NO328580B1 - 4-(2-butylamino)-2,7-dimetyl-8-(2-metyl-6-metoksypyrid-3-yl)pyrazolo-[1,5-A]-1,3,5-triazin, et farmasoytisk akseptabelt promedikament derav, farmasoytisk preparat, anvendelse av forbindelsen samt fremstilt gjenstand omfattende denne - Google Patents
4-(2-butylamino)-2,7-dimetyl-8-(2-metyl-6-metoksypyrid-3-yl)pyrazolo-[1,5-A]-1,3,5-triazin, et farmasoytisk akseptabelt promedikament derav, farmasoytisk preparat, anvendelse av forbindelsen samt fremstilt gjenstand omfattende denne Download PDFInfo
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- NO328580B1 NO328580B1 NO20034023A NO20034023A NO328580B1 NO 328580 B1 NO328580 B1 NO 328580B1 NO 20034023 A NO20034023 A NO 20034023A NO 20034023 A NO20034023 A NO 20034023A NO 328580 B1 NO328580 B1 NO 328580B1
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- compound
- prodrug
- pharmaceutically acceptable
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Applications Claiming Priority (2)
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| US27540301P | 2001-03-13 | 2001-03-13 | |
| PCT/US2002/006837 WO2002072202A1 (en) | 2001-03-13 | 2002-03-06 | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands |
Publications (3)
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| NO20034023L NO20034023L (no) | 2003-09-11 |
| NO20034023D0 NO20034023D0 (no) | 2003-09-11 |
| NO328580B1 true NO328580B1 (no) | 2010-03-22 |
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| NO20034023A NO328580B1 (no) | 2001-03-13 | 2003-09-11 | 4-(2-butylamino)-2,7-dimetyl-8-(2-metyl-6-metoksypyrid-3-yl)pyrazolo-[1,5-A]-1,3,5-triazin, et farmasoytisk akseptabelt promedikament derav, farmasoytisk preparat, anvendelse av forbindelsen samt fremstilt gjenstand omfattende denne |
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| US7094782B1 (en) * | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
| BR0208357A (pt) * | 2001-03-13 | 2004-06-29 | Bristol Myers Squibb Pharma Co | Composto, composição farmacêutica, método de antagonização de um receptor de fator de liberação de corticotropina (crf), método de tratamento de disfunção, método de triagem de ligantes, método de detecção de receptores de crf, método de inibição da ligação de crf, artigo industrializado e usos do composto |
| FR2842809A1 (fr) * | 2002-07-26 | 2004-01-30 | Greenpharma Sas | NOUVELLES PYRAZOLO[1,5-a]-1,3,5-TRIAZINES SUBSTITUEES ET LEURS ANALOGUES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, UTILISATION A TITRE DE MEDICAMENT ET PROCEDES POUR LEUR PREPARATION |
| AR041470A1 (es) * | 2002-10-17 | 2005-05-18 | Upjohn Co | Compuestos de pirrolo (1,2 - b) piridazina y sus usos |
| US7329658B2 (en) | 2003-02-06 | 2008-02-12 | Pfizer Inc | Cannabinoid receptor ligands and uses thereof |
| US7176210B2 (en) * | 2003-02-10 | 2007-02-13 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
| US7041671B2 (en) | 2003-04-02 | 2006-05-09 | Pfizer Inc | Pyrrolo[1,2-b]pyridazine compounds and their uses |
| US7034023B2 (en) * | 2003-04-04 | 2006-04-25 | Pfizer Inc | Pyrrolo[1,2-B]pyridazine compounds and their uses |
| US7056920B2 (en) | 2003-04-04 | 2006-06-06 | Pfizer Inc | Pyrrolo[1,2-B]pyridazine compounds and their uses |
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| US7153961B2 (en) | 2003-11-25 | 2006-12-26 | Bristol-Myers Squibb Pharma Co. | Salt and crystalline form thereof of a corticotropin releasing factor receptor antagonist |
| US7208596B2 (en) * | 2003-11-25 | 2007-04-24 | Bristol-Myers Squibb Pharma Company | Processes for the preparation of pyrazolo[1,5-a]-1,3,5-triazines and intermediates thereof |
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| WO1995010506A1 (en) | 1993-10-12 | 1995-04-20 | The Du Pont Merck Pharmaceutical Company | 1n-alkyl-n-arylpyrimidinamines and derivatives thereof |
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| CN1227554A (zh) * | 1996-08-28 | 1999-09-01 | 辉瑞大药厂 | 取代的6,5－杂二环衍生物 |
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| UA62972C2 (en) | 1997-07-03 | 2004-01-15 | Application of imidazopyrimidins and imidazopyridins for the treatment of neural disorders | |
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| BR0208357A (pt) * | 2001-03-13 | 2004-06-29 | Bristol Myers Squibb Pharma Co | Composto, composição farmacêutica, método de antagonização de um receptor de fator de liberação de corticotropina (crf), método de tratamento de disfunção, método de triagem de ligantes, método de detecção de receptores de crf, método de inibição da ligação de crf, artigo industrializado e usos do composto |
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