NO326106B1 - Mustarinagonister, farmasoytiske sammensetninger som inneholder slike, samt anvendelse derav ved behandling av en sykdomstilstand - Google Patents
Mustarinagonister, farmasoytiske sammensetninger som inneholder slike, samt anvendelse derav ved behandling av en sykdomstilstand Download PDFInfo
- Publication number
- NO326106B1 NO326106B1 NO20025115A NO20025115A NO326106B1 NO 326106 B1 NO326106 B1 NO 326106B1 NO 20025115 A NO20025115 A NO 20025115A NO 20025115 A NO20025115 A NO 20025115A NO 326106 B1 NO326106 B1 NO 326106B1
- Authority
- NO
- Norway
- Prior art keywords
- propyl
- indazole
- butyl
- piperidin
- compound according
- Prior art date
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
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- Psychiatry (AREA)
- Psychology (AREA)
- Rheumatology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US20079100P | 2000-04-28 | 2000-04-28 | |
PCT/US2001/013561 WO2001083472A1 (en) | 2000-04-28 | 2001-04-27 | Muscarinic agonists |
Publications (3)
Publication Number | Publication Date |
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NO20025115D0 NO20025115D0 (no) | 2002-10-24 |
NO20025115L NO20025115L (no) | 2002-12-19 |
NO326106B1 true NO326106B1 (no) | 2008-09-22 |
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NO20025115A NO326106B1 (no) | 2000-04-28 | 2002-10-24 | Mustarinagonister, farmasoytiske sammensetninger som inneholder slike, samt anvendelse derav ved behandling av en sykdomstilstand |
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US (3) | US6627645B2 (ko) |
EP (1) | EP1278741B1 (ko) |
JP (2) | JP4119126B2 (ko) |
KR (2) | KR100901221B1 (ko) |
CN (3) | CN101016296A (ko) |
AR (1) | AR028385A1 (ko) |
AT (1) | ATE290000T1 (ko) |
AU (2) | AU2001259190B2 (ko) |
BR (1) | BR0110420A (ko) |
CA (1) | CA2407594A1 (ko) |
DE (1) | DE60109148T2 (ko) |
ES (1) | ES2238437T3 (ko) |
HK (1) | HK1058196A1 (ko) |
MX (1) | MXPA02010550A (ko) |
NO (1) | NO326106B1 (ko) |
NZ (1) | NZ521978A (ko) |
RU (1) | RU2269523C2 (ko) |
TW (3) | TW200505900A (ko) |
WO (1) | WO2001083472A1 (ko) |
ZA (1) | ZA200208504B (ko) |
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US3412097A (en) | 1964-09-07 | 1968-11-19 | Koninklijke Pharma Fab Nv | Indole derivatives |
BE669095A (ko) | 1964-09-07 | |||
US3417087A (en) * | 1965-12-27 | 1968-12-17 | Research Corp | 3(aminopropionyl)benzothiophenes |
US3855242A (en) * | 1967-12-15 | 1974-12-17 | Aspro Nicholas Ltd | Benzo{8 b{9 thienyl-alkyl-guanidines |
FR2305982A1 (fr) * | 1975-04-03 | 1976-10-29 | Innothera Lab Sa | Nouvelles benzothienyl amino (propyl et butyl) cetones, leur procede de preparation et leur application en therapeutique |
US4458075A (en) | 1982-04-09 | 1984-07-03 | Hoechst-Roussel Pharmaceuticals Inc. | 6-Fluoro-3-[3-(1-heterocyclo)propyl]-1,2-benzisoxazoles |
DE3430284A1 (de) | 1984-08-17 | 1986-02-27 | Troponwerke GmbH & Co KG, 5000 Köln | Neue tryptamin-derivate, ein verfahren zu ihrer herstellung und ihre verwendung |
DE4039631A1 (de) | 1990-12-12 | 1992-06-17 | Troponwerke Gmbh & Co Kg | Neuroprotektive kombination |
US5143923B1 (en) | 1991-04-29 | 1993-11-02 | Hoechst-Roussel Pharmaceuticals Incorporated | Benzoisothiazole-and benzisoxazole-3-carboxamides |
DE69332691T2 (de) | 1992-11-23 | 2003-12-18 | Aventis Pharma Inc | Substituierte 3-(aminoalkylamino)-1,2-benzisoxazole und verwandte verbindungen |
US5494908A (en) | 1992-11-23 | 1996-02-27 | Hoechst-Roussel Pharmaceutical Incorporated | Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related compounds |
IL110298A (en) | 1993-07-13 | 1999-04-11 | Brann Mark Robert | Identification of ligands by selective amplification of cells transfected with receptors |
US5654320A (en) * | 1995-03-16 | 1997-08-05 | Eli Lilly And Company | Indazolecarboxamides |
FR2735129B1 (fr) * | 1995-06-07 | 1997-07-11 | Adir | Nouveaux derives de l'indole, de l'indazole et du benzisoxazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2751647B1 (fr) | 1996-07-25 | 1998-09-11 | Synthelabo | Derives de benzimidazole, leurs preparations et leurs applications en therapeutique |
US5900312A (en) | 1996-11-08 | 1999-05-04 | W. L. Gore & Associates, Inc. | Integrated circuit chip package assembly |
DE19725664A1 (de) | 1997-06-18 | 1998-12-24 | Merck Patent Gmbh | 3-Benzylpiperidine |
FR2803298A1 (fr) | 1999-12-30 | 2001-07-06 | Adir | Nouvelles urees lineaires ou cycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2804429B1 (fr) | 2000-01-31 | 2003-05-09 | Adir | Nouveaux derives de 4-sulfonamides piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
TW200505900A (en) * | 2000-04-28 | 2005-02-16 | Acadia Pharm Inc | Muscarinic agonists |
-
2001
- 2001-04-27 TW TW093131300A patent/TW200505900A/zh unknown
- 2001-04-27 CN CNA2006101006886A patent/CN101016296A/zh active Pending
- 2001-04-27 MX MXPA02010550A patent/MXPA02010550A/es active IP Right Grant
- 2001-04-27 AR ARP010102000A patent/AR028385A1/es unknown
- 2001-04-27 CA CA002407594A patent/CA2407594A1/en not_active Abandoned
- 2001-04-27 NZ NZ521978A patent/NZ521978A/en unknown
- 2001-04-27 WO PCT/US2001/013561 patent/WO2001083472A1/en active IP Right Grant
- 2001-04-27 CN CNA2006100037035A patent/CN1814596A/zh active Pending
- 2001-04-27 US US09/844,685 patent/US6627645B2/en not_active Expired - Fee Related
- 2001-04-27 TW TW090110141A patent/TWI306859B/zh active
- 2001-04-27 RU RU2002131937/04A patent/RU2269523C2/ru active
- 2001-04-27 CN CNB01811718XA patent/CN1249051C/zh not_active Expired - Fee Related
- 2001-04-27 EP EP01932682A patent/EP1278741B1/en not_active Expired - Lifetime
- 2001-04-27 BR BR0110420-9A patent/BR0110420A/pt not_active IP Right Cessation
- 2001-04-27 AT AT01932682T patent/ATE290000T1/de not_active IP Right Cessation
- 2001-04-27 ES ES01932682T patent/ES2238437T3/es not_active Expired - Lifetime
- 2001-04-27 KR KR1020077014206A patent/KR100901221B1/ko not_active IP Right Cessation
- 2001-04-27 JP JP2001580900A patent/JP4119126B2/ja not_active Expired - Fee Related
- 2001-04-27 AU AU2001259190A patent/AU2001259190B2/en not_active Ceased
- 2001-04-27 AU AU5919001A patent/AU5919001A/xx active Pending
- 2001-04-27 DE DE60109148T patent/DE60109148T2/de not_active Expired - Fee Related
- 2001-04-27 KR KR1020027014436A patent/KR20030005306A/ko not_active IP Right Cessation
- 2001-04-27 TW TW093131368A patent/TWI310035B/zh not_active IP Right Cessation
-
2002
- 2002-10-21 ZA ZA200208504A patent/ZA200208504B/en unknown
- 2002-10-24 NO NO20025115A patent/NO326106B1/no unknown
-
2003
- 2003-07-17 US US10/623,119 patent/US7238713B2/en not_active Expired - Fee Related
-
2004
- 2004-02-12 HK HK04100926A patent/HK1058196A1/xx not_active IP Right Cessation
-
2007
- 2007-02-16 US US11/676,178 patent/US20070155795A1/en not_active Abandoned
-
2008
- 2008-02-07 JP JP2008028114A patent/JP2008133297A/ja not_active Withdrawn
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