PE20211657A1 - Composiciones terapeuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato - Google Patents

Composiciones terapeuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato

Info

Publication number
PE20211657A1
PE20211657A1 PE2021000720A PE2021000720A PE20211657A1 PE 20211657 A1 PE20211657 A1 PE 20211657A1 PE 2021000720 A PE2021000720 A PE 2021000720A PE 2021000720 A PE2021000720 A PE 2021000720A PE 20211657 A1 PE20211657 A1 PE 20211657A1
Authority
PE
Peru
Prior art keywords
tablet
tenofovir disoproxil
disoproxil fumarate
hcl
rilpivirin
Prior art date
Application number
PE2021000720A
Other languages
English (en)
Spanish (es)
Inventor
Reza Oliyai
Lauren Wiser
Mark Menning
Original Assignee
Gilead Sciences Inc
Janssen Sciences Ireland Uc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45094284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20211657(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc, Janssen Sciences Ireland Uc filed Critical Gilead Sciences Inc
Publication of PE20211657A1 publication Critical patent/PE20211657A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PE2021000720A 2010-11-19 2011-11-18 Composiciones terapeuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato PE20211657A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41560010P 2010-11-19 2010-11-19
PCT/US2011/061515 WO2012068535A1 (en) 2010-11-19 2011-11-18 Therapeutic compositions comprising rilpivirine hcl and tenofovir disoproxil fumarate

Publications (1)

Publication Number Publication Date
PE20211657A1 true PE20211657A1 (es) 2021-08-24

Family

ID=45094284

Family Applications (3)

Application Number Title Priority Date Filing Date
PE2021000720A PE20211657A1 (es) 2010-11-19 2011-11-18 Composiciones terapeuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato
PE2013001214A PE20140163A1 (es) 2010-11-19 2011-11-18 Composiciones terapeuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato
PE2016002828A PE20170521A1 (es) 2010-11-19 2011-11-18 Combinacion farmaceutica que comprende rilpivirina hcl, tenofovir disoproxil fumarato y emtricitabina

Family Applications After (2)

Application Number Title Priority Date Filing Date
PE2013001214A PE20140163A1 (es) 2010-11-19 2011-11-18 Composiciones terapeuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato
PE2016002828A PE20170521A1 (es) 2010-11-19 2011-11-18 Combinacion farmaceutica que comprende rilpivirina hcl, tenofovir disoproxil fumarato y emtricitabina

Country Status (36)

Country Link
US (1) US10857102B2 (enExample)
EP (2) EP2826466A1 (enExample)
JP (2) JP2014500261A (enExample)
KR (1) KR101923103B1 (enExample)
CN (2) CN103491948B (enExample)
AP (1) AP3816A (enExample)
AR (2) AR084500A1 (enExample)
AU (3) AU2011329642B2 (enExample)
BR (1) BR112013012245B1 (enExample)
CA (1) CA2818097C (enExample)
CL (1) CL2013001402A1 (enExample)
CO (1) CO6761300A2 (enExample)
CR (1) CR20130293A (enExample)
DK (1) DK2640362T4 (enExample)
EA (2) EA201691695A1 (enExample)
EC (2) ECSP13012700A (enExample)
ES (1) ES2524408T5 (enExample)
HK (1) HK1206592A1 (enExample)
HR (1) HRP20140946T1 (enExample)
IL (1) IL226300B (enExample)
MA (1) MA34735B1 (enExample)
ME (1) ME01980B (enExample)
MX (1) MX347512B (enExample)
MY (1) MY185604A (enExample)
NZ (1) NZ610729A (enExample)
PE (3) PE20211657A1 (enExample)
PH (1) PH12013501002A1 (enExample)
PL (1) PL2640362T5 (enExample)
PT (1) PT2640362E (enExample)
RS (1) RS53691B1 (enExample)
SG (3) SG10201509521WA (enExample)
SM (1) SMT201400150B (enExample)
TW (1) TWI556840B (enExample)
UA (1) UA114075C2 (enExample)
WO (1) WO2012068535A1 (enExample)
ZA (1) ZA201304481B (enExample)

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TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
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KR20170003063A (ko) * 2015-06-30 2017-01-09 한미약품 주식회사 테노포비어 디소프록실 함유 경구용 고형제제 및 그 제조방법
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US10561614B2 (en) * 2017-01-27 2020-02-18 Steerlife India Private Limited Tenofovir granules
RU2755710C2 (ru) * 2017-06-30 2021-09-20 Вайв Хелткер Компани Комбинация, ее применение и способы лечения с использованием указанной комбинации
LT3706762T (lt) 2017-12-07 2024-12-27 Emory University N4-hidroksicitidinas ir jo dariniai bei susiję naudojimo prieš virusus būdai
CN114126655A (zh) * 2019-07-03 2022-03-01 爱尔兰詹森科学公司 用利匹韦林治疗儿科患者的hiv的方法
CN112137981A (zh) * 2020-11-02 2020-12-29 成都晶富医药科技有限公司 富马酸丙酚替诺福韦片及其制备工艺
WO2024211882A1 (en) * 2023-04-07 2024-10-10 Navinta, Llc Stable compositions of rilpivirine hcl in combination with other anti-retroviral agents
CN119174735A (zh) * 2024-09-03 2024-12-24 安徽贝克生物制药有限公司 一种含利匹韦林的复方片及制备方法

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Also Published As

Publication number Publication date
AU2011329642A1 (en) 2013-05-02
HK1206592A1 (en) 2016-01-15
TW201238612A (en) 2012-10-01
MX347512B (es) 2017-04-28
DK2640362T4 (da) 2022-03-07
ECSP19078196A (es) 2019-11-30
SG10201509521WA (en) 2015-12-30
CN103491948B (zh) 2016-11-02
AU2011329642B2 (en) 2016-08-11
CN106511357A (zh) 2017-03-22
PH12013501002A1 (en) 2013-09-09
EA201390651A1 (ru) 2013-11-29
AU2016208417B2 (en) 2018-04-05
AP3816A (en) 2016-09-30
MY185604A (en) 2021-05-25
EA201691695A1 (ru) 2017-11-30
DK2640362T3 (en) 2014-12-01
CN103491948A (zh) 2014-01-01
AR084500A1 (es) 2013-05-22
EA025852B1 (ru) 2017-02-28
CR20130293A (es) 2013-10-03
US10857102B2 (en) 2020-12-08
PL2640362T5 (pl) 2022-05-02
EP2640362B2 (en) 2021-12-01
JP2015131853A (ja) 2015-07-23
AR123409A2 (es) 2022-11-30
KR20140037799A (ko) 2014-03-27
EP2640362A1 (en) 2013-09-25
ES2524408T3 (es) 2014-12-09
CL2013001402A1 (es) 2013-12-27
MX2013005669A (es) 2013-11-04
PT2640362E (pt) 2014-11-28
JP6138851B2 (ja) 2017-05-31
EP2826466A1 (en) 2015-01-21
HRP20140946T1 (hr) 2015-02-13
CA2818097A1 (en) 2012-05-24
IL226300B (en) 2019-05-30
AP2013006931A0 (en) 2013-06-30
SMT201400150B (it) 2015-01-15
RS53691B1 (sr) 2015-04-30
WO2012068535A1 (en) 2012-05-24
EP2640362B1 (en) 2014-09-10
PE20170521A1 (es) 2017-05-27
CA2818097C (en) 2019-07-30
AU2018202635A1 (en) 2018-05-10
ECSP13012700A (es) 2013-08-30
BR112013012245B1 (pt) 2022-09-27
ZA201304481B (en) 2022-03-30
NZ610729A (en) 2015-10-30
CO6761300A2 (es) 2013-09-30
TWI556840B (zh) 2016-11-11
JP2014500261A (ja) 2014-01-09
HK1190064A1 (en) 2014-06-27
PL2640362T3 (pl) 2015-03-31
MA34735B1 (fr) 2013-12-03
SG190333A1 (en) 2013-06-28
UA114075C2 (xx) 2017-04-25
ME01980B (me) 2015-05-20
PE20140163A1 (es) 2014-02-08
US20130243857A1 (en) 2013-09-19
ES2524408T5 (es) 2022-04-25
BR112013012245A2 (pt) 2016-08-09
KR101923103B1 (ko) 2018-11-28
SG10201912527XA (en) 2020-02-27
AU2016208417A1 (en) 2016-08-18

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