NO20092960L - Krystallinsk minocycline base og framgangsmater for framstilling av denne - Google Patents

Krystallinsk minocycline base og framgangsmater for framstilling av denne

Info

Publication number
NO20092960L
NO20092960L NO20092960A NO20092960A NO20092960L NO 20092960 L NO20092960 L NO 20092960L NO 20092960 A NO20092960 A NO 20092960A NO 20092960 A NO20092960 A NO 20092960A NO 20092960 L NO20092960 L NO 20092960L
Authority
NO
Norway
Prior art keywords
minocycline base
processes
preparation
crystalline
crystalline minocycline
Prior art date
Application number
NO20092960A
Other languages
English (en)
Norwegian (no)
Inventor
Zita Mendes
William Heggie
Susana Marto
Jose Rafael Antunes
Original Assignee
Hovione Int Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hovione Int Ltd filed Critical Hovione Int Ltd
Publication of NO20092960L publication Critical patent/NO20092960L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/24—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
    • C07C237/26—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton of a ring being part of a condensed ring system formed by at least four rings, e.g. tetracycline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/65—Tetracyclines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20092960A 2007-02-23 2009-09-04 Krystallinsk minocycline base og framgangsmater for framstilling av denne NO20092960L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PT103661A PT103661B (pt) 2007-02-23 2007-02-23 Processo de preparação de minociclina base cristalina
PCT/GB2008/000625 WO2008102161A2 (en) 2007-02-23 2008-02-22 Crystalline minocycline base and processes for its preparation

Publications (1)

Publication Number Publication Date
NO20092960L true NO20092960L (no) 2009-11-20

Family

ID=39432804

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20092960A NO20092960L (no) 2007-02-23 2009-09-04 Krystallinsk minocycline base og framgangsmater for framstilling av denne

Country Status (20)

Country Link
US (2) US8258327B2 (https=)
EP (1) EP2125705B1 (https=)
JP (4) JP2010519247A (https=)
KR (1) KR101391132B1 (https=)
CN (1) CN101679218B (https=)
AU (1) AU2008217619B2 (https=)
BR (2) BRPI0807319B1 (https=)
CA (2) CA2722496C (https=)
DK (1) DK2125705T3 (https=)
ES (1) ES2610434T3 (https=)
HU (1) HUE033030T2 (https=)
IL (1) IL200544A0 (https=)
MX (2) MX2009008980A (https=)
NO (1) NO20092960L (https=)
NZ (1) NZ579626A (https=)
PL (1) PL2125705T3 (https=)
PT (1) PT103661B (https=)
RU (2) RU2577331C2 (https=)
WO (1) WO2008102161A2 (https=)
ZA (1) ZA200906517B (https=)

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US8636982B2 (en) 2007-08-07 2014-01-28 Foamix Ltd. Wax foamable vehicle and pharmaceutical compositions thereof
WO2009069006A2 (en) 2007-11-30 2009-06-04 Foamix Ltd. Foam containing benzoyl peroxide
WO2009072007A2 (en) 2007-12-07 2009-06-11 Foamix Ltd. Carriers, formulations, methods for formulating unstable active agents for external application and uses thereof
WO2010017310A1 (en) 2008-08-06 2010-02-11 Medicis Pharmaceutical Corporation Method for the treatment of acne and certain dosage forms thereof
PT104350A (pt) 2009-01-23 2010-07-23 Hovione Farmaci Ncia S A Processo de isolamento de tigeciclina
US20120087872A1 (en) 2009-04-28 2012-04-12 Foamix Ltd. Foamable Vehicles and Pharmaceutical Compositions Comprising Aprotic Polar Solvents and Uses Thereof
PT104644B (pt) 2009-06-26 2012-11-06 Hovione Farmaciencia S A Formulação tópica contendo uma tetraciclina e método de tratamento de infecções cutâneas usando a mesma
CA2769625C (en) 2009-07-29 2017-04-11 Foamix Ltd. Non surfactant hydro-alcoholic foamable compositions, breakable foams and their uses
WO2011013008A2 (en) 2009-07-29 2011-02-03 Foamix Ltd. Non surface active agent non polymeric agent hydro-alcoholic foamable compositions, breakable foams and their uses
US9849142B2 (en) 2009-10-02 2017-12-26 Foamix Pharmaceuticals Ltd. Methods for accelerated return of skin integrity and for the treatment of impetigo
US10029013B2 (en) 2009-10-02 2018-07-24 Foamix Pharmaceuticals Ltd. Surfactant-free, water-free formable composition and breakable foams and their uses
US9561241B1 (en) 2011-06-28 2017-02-07 Medicis Pharmaceutical Corporation Gastroretentive dosage forms for minocycline
PT106063B (pt) * 2011-12-19 2017-05-30 Inst Superior Tecnico Minociclina cristalina termorresistente produzida por recristalização com dióxido de carbono
CN104151186B (zh) * 2014-08-11 2016-06-15 重庆福安药业(集团)股份有限公司 替加环素杂质的立体选择性制备方法
PT108223B (pt) 2015-02-13 2018-05-08 Hovione Farm S A Novas formas polimórficas de minociclina base e processos para a sua preparação
MX2017012062A (es) 2015-03-23 2018-06-18 Biopharmx Inc Composicion farmaceutica de tetraciclina para uso dermatologico.
WO2017097891A1 (en) * 2015-12-10 2017-06-15 Sandoz Ag Crystalline eravacycline
MX377365B (es) 2016-09-08 2025-03-10 Journey Medical Corp Composiciones y métodos para tratar rosácea y acné.
MY203238A (en) 2018-10-29 2024-06-19 Fraunhofer Ges Zur Frderung Der Angewandten Forschung E V Tetracycline complexes with sustained activity
WO2021191273A1 (en) 2020-03-24 2021-09-30 Hovione Scientia Limited Compositions for use in treating meibomian gland dysfunction
WO2022043457A1 (en) 2020-08-27 2022-03-03 Hovione Scientia Limited Methods and compositions for treating rosacea
CN117105812B (zh) * 2023-08-16 2025-09-26 常州市第四制药厂有限公司 一种米诺环素无菌软膏剂及制备方法

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AR057649A1 (es) * 2005-05-27 2007-12-12 Wyeth Corp Formas solidas cristalinas de tigeciclina y metodos para preparar las mismas
US20070093455A1 (en) * 2005-07-21 2007-04-26 Paul Abato 10-substituted tetracyclines and methods of use thereof
PT103661B (pt) 2007-02-23 2010-09-07 Hovione Farmaciencia S A Processo de preparação de minociclina base cristalina

Also Published As

Publication number Publication date
RU2013112021A (ru) 2014-09-27
KR101391132B1 (ko) 2014-05-02
PL2125705T3 (pl) 2017-02-28
RU2485095C2 (ru) 2013-06-20
DK2125705T3 (en) 2017-01-16
US20130030195A1 (en) 2013-01-31
WO2008102161A9 (en) 2008-11-13
EP2125705A2 (en) 2009-12-02
BRPI0807319A2 (pt) 2017-05-02
JP2017039742A (ja) 2017-02-23
RU2577331C2 (ru) 2016-03-20
PT103661B (pt) 2010-09-07
IL200544A0 (en) 2010-05-17
ES2610434T3 (es) 2017-04-27
RU2009135403A (ru) 2011-03-27
JP2010519247A (ja) 2010-06-03
CN101679218A (zh) 2010-03-24
JP2019142882A (ja) 2019-08-29
CA2835788A1 (en) 2008-08-28
PT103661A (pt) 2008-08-25
HUE033030T2 (hu) 2017-11-28
US20100286417A1 (en) 2010-11-11
US8258327B2 (en) 2012-09-04
EP2125705B1 (en) 2016-10-12
CN101679218B (zh) 2013-10-30
MX340539B (es) 2016-07-13
JP2014169319A (ja) 2014-09-18
WO2008102161A3 (en) 2009-01-08
KR20100014520A (ko) 2010-02-10
CA2835788C (en) 2018-03-27
WO2008102161A2 (en) 2008-08-28
AU2008217619A1 (en) 2008-08-28
BRPI0807319B1 (pt) 2021-08-10
BR122021000846B1 (pt) 2021-08-10
US9416097B2 (en) 2016-08-16
CA2722496C (en) 2014-06-10
ZA200906517B (en) 2010-09-29
NZ579626A (en) 2011-12-22
AU2008217619B2 (en) 2013-01-10
CA2722496A1 (en) 2008-08-28
MX2009008980A (es) 2009-11-11

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Legal Events

Date Code Title Description
CHAD Change of the owner's name or address (par. 44 patent law, par. patentforskriften)

Owner name: HOVIONE SCIENTIA LIMITED, IE

FC2A Withdrawal, rejection or dismissal of laid open patent application