NO20065148L - Monocykliske heterocykler som kinase inhibitorer - Google Patents

Monocykliske heterocykler som kinase inhibitorer

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Publication number
NO20065148L
NO20065148L NO20065148A NO20065148A NO20065148L NO 20065148 L NO20065148 L NO 20065148L NO 20065148 A NO20065148 A NO 20065148A NO 20065148 A NO20065148 A NO 20065148A NO 20065148 L NO20065148 L NO 20065148L
Authority
NO
Norway
Prior art keywords
kinase inhibitors
monocyclic heterocycles
heterocycles
monocyclic
cancer
Prior art date
Application number
NO20065148A
Other languages
English (en)
Other versions
NO339960B1 (no
Inventor
Robert M Borzilleri
Kyoung S Kim
Lyndon A M Cornelius
Robert Joseph Schmidt
Gretchen M Schroeder
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35187908&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20065148(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20065148L publication Critical patent/NO20065148L/no
Publication of NO339960B1 publication Critical patent/NO339960B1/no

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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C—CHEMISTRY; METALLURGY
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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Abstract

Foreliggende oppfinnelse angår forbindelser som har formel I og II og metoder for anvendelse av dem for behandling av kreft.
NO20065148A 2004-04-23 2006-11-08 Monocykliske heterocykler, farmasøytiske preparater omfattende slike samt anvendelse av slike for behandling av kreft NO339960B1 (no)

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