BG108554A - Метод за получаване на 5-заместени изобензофурани - Google Patents

Метод за получаване на 5-заместени изобензофурани Download PDF

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Publication number
BG108554A
BG108554A BG108554A BG10855404A BG108554A BG 108554 A BG108554 A BG 108554A BG 108554 A BG108554 A BG 108554A BG 10855404 A BG10855404 A BG 10855404A BG 108554 A BG108554 A BG 108554A
Authority
BG
Bulgaria
Prior art keywords
formula
group
triphenylmethyl
citalopram
alkyl
Prior art date
Application number
BG108554A
Other languages
Bulgarian (bg)
English (en)
Inventor
Leone Dall'asta
Giovanni Coticelli
Original Assignee
Infosint Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Infosint Sa filed Critical Infosint Sa
Publication of BG108554A publication Critical patent/BG108554A/bg

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32Oximes
    • C07C251/34Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG108554A 2001-08-02 2004-01-30 Метод за получаване на 5-заместени изобензофурани BG108554A (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01830517A EP1281707B1 (en) 2001-08-02 2001-08-02 Process for the preparation of 5-subtituted isobenzofurans

Publications (1)

Publication Number Publication Date
BG108554A true BG108554A (bg) 2005-03-31

Family

ID=8184643

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108554A BG108554A (bg) 2001-08-02 2004-01-30 Метод за получаване на 5-заместени изобензофурани

Country Status (23)

Country Link
US (1) US7166729B2 (pt)
EP (1) EP1281707B1 (pt)
JP (1) JP2005501056A (pt)
KR (1) KR20040043176A (pt)
CN (1) CN1298713C (pt)
AR (1) AR036212A1 (pt)
AT (1) ATE286037T1 (pt)
AU (1) AU2002325385B2 (pt)
BG (1) BG108554A (pt)
BR (1) BR0211858A (pt)
CA (1) CA2456004A1 (pt)
DE (1) DE60108105T2 (pt)
DK (1) DK1281707T3 (pt)
ES (1) ES2234797T3 (pt)
HK (1) HK1070357A1 (pt)
HU (1) HUP0401166A3 (pt)
MX (1) MXPA04001030A (pt)
PL (1) PL368320A1 (pt)
PT (1) PT1281707E (pt)
RO (1) RO122147B1 (pt)
TW (1) TWI225055B (pt)
WO (1) WO2003011846A2 (pt)
ZA (1) ZA200400841B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IS7239A (is) * 2001-12-14 2004-04-29 H. Lundbeck A/S Aðferð til framleiðslu á essítalóprami
AU2003263155A1 (en) * 2002-09-20 2004-04-08 H. Lundbeck A/S Method for manufacture of dihydroisobenzofuran derivatives
GB0601286D0 (en) * 2006-01-23 2006-03-01 Sandoz Ag Asymmetric synthesis
WO2009073620A2 (en) 2007-11-30 2009-06-11 Newlink Genetics Ido inhibitors
CN106632182A (zh) * 2016-12-07 2017-05-10 万全万特制药(厦门)有限公司 草酸艾司西酞普兰脱甲基杂质的制备方法
CN113784945A (zh) * 2018-12-22 2021-12-10 马拉迪制药有限公司 制备R-苯基乙酰基甲醇和β-氨基醇的新方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8419963D0 (en) * 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
JP3526581B2 (ja) * 1997-07-08 2004-05-17 ハー・ルンドベック・アクティーゼルスカブ シタロプラムの製造方法
ATE237604T1 (de) * 1999-04-14 2003-05-15 Lundbeck & Co As H Verfahren zur herstellung von citalopram
ITMI991486A1 (it) * 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
IES20010143A2 (en) * 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
IT1319686B1 (it) * 2000-12-12 2003-10-23 C D Farmasint S R L Procedimento di preparazione di citalopram.

Also Published As

Publication number Publication date
HUP0401166A2 (hu) 2004-09-28
AR036212A1 (es) 2004-08-18
DE60108105D1 (de) 2005-02-03
CN1555370A (zh) 2004-12-15
DK1281707T3 (da) 2005-05-02
WO2003011846B1 (en) 2003-12-24
DE60108105T2 (de) 2005-12-08
BR0211858A (pt) 2004-09-21
HUP0401166A3 (en) 2007-05-29
ATE286037T1 (de) 2005-01-15
US7166729B2 (en) 2007-01-23
AU2002325385B2 (en) 2007-07-05
CN1298713C (zh) 2007-02-07
US20040230065A1 (en) 2004-11-18
KR20040043176A (ko) 2004-05-22
RO122147B1 (ro) 2009-01-30
WO2003011846A2 (en) 2003-02-13
PT1281707E (pt) 2005-04-29
ZA200400841B (en) 2005-02-02
MXPA04001030A (es) 2004-12-03
HK1070357A1 (en) 2005-06-17
EP1281707A1 (en) 2003-02-05
ES2234797T3 (es) 2005-07-01
AU2002325385B8 (en) 2003-02-17
TWI225055B (en) 2004-12-11
PL368320A1 (en) 2005-03-21
EP1281707B1 (en) 2004-12-29
WO2003011846A3 (en) 2003-11-27
CA2456004A1 (en) 2003-02-13
JP2005501056A (ja) 2005-01-13

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