OA12050A - Certain alkylene diamine-substituted heterocycles. - Google Patents

Certain alkylene diamine-substituted heterocycles. Download PDF

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Publication number
OA12050A
OA12050A OA1200200089A OA1200200089A OA12050A OA 12050 A OA12050 A OA 12050A OA 1200200089 A OA1200200089 A OA 1200200089A OA 1200200089 A OA1200200089 A OA 1200200089A OA 12050 A OA12050 A OA 12050A
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OA
OAPI
Prior art keywords
methylene
compound
formula
hydrogen
alkyl
Prior art date
Application number
OA1200200089A
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English (en)
Inventor
Raymond E Horvath
Jennifer Tran
Stephane De Lombaert
Kevin Julian Hodgetts
Philip A Carpino
David A Griffith
Original Assignee
Neurogen Corp
Pfizer
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Publication date
Application filed by Neurogen Corp, Pfizer filed Critical Neurogen Corp
Publication of OA12050A publication Critical patent/OA12050A/en

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/73—Unsubstituted amino or imino radicals
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    • C07D215/38—Nitrogen atoms
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  • Psychiatry (AREA)
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OA1200200089A 1999-09-30 2000-09-29 Certain alkylene diamine-substituted heterocycles. OA12050A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15687099P 1999-09-30 1999-09-30

Publications (1)

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OA12050A true OA12050A (en) 2006-05-02

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OA1200200089A OA12050A (en) 1999-09-30 2000-09-29 Certain alkylene diamine-substituted heterocycles.

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US (3) US6506762B1 (fr)
EP (1) EP1224187B1 (fr)
JP (2) JP2003510327A (fr)
KR (1) KR20020043223A (fr)
CN (1) CN1377356A (fr)
AT (1) ATE318267T1 (fr)
AU (1) AU7738000A (fr)
BG (1) BG106508A (fr)
CA (1) CA2379640C (fr)
CZ (1) CZ20021086A3 (fr)
DE (1) DE60026155T2 (fr)
EA (1) EA200200424A1 (fr)
ES (1) ES2258476T3 (fr)
HU (1) HUP0202636A3 (fr)
IL (1) IL148903A0 (fr)
NO (1) NO20021358L (fr)
NZ (1) NZ517575A (fr)
OA (1) OA12050A (fr)
PL (1) PL354784A1 (fr)
WO (1) WO2001023389A2 (fr)
ZA (1) ZA200202518B (fr)

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US20030158197A1 (en) 2003-08-21
CA2379640A1 (fr) 2001-04-05
PL354784A1 (en) 2004-02-23
WO2001023389A3 (fr) 2002-05-10
DE60026155D1 (de) 2006-04-27
AU7738000A (en) 2001-04-30
DE60026155T2 (de) 2006-08-10
EA200200424A1 (ru) 2002-12-26
HUP0202636A3 (en) 2004-06-28
US20040229870A1 (en) 2004-11-18
JP2008007515A (ja) 2008-01-17
CZ20021086A3 (cs) 2002-10-16
US6506762B1 (en) 2003-01-14
WO2001023389A2 (fr) 2001-04-05
CN1377356A (zh) 2002-10-30
IL148903A0 (en) 2002-09-12
JP2003510327A (ja) 2003-03-18
EP1224187A2 (fr) 2002-07-24
US6696445B2 (en) 2004-02-24
US7074929B2 (en) 2006-07-11
ZA200202518B (en) 2003-08-27
NO20021358D0 (no) 2002-03-19
KR20020043223A (ko) 2002-06-08
BG106508A (en) 2003-02-28
ES2258476T3 (es) 2006-09-01
ATE318267T1 (de) 2006-03-15
NZ517575A (en) 2004-04-30
EP1224187B1 (fr) 2006-02-22

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