NO172540C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrrolderivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrrolderivater

Info

Publication number
NO172540C
NO172540C NO890568A NO890568A NO172540C NO 172540 C NO172540 C NO 172540C NO 890568 A NO890568 A NO 890568A NO 890568 A NO890568 A NO 890568A NO 172540 C NO172540 C NO 172540C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
analogy procedure
pyrrol derivatives
pyrrol
Prior art date
Application number
NO890568A
Other languages
English (en)
Other versions
NO172540B (no
NO890568D0 (no
NO890568L (no
Inventor
Peter David Davis
Christopher Huw Hill
Geoffrey Lawton
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB888803048A external-priority patent/GB8803048D0/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO890568D0 publication Critical patent/NO890568D0/no
Publication of NO890568L publication Critical patent/NO890568L/no
Publication of NO172540B publication Critical patent/NO172540B/no
Publication of NO172540C publication Critical patent/NO172540C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/044Pyrrole radicals
NO890568A 1988-02-10 1989-02-09 Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrrolderivater NO172540C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB888803048A GB8803048D0 (en) 1988-02-10 1988-02-10 Substituted pyrroles
GB888827565A GB8827565D0 (en) 1988-02-10 1988-11-25 Substituted pyrroles

Publications (4)

Publication Number Publication Date
NO890568D0 NO890568D0 (no) 1989-02-09
NO890568L NO890568L (no) 1989-08-11
NO172540B NO172540B (no) 1993-04-26
NO172540C true NO172540C (no) 1993-08-04

Family

ID=26293462

Family Applications (1)

Application Number Title Priority Date Filing Date
NO890568A NO172540C (no) 1988-02-10 1989-02-09 Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrrolderivater

Country Status (22)

Country Link
US (1) US5057614A (no)
EP (1) EP0328026B1 (no)
JP (1) JPH0730071B2 (no)
AU (1) AU623630B2 (no)
CA (1) CA1320194C (no)
CZ (1) CZ280738B6 (no)
DE (1) DE58904168D1 (no)
DK (1) DK171891B1 (no)
DZ (1) DZ1323A1 (no)
ES (1) ES2054890T3 (no)
FI (1) FI96861C (no)
HU (1) HU201054B (no)
IE (1) IE63489B1 (no)
IL (1) IL89167A (no)
IS (1) IS1941B (no)
MC (1) MC2010A1 (no)
NO (1) NO172540C (no)
NZ (1) NZ227850A (no)
PH (1) PH25185A (no)
PT (1) PT89661B (no)
SK (1) SK75289A3 (no)
YU (1) YU47101B (no)

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EP3187495A1 (en) 2015-12-30 2017-07-05 Johannes Gutenberg-Universität Mainz 3-(5-fluoroindolyl)-4-arylmaleimide compounds and their use in tumor treatment
CN105777751B (zh) * 2016-04-26 2018-12-11 浙江工业大学 一种双芳基马来酰亚胺类化合物及其药学上可接受的盐及其制备方法和应用
US20230203017A1 (en) * 2021-12-28 2023-06-29 Kamal D. Mehta Protein Kinase C Beta Inhibitors and Uses Thereof

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HUT49348A (en) 1989-09-28
US5057614A (en) 1991-10-15
MC2010A1 (fr) 1990-02-16
AU623630B2 (en) 1992-05-21
NO172540B (no) 1993-04-26
PH25185A (en) 1991-03-27
DK55889A (da) 1989-08-11
IL89167A0 (en) 1989-09-10
NO890568D0 (no) 1989-02-09
PT89661B (pt) 1994-02-28
DZ1323A1 (fr) 2004-09-13
JPH01233281A (ja) 1989-09-19
HU201054B (en) 1990-09-28
SK278989B6 (sk) 1998-05-06
CZ75289A3 (en) 1995-12-13
PT89661A (pt) 1989-10-04
IL89167A (en) 1994-02-27
IE890416L (en) 1989-08-10
YU28489A (en) 1991-06-30
FI96861B (fi) 1996-05-31
DE58904168D1 (de) 1993-06-03
EP0328026A1 (de) 1989-08-16
IE63489B1 (en) 1995-05-03
CZ280738B6 (cs) 1996-04-17
IS3433A7 (is) 1989-08-11
NZ227850A (en) 1991-11-26
YU47101B (sh) 1994-12-28
FI96861C (fi) 1996-09-10
DK171891B1 (da) 1997-08-04
DK55889D0 (da) 1989-02-07
IS1941B (is) 2004-07-30
ES2054890T3 (es) 1994-08-16
EP0328026B1 (de) 1993-04-28
AU2965889A (en) 1989-08-10
CA1320194C (en) 1993-07-13
SK75289A3 (en) 1998-05-06
JPH0730071B2 (ja) 1995-04-05
NO890568L (no) 1989-08-11
FI890652A (fi) 1989-08-11
FI890652A0 (fi) 1989-02-10

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