EE05433B1 - 4-(2-butlamino)-2,7-dimetl-8-(2-metl-6-metoksprid-3-l)[1,5-a]prasolo-1,3,5-triasiin, selle farmatseutiliselt vastuv?etavad eelravimid v?i farmatseutiliselt vastuv?etavad soolad ning nende kasutamine - Google Patents

4-(2-butlamino)-2,7-dimetl-8-(2-metl-6-metoksprid-3-l)[1,5-a]prasolo-1,3,5-triasiin, selle farmatseutiliselt vastuv?etavad eelravimid v?i farmatseutiliselt vastuv?etavad soolad ning nende kasutamine

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Publication number
EE05433B1
EE05433B1 EEP200300435A EEP200300435A EE05433B1 EE 05433 B1 EE05433 B1 EE 05433B1 EE P200300435 A EEP200300435 A EE P200300435A EE P200300435 A EEP200300435 A EE P200300435A EE 05433 B1 EE05433 B1 EE 05433B1
Authority
EE
Estonia
Prior art keywords
pharmaceutically acceptable
rasolo
methoxypyrid
butylamino
triazine
Prior art date
Application number
EEP200300435A
Other languages
English (en)
Estonian (et)
Inventor
J. Gilligan Paul
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Publication of EE200300435A publication Critical patent/EE200300435A/xx
Publication of EE05433B1 publication Critical patent/EE05433B1/xx

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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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EEP200300435A 2001-03-13 2002-03-06 4-(2-butlamino)-2,7-dimetl-8-(2-metl-6-metoksprid-3-l)[1,5-a]prasolo-1,3,5-triasiin, selle farmatseutiliselt vastuv?etavad eelravimid v?i farmatseutiliselt vastuv?etavad soolad ning nende kasutamine EE05433B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27540301P 2001-03-13 2001-03-13
PCT/US2002/006837 WO2002072202A1 (en) 2001-03-13 2002-03-06 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands

Publications (2)

Publication Number Publication Date
EE200300435A EE200300435A (et) 2003-12-15
EE05433B1 true EE05433B1 (et) 2011-06-15

Family

ID=23052141

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300435A EE05433B1 (et) 2001-03-13 2002-03-06 4-(2-butlamino)-2,7-dimetl-8-(2-metl-6-metoksprid-3-l)[1,5-a]prasolo-1,3,5-triasiin, selle farmatseutiliselt vastuv?etavad eelravimid v?i farmatseutiliselt vastuv?etavad soolad ning nende kasutamine

Country Status (36)

Country Link
US (4) US20030125330A1 (pt)
EP (1) EP1368094B1 (pt)
JP (1) JP4549630B2 (pt)
KR (1) KR100875595B1 (pt)
CN (1) CN100427093C (pt)
AR (1) AR032986A1 (pt)
AT (1) ATE355102T1 (pt)
AU (1) AU2002245605B2 (pt)
BG (1) BG66331B1 (pt)
BR (1) BR0208357A (pt)
CA (1) CA2440553C (pt)
CY (1) CY1106607T1 (pt)
CZ (1) CZ20032481A3 (pt)
DE (1) DE60218434T2 (pt)
DK (1) DK1368094T3 (pt)
EE (1) EE05433B1 (pt)
ES (1) ES2282401T3 (pt)
GE (1) GEP20053608B (pt)
HK (1) HK1057182A1 (pt)
HR (1) HRP20030822B1 (pt)
HU (1) HU229317B1 (pt)
IL (2) IL157615A0 (pt)
IS (1) IS2839B (pt)
MX (1) MXPA03008185A (pt)
MY (1) MY146935A (pt)
NO (1) NO328580B1 (pt)
NZ (1) NZ528207A (pt)
PL (1) PL208278B1 (pt)
PT (1) PT1368094E (pt)
RS (1) RS50863B (pt)
RU (1) RU2292347C2 (pt)
SK (1) SK287603B6 (pt)
TW (1) TWI257388B (pt)
UA (1) UA74634C2 (pt)
WO (1) WO2002072202A1 (pt)
ZA (1) ZA200306995B (pt)

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BR0208357A (pt) * 2001-03-13 2004-06-29 Bristol Myers Squibb Pharma Co Composto, composição farmacêutica, método de antagonização de um receptor de fator de liberação de corticotropina (crf), método de tratamento de disfunção, método de triagem de ligantes, método de detecção de receptores de crf, método de inibição da ligação de crf, artigo industrializado e usos do composto

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