)
WO (1) WO2003011846A2 (pt)
ZA (1) ZA200400841B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IS7239A (is) * 2001-12-14 2004-04-29 H. Lundbeck A/S Aðferð til framleiðslu á essítalóprami
AU2003263155A1 (en) * 2002-09-20 2004-04-08 H. Lundbeck A/S Method for manufacture of dihydroisobenzofuran derivatives
GB0601286D0 (en) * 2006-01-23 2006-03-01 Sandoz Ag Asymmetric synthesis
WO2009073620A2 (en) 2007-11-30 2009-06-11 Newlink Genetics Ido inhibitors
CN106632182A (zh) * 2016-12-07 2017-05-10 万全万特制药(厦门)有限公司 草酸艾司西酞普兰脱甲基杂质的制备方法
CN113784945A (zh) * 2018-12-22 2021-12-10 马拉迪制药有限公司 制备R-苯基乙酰基甲醇和β-氨基醇的新方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8419963D0 (en) * 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
JP3526581B2 (ja) * 1997-07-08 2004-05-17 ハー・ルンドベック・アクティーゼルスカブ シタロプラムの製造方法
ATE237604T1 (de) * 1999-04-14 2003-05-15 Lundbeck & Co As H Verfahren zur herstellung von citalopram
ITMI991486A1 (it) * 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
IES20010143A2 (en) * 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
IT1319686B1 (it) * 2000-12-12 2003-10-23 C D Farmasint S R L Procedimento di preparazione di citalopram.

Also Published As

Publication number Publication date
HUP0401166A2 (hu) 2004-09-28
AR036212A1 (es) 2004-08-18
DE60108105D1 (de) 2005-02-03
CN1555370A (zh) 2004-12-15
DK1281707T3 (da) 2005-05-02
WO2003011846B1 (en) 2003-12-24
DE60108105T2 (de) 2005-12-08
BR0211858A (pt) 2004-09-21
HUP0401166A3 (en) 2007-05-29
ATE286037T1 (de) 2005-01-15
US7166729B2 (en) 2007-01-23
AU2002325385B2 (en) 2007-07-05
CN1298713C (zh) 2007-02-07
US20040230065A1 (en) 2004-11-18
KR20040043176A (ko) 2004-05-22
RO122147B1 (ro) 2009-01-30
WO2003011846A2 (en) 2003-02-13
BG108554A (bg) 2005-03-31
ZA200400841B (en) 2005-02-02
MXPA04001030A (es) 2004-12-03
HK1070357A1 (en) 2005-06-17
EP1281707A1 (en) 2003-02-05
ES2234797T3 (es) 2005-07-01
AU2002325385B8 (en) 2003-02-17
TWI225055B (en) 2004-12-11
PL368320A1 (en) 2005-03-21
EP1281707B1 (en) 2004-12-29
WO2003011846A3 (en) 2003-11-27
CA2456004A1 (en) 2003-02-13
JP2005501056A (ja) 2005-01-13

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