PL363264A1 - Pochodne izoksazoliny jako środki przeciwdepresyjne - Google Patents
Pochodne izoksazoliny jako środki przeciwdepresyjneInfo
- Publication number
- PL363264A1 PL363264A1 PL02363264A PL36326402A PL363264A1 PL 363264 A1 PL363264 A1 PL 363264A1 PL 02363264 A PL02363264 A PL 02363264A PL 36326402 A PL36326402 A PL 36326402A PL 363264 A1 PL363264 A1 PL 363264A1
- Authority
- PL
- Poland
- Prior art keywords
- depressants
- isoxazoline derivatives
- isoxazoline
- derivatives
- Prior art date
Links
- 230000001430 anti-depressive effect Effects 0.000 title 1
- 239000000935 antidepressant agent Substances 0.000 title 1
- 229940005513 antidepressants Drugs 0.000 title 1
- 150000002547 isoxazolines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01200611 | 2001-02-21 | ||
| EP01201264 | 2001-04-05 | ||
| PCT/EP2002/001567 WO2002066484A1 (en) | 2001-02-21 | 2002-02-13 | Isoxazoline derivatives as anti-depressants |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL363264A1 true PL363264A1 (pl) | 2004-11-15 |
| PL208593B1 PL208593B1 (pl) | 2011-05-31 |
Family
ID=26076836
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL363264A PL208593B1 (pl) | 2001-02-21 | 2002-02-13 | Pochodne izoksazoliny, kompozycja farmaceutyczna je zawierająca oraz ich zastosowanie |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US7169786B2 (pl) |
| EP (1) | EP1368358B1 (pl) |
| JP (1) | JP3953424B2 (pl) |
| KR (1) | KR100848898B1 (pl) |
| CN (1) | CN100400540C (pl) |
| AR (1) | AR035685A1 (pl) |
| AT (1) | ATE337322T1 (pl) |
| AU (1) | AU2002244717B2 (pl) |
| BG (1) | BG107984A (pl) |
| BR (1) | BR0207433A (pl) |
| CA (1) | CA2437505C (pl) |
| CY (1) | CY1106448T1 (pl) |
| CZ (1) | CZ20032515A3 (pl) |
| DE (1) | DE60214138T2 (pl) |
| DK (1) | DK1368358T3 (pl) |
| EA (1) | EA006747B1 (pl) |
| EE (1) | EE200300398A (pl) |
| EG (1) | EG23929A (pl) |
| ES (1) | ES2271230T3 (pl) |
| HR (1) | HRP20030647A2 (pl) |
| HU (1) | HUP0303270A3 (pl) |
| IL (2) | IL157470A0 (pl) |
| MX (1) | MXPA03007432A (pl) |
| MY (1) | MY137836A (pl) |
| NO (1) | NO20033700L (pl) |
| NZ (1) | NZ526741A (pl) |
| PL (1) | PL208593B1 (pl) |
| PT (1) | PT1368358E (pl) |
| SI (1) | SI1368358T1 (pl) |
| SK (1) | SK11612003A3 (pl) |
| TW (1) | TWI257392B (pl) |
| WO (1) | WO2002066484A1 (pl) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0203299D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel compounds |
| KR20040093061A (ko) * | 2002-04-02 | 2004-11-04 | 얀센 파마슈티카 엔.브이. | 치환된 아미노 이속사졸린 유도체 및 항-우울제로서의그의 용도 |
| TW200409777A (en) | 2002-08-12 | 2004-06-16 | Janssen Pharmaceutica Nv | C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants |
| DE60331160D1 (de) * | 2002-08-15 | 2010-03-18 | Janssen Pharmaceutica Nv | Kondensierte heterocyclische isoxazolinderivate und deren verwendung als antidepressiva |
| EP1532155B1 (en) * | 2002-08-21 | 2008-02-27 | Janssen Pharmaceutica N.V. | C6- AND C9-SUBSTITUTED CHROMENO[4,3-c]ISOXAZOLINE DERIVATIVES AND THEIR USE AS ANTI-DEPRESSANTS |
| WO2004078715A1 (ja) * | 2003-03-07 | 2004-09-16 | Astellas Pharma Inc. | 2,6-ジ置換スチリルを有する含窒素へテロ環誘導体 |
| CN103788089A (zh) | 2003-09-17 | 2014-05-14 | 詹森药业有限公司 | 作为血清素受体调节剂的稠合杂环化合物 |
| EP1944306A1 (en) * | 2003-09-17 | 2008-07-16 | Janssen Pharmaceutica, N.V. | Fused heterocyclic compounds as serotonin receptor modulators |
| CA2585857A1 (en) * | 2004-11-26 | 2006-06-01 | Janssen Pharmaceutica N.V. | Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic activity |
| NZ579431A (en) * | 2007-03-09 | 2012-04-27 | Sanofi Aventis | Substituted dihydro and tetrahydro oxazolopyrimidinones, preparation and use thereof |
| MX2009013205A (es) * | 2007-06-08 | 2010-04-09 | Helicon Therapeutics Inc | Derivados de pirazoloquinolina urea terapeuticos. |
| WO2009082268A2 (ru) | 2007-12-21 | 2009-07-02 | Alla Chem, Llc | ЛИГАНДЫ α-АДРЕНОЦЕПТОРОВ, ДОПАМИНОВЫХ, ГИСТАМИНОВЫХ, ИМИДАЗОЛИНОВЫХ И СЕРОТОНИНОВЫХ РЕЦЕПТОРОВ И ИХ ПРИМЕНЕНИЕ |
| AR078171A1 (es) | 2009-09-15 | 2011-10-19 | Sanofi Aventis | Dihidrobenzocicloalquiloximetil-oxazolopirimidinonas sustituidas, preparacion y uso de las mismas |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0361577B1 (en) * | 1988-09-19 | 1993-05-05 | Akzo N.V. | Tetrahydronaphthalene and indane derivatives |
| US5880121A (en) * | 1996-01-05 | 1999-03-09 | Hoechst Marion Roussel Inc. | 4,5-dihydronaphth (1,2-c) isoxazoles and derivatives thereof |
| PT892804E (pt) * | 1996-04-12 | 2003-01-31 | Janssen Pharmaceutica Nv | Derivados de isoxazolidina |
| HUP9602763A3 (en) * | 1996-10-09 | 1999-05-28 | Egyt Gyogyszervegyeszeti Gyar | 3-phenyl isoxazole derivatives, process for producing them and pharmaceutical compositions containing the same |
| EP1119568B1 (en) * | 1998-10-09 | 2004-02-18 | Janssen Pharmaceutica N.V. | 4,5-dihydro-isoxazole derivatives and their pharmaceutical use |
-
2002
- 2002-02-13 HU HU0303270A patent/HUP0303270A3/hu unknown
- 2002-02-13 AT AT02712909T patent/ATE337322T1/de not_active IP Right Cessation
- 2002-02-13 DK DK02712909T patent/DK1368358T3/da active
- 2002-02-13 CA CA2437505A patent/CA2437505C/en not_active Expired - Lifetime
- 2002-02-13 EP EP02712909A patent/EP1368358B1/en not_active Expired - Lifetime
- 2002-02-13 BR BR0207433-8A patent/BR0207433A/pt not_active IP Right Cessation
- 2002-02-13 WO PCT/EP2002/001567 patent/WO2002066484A1/en not_active Ceased
- 2002-02-13 CZ CZ20032515A patent/CZ20032515A3/cs unknown
- 2002-02-13 CN CNB028052439A patent/CN100400540C/zh not_active Expired - Fee Related
- 2002-02-13 SI SI200230433T patent/SI1368358T1/sl unknown
- 2002-02-13 US US10/468,555 patent/US7169786B2/en not_active Expired - Lifetime
- 2002-02-13 HR HR20030647A patent/HRP20030647A2/hr not_active Application Discontinuation
- 2002-02-13 PT PT02712909T patent/PT1368358E/pt unknown
- 2002-02-13 IL IL15747002A patent/IL157470A0/xx unknown
- 2002-02-13 KR KR1020037008328A patent/KR100848898B1/ko not_active Expired - Fee Related
- 2002-02-13 JP JP2002565998A patent/JP3953424B2/ja not_active Expired - Lifetime
- 2002-02-13 SK SK1161-2003A patent/SK11612003A3/sk unknown
- 2002-02-13 ES ES02712909T patent/ES2271230T3/es not_active Expired - Lifetime
- 2002-02-13 EE EEP200300398A patent/EE200300398A/xx unknown
- 2002-02-13 MX MXPA03007432A patent/MXPA03007432A/es active IP Right Grant
- 2002-02-13 DE DE60214138T patent/DE60214138T2/de not_active Expired - Lifetime
- 2002-02-13 AU AU2002244717A patent/AU2002244717B2/en not_active Expired
- 2002-02-13 EA EA200300915A patent/EA006747B1/ru not_active IP Right Cessation
- 2002-02-13 NZ NZ526741A patent/NZ526741A/en unknown
- 2002-02-13 PL PL363264A patent/PL208593B1/pl unknown
- 2002-02-19 MY MYPI20020548A patent/MY137836A/en unknown
- 2002-02-19 EG EG20020197A patent/EG23929A/xx active
- 2002-02-20 TW TW091102853A patent/TWI257392B/zh not_active IP Right Cessation
- 2002-02-20 AR ARP020100583A patent/AR035685A1/es unknown
-
2003
- 2003-07-08 BG BG107984A patent/BG107984A/bg unknown
- 2003-08-19 IL IL157470A patent/IL157470A/en unknown
- 2003-08-20 NO NO20033700A patent/NO20033700L/no not_active Application Discontinuation
-
2006
- 2006-11-22 CY CY20061101693T patent/CY1106448T1/el unknown
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