NO145382C - Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater. - Google Patents

Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater.

Info

Publication number
NO145382C
NO145382C NO754024A NO754024A NO145382C NO 145382 C NO145382 C NO 145382C NO 754024 A NO754024 A NO 754024A NO 754024 A NO754024 A NO 754024A NO 145382 C NO145382 C NO 145382C
Authority
NO
Norway
Prior art keywords
amino
preparation
acid derivatives
therapeutic active
analogue procedure
Prior art date
Application number
NO754024A
Other languages
English (en)
Norwegian (no)
Other versions
NO145382B (no
NO754024L (OSRAM
Inventor
Karl Heinrich Mayer
Siegfried Petersen
Erich Klauke
Friedrich Hoffmeister
Wolfgang Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO754024L publication Critical patent/NO754024L/no
Publication of NO145382B publication Critical patent/NO145382B/no
Publication of NO145382C publication Critical patent/NO145382C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
NO754024A 1974-12-13 1975-11-28 Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater. NO145382C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (3)

Publication Number Publication Date
NO754024L NO754024L (OSRAM) 1976-06-15
NO145382B NO145382B (no) 1981-11-30
NO145382C true NO145382C (no) 1982-03-10

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
NO754024A NO145382C (no) 1974-12-13 1975-11-28 Analogifremgangsmaate til fremstilling av terapeutisk aktive 3-amino-indazolkarboksylsyrederivater.

Country Status (27)

Country Link
US (1) US4051252A (OSRAM)
JP (1) JPS5182266A (OSRAM)
AT (1) AT343653B (OSRAM)
BE (1) BE836528A (OSRAM)
CA (1) CA1059523A (OSRAM)
CH (1) CH622250A5 (OSRAM)
CS (1) CS189731B2 (OSRAM)
DD (1) DD125484A5 (OSRAM)
DE (1) DE2458965C3 (OSRAM)
DK (1) DK137082C (OSRAM)
ES (1) ES443429A1 (OSRAM)
FI (1) FI753493A7 (OSRAM)
FR (1) FR2293928A1 (OSRAM)
GB (1) GB1490306A (OSRAM)
HK (1) HK52580A (OSRAM)
HU (1) HU173557B (OSRAM)
IE (1) IE42208B1 (OSRAM)
IL (1) IL48642A (OSRAM)
KE (1) KE3078A (OSRAM)
LU (1) LU73993A1 (OSRAM)
NL (1) NL7514521A (OSRAM)
NO (1) NO145382C (OSRAM)
PL (1) PL99858B1 (OSRAM)
SE (1) SE419645B (OSRAM)
SU (1) SU604487A3 (OSRAM)
YU (1) YU315275A (OSRAM)
ZA (1) ZA757777B (OSRAM)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
KR20030030005A (ko) * 2000-09-15 2003-04-16 버텍스 파마슈티칼스 인코포레이티드 단백질 키나제 억제제로서 유용한 피라졸 화합물
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
EP1698627A1 (en) * 2000-09-15 2006-09-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
EP1345927B1 (en) 2000-12-21 2006-05-17 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
DE60238999D1 (de) 2001-09-26 2011-03-03 Pfizer Italia Srl Aminoindazolderivate mit kinaseinhibierender wirkung, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzungen
PL372198A1 (en) * 2002-02-06 2005-07-11 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
WO2003078427A1 (en) 2002-03-15 2003-09-25 Vertex Pharmaceuticals, Inc. Azolylaminoazines as inhibitors of protein kinases
BR0311291A (pt) 2002-05-17 2005-03-29 Pharmacia Italia Spa Derivados de aminoindazol ativos como inibidores da cinase, processo para sua preparação e composições farmacêuticas compreendendo os mesmos
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
KR20050032105A (ko) 2002-08-02 2005-04-06 버텍스 파마슈티칼스 인코포레이티드 Ｇｓｋ-3의 억제제로서 유용한 피라졸 조성물
WO2004041285A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
US7601718B2 (en) 2003-02-06 2009-10-13 Vertex Pharmaceuticals Incorporated Compositions useful as inhibitors of protein kinases
CA2548172A1 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
ATE542814T1 (de) 2005-08-18 2012-02-15 Vertex Pharma Pyrazinkinaseinhibitoren
WO2007056163A2 (en) 2005-11-03 2007-05-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
KR101118932B1 (ko) * 2006-04-14 2012-02-27 아보트 러보러터리즈 바닐로이드 서브타입 1(ｖｒ1) 수용체를 억제하는 인다졸릴우레아의 제조방법
WO2008057940A1 (en) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
DE602007007985D1 (de) 2006-12-19 2010-09-02 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyrimidine
CA2679884A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
RU2009137390A (ru) 2007-03-09 2011-04-20 Вертекс Фармасьютикалз Инкорпорейтед (Us) Аминопиримидины, пригодные в качестве ингибиторов протеинкиназ
AU2008226461A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyridines useful as inhibitors of protein kinases
EP2146982A2 (en) 2007-04-13 2010-01-27 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2155730A2 (en) * 2007-05-02 2010-02-24 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2152694A2 (en) * 2007-05-02 2010-02-17 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
CA2694381A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CN101687852A (zh) * 2007-05-24 2010-03-31 沃泰克斯药物股份有限公司 可用作激酶抑制剂的噻唑类和吡唑类化合物
CN101790532B (zh) 2007-07-31 2013-11-20 沃泰克斯药物股份有限公司 5-氟-1H-吡唑并[3，4-b]吡啶-3-胺及其衍生物的制备方法
JP2012501971A (ja) * 2008-09-03 2012-01-26 バーテックス ファーマシューティカルズ インコーポレイテッド 共結晶および共結晶を含む薬学的処方物
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
SI2890684T1 (en) 2012-07-24 2018-06-29 Bial-Portela & Ca, S.A. THE CLOTHING MACHINE AND THEIR USE AS ENCLOSURE INHIBITORS
EP2882712A2 (en) * 2012-07-27 2015-06-17 BIAL - Portela & Cª S.A. Process for the synthesis of substituted urea compounds
LT3024825T (lt) 2013-07-24 2017-12-11 Bial - Portela & C, S.A. Imidazolo karboksamidai ir jų panaudojimas kaip faah inhibitorių

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3274203A (en) * 1963-05-31 1966-09-20 Du Pont 1-carbamyl and thiocarbamyl-3-amino-4-nonsubstituted and substituted pyrazoles
NL6707299A (OSRAM) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
IE42208L (en) 1976-06-13
FR2293928A1 (fr) 1976-07-09
DD125484A5 (OSRAM) 1977-04-20
BE836528A (fr) 1976-06-11
KE3078A (en) 1980-10-03
ATA939775A (de) 1977-10-15
HU173557B (hu) 1979-06-28
IL48642A0 (en) 1976-02-29
AT343653B (de) 1978-06-12
DE2458965A1 (de) 1976-06-16
SE419645B (sv) 1981-08-17
SE7513990L (sv) 1976-06-14
DK137082C (da) 1978-06-19
DE2458965C3 (de) 1979-10-11
JPS5182266A (en) 1976-07-19
GB1490306A (en) 1977-11-02
LU73993A1 (OSRAM) 1976-11-11
DE2458965B2 (de) 1979-02-22
DK567275A (da) 1976-06-14
CA1059523A (en) 1979-07-31
ES443429A1 (es) 1977-04-16
FR2293928B1 (OSRAM) 1979-09-21
CH622250A5 (OSRAM) 1981-03-31
YU315275A (en) 1982-02-28
IL48642A (en) 1979-12-30
NO145382B (no) 1981-11-30
PL99858B1 (pl) 1978-08-31
US4051252A (en) 1977-09-27
CS189731B2 (en) 1979-04-30
DK137082B (da) 1978-01-16
ZA757777B (en) 1976-11-24
SU604487A3 (ru) 1978-04-25
HK52580A (en) 1980-09-26
IE42208B1 (en) 1980-06-18
NL7514521A (nl) 1976-06-15
NO754024L (OSRAM) 1976-06-15
FI753493A7 (OSRAM) 1976-06-14
AU8717075A (en) 1977-06-09

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