OA10488A - Conjugué peg-ifn alpha physiologiquement actif procédé pour sa préparation compositions pharmaceutiques le contenant et leur utilisation - Google Patents

Conjugué peg-ifn alpha physiologiquement actif procédé pour sa préparation compositions pharmaceutiques le contenant et leur utilisation Download PDF

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Publication number
OA10488A
OA10488A OA70015A OA70015A OA10488A OA 10488 A OA10488 A OA 10488A OA 70015 A OA70015 A OA 70015A OA 70015 A OA70015 A OA 70015A OA 10488 A OA10488 A OA 10488A
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OA
OAPI
Prior art keywords
conjugate
peg
ifna
conjugate according
formula
Prior art date
Application number
OA70015A
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English (en)
French (fr)
Inventor
Pascal Sebastian Bailon
Alicia Vallejo Palleroni
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21790006&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA10488(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of OA10488A publication Critical patent/OA10488A/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/52—Cytokines; Lymphokines; Interferons
    • C07K14/555—Interferons [IFN]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
    • A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Toxicology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
OA70015A 1996-05-31 1997-05-30 Conjugué peg-ifn alpha physiologiquement actif procédé pour sa préparation compositions pharmaceutiques le contenant et leur utilisation OA10488A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1883496P 1996-05-31 1996-05-31

Publications (1)

Publication Number Publication Date
OA10488A true OA10488A (fr) 2002-04-11

Family

ID=21790006

Family Applications (1)

Application Number Title Priority Date Filing Date
OA70015A OA10488A (fr) 1996-05-31 1997-05-30 Conjugué peg-ifn alpha physiologiquement actif procédé pour sa préparation compositions pharmaceutiques le contenant et leur utilisation

Country Status (48)

Country Link
US (1) US7201897B2 (tr)
EP (1) EP0809996B1 (tr)
JP (1) JP2980569B2 (tr)
KR (1) KR100254097B1 (tr)
CN (1) CN1088721C (tr)
AR (1) AR008378A1 (tr)
AT (1) ATE235920T1 (tr)
AU (1) AU725195B2 (tr)
BG (1) BG62273B1 (tr)
BR (1) BR9703421A (tr)
CA (1) CA2203480C (tr)
CO (1) CO4950528A1 (tr)
CY (2) CY2433B1 (tr)
CZ (1) CZ292775B6 (tr)
DE (3) DE10399018I1 (tr)
DK (1) DK0809996T3 (tr)
EG (1) EG24292A (tr)
ES (1) ES2110386T3 (tr)
GR (1) GR970300063T1 (tr)
HK (1) HK1005225A1 (tr)
HR (1) HRP970298B1 (tr)
HU (1) HU227992B1 (tr)
IL (1) IL120902A (tr)
IS (1) IS1988B (tr)
LU (1) LU91029I2 (tr)
MA (1) MA24193A1 (tr)
MY (1) MY117909A (tr)
NL (1) NL300127I2 (tr)
NO (1) NO322964B1 (tr)
NZ (1) NZ314903A (tr)
OA (1) OA10488A (tr)
PA (1) PA8431001A1 (tr)
PL (1) PL186949B1 (tr)
PT (1) PT809996E (tr)
RS (1) RS49533B (tr)
RU (1) RU2180595C2 (tr)
SA (1) SA97180030B1 (tr)
SG (1) SG55314A1 (tr)
SI (1) SI0809996T1 (tr)
SK (1) SK284458B6 (tr)
SV (1) SV1997000049A (tr)
TJ (1) TJ328B (tr)
TN (1) TNSN97091A1 (tr)
TR (1) TR199700358A2 (tr)
TW (1) TW517067B (tr)
UA (1) UA56989C2 (tr)
UY (1) UY24572A1 (tr)
ZA (1) ZA974583B (tr)

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