CS189731B2 - Method of producing new derivatives of 3-aminoindazolcarboxylic acid - Google Patents

Method of producing new derivatives of 3-aminoindazolcarboxylic acid

Info

Publication number
CS189731B2
CS189731B2 CS758165A CS816575A CS189731B2 CS 189731 B2 CS189731 B2 CS 189731B2 CS 758165 A CS758165 A CS 758165A CS 816575 A CS816575 A CS 816575A CS 189731 B2 CS189731 B2 CS 189731B2
Authority
CS
Czechoslovakia
Prior art keywords
aminoindazolcarboxylic
acid
producing new
new derivatives
derivatives
Prior art date
Application number
CS758165A
Other languages
Czech (cs)
English (en)
Inventor
Karl H Mayer
Siegfried Petersen
Erich Klauke
Friedrich Hoffmeister
Wolfgang Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of CS189731B2 publication Critical patent/CS189731B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CS758165A 1974-12-13 1975-12-02 Method of producing new derivatives of 3-aminoindazolcarboxylic acid CS189731B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
CS189731B2 true CS189731B2 (en) 1979-04-30

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
CS758165A CS189731B2 (en) 1974-12-13 1975-12-02 Method of producing new derivatives of 3-aminoindazolcarboxylic acid

Country Status (27)

Country Link
US (1) US4051252A (OSRAM)
JP (1) JPS5182266A (OSRAM)
AT (1) AT343653B (OSRAM)
BE (1) BE836528A (OSRAM)
CA (1) CA1059523A (OSRAM)
CH (1) CH622250A5 (OSRAM)
CS (1) CS189731B2 (OSRAM)
DD (1) DD125484A5 (OSRAM)
DE (1) DE2458965C3 (OSRAM)
DK (1) DK137082C (OSRAM)
ES (1) ES443429A1 (OSRAM)
FI (1) FI753493A7 (OSRAM)
FR (1) FR2293928A1 (OSRAM)
GB (1) GB1490306A (OSRAM)
HK (1) HK52580A (OSRAM)
HU (1) HU173557B (OSRAM)
IE (1) IE42208B1 (OSRAM)
IL (1) IL48642A (OSRAM)
KE (1) KE3078A (OSRAM)
LU (1) LU73993A1 (OSRAM)
NL (1) NL7514521A (OSRAM)
NO (1) NO145382C (OSRAM)
PL (1) PL99858B1 (OSRAM)
SE (1) SE419645B (OSRAM)
SU (1) SU604487A3 (OSRAM)
YU (1) YU315275A (OSRAM)
ZA (1) ZA757777B (OSRAM)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
ZA200301701B (en) * 2000-09-15 2004-03-01 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
WO2002022605A1 (en) * 2000-09-15 2002-03-21 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
AP2003002825A0 (en) 2000-12-21 2003-09-30 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
NZ531765A (en) 2001-09-26 2006-02-24 Pharmacia Italia S Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
WO2003066629A2 (en) * 2002-02-06 2003-08-14 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
US20040009981A1 (en) 2002-03-15 2004-01-15 David Bebbington Compositions useful as inhibitors of protein kinases
AU2003227741A1 (en) 2002-05-17 2003-12-02 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
ATE339419T1 (de) 2002-08-02 2006-10-15 Vertex Pharma Pyrazolenthaltende zusammensetzungen und ihre verwendung als gsk-3 inhibitoren
EP1556053A4 (en) * 2002-10-31 2006-04-19 Amgen Inc ANTI-INFLAMMATORY AGENTS
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
JP2007513184A (ja) * 2003-12-04 2007-05-24 バーテックス　ファーマシューティカルズ　インコーポレイテッド プロテインキナーゼのインヒビターとして有用なキノキサリン
DE102004005172A1 (de) 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
US7737151B2 (en) 2005-08-18 2010-06-15 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
US7528142B2 (en) 2005-11-03 2009-05-05 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CN102775350A (zh) * 2006-04-14 2012-11-14 雅培制药有限公司 制备抑制香草素亚型1（vr1）受体的吲唑基脲的方法
ATE457311T1 (de) 2006-11-02 2010-02-15 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyridine und aminopyrimidine
NZ577768A (en) 2006-12-19 2012-01-12 Vertex Pharma Aminopyrimidines useful as inhibitors of protein kinases
AU2008226461A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyridines useful as inhibitors of protein kinases
CN101663295B (zh) 2007-03-09 2014-11-05 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的氨基嘧啶类化合物
AU2008226466B2 (en) 2007-03-09 2013-06-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
JP2010523700A (ja) 2007-04-13 2010-07-15 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼインヒビターとして有用なアミノピリミジン
AU2008247594A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
WO2008137619A2 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
CA2688584A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
WO2008147626A2 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
NZ582879A (en) 2007-07-31 2012-03-30 Vertex Pharma Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
MX2011002312A (es) * 2008-09-03 2011-04-26 Vertex Pharma Co-cristales y formulaciones farmaceuticas que comprenden los mismos.
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
MX365772B (es) 2012-07-24 2019-06-13 Bial Portela & Ca Sa Compuestos de urea y su uso como inhibidores de enzimas.
EP2882712A2 (en) * 2012-07-27 2015-06-17 BIAL - Portela & Cª S.A. Process for the synthesis of substituted urea compounds
EP3024825B1 (en) 2013-07-24 2017-06-21 BIAL - PORTELA & Cª, S.A. Imidazolecarboxamides and their use as faah inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (OSRAM) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
SE7513990L (sv) 1976-06-14
SE419645B (sv) 1981-08-17
HK52580A (en) 1980-09-26
DK567275A (da) 1976-06-14
DK137082B (da) 1978-01-16
DD125484A5 (OSRAM) 1977-04-20
ATA939775A (de) 1977-10-15
US4051252A (en) 1977-09-27
FR2293928B1 (OSRAM) 1979-09-21
AU8717075A (en) 1977-06-09
KE3078A (en) 1980-10-03
BE836528A (fr) 1976-06-11
CH622250A5 (OSRAM) 1981-03-31
HU173557B (hu) 1979-06-28
IE42208B1 (en) 1980-06-18
DK137082C (da) 1978-06-19
AT343653B (de) 1978-06-12
FR2293928A1 (fr) 1976-07-09
DE2458965B2 (de) 1979-02-22
PL99858B1 (pl) 1978-08-31
GB1490306A (en) 1977-11-02
DE2458965A1 (de) 1976-06-16
FI753493A7 (OSRAM) 1976-06-14
NL7514521A (nl) 1976-06-15
YU315275A (en) 1982-02-28
JPS5182266A (en) 1976-07-19
NO145382C (no) 1982-03-10
DE2458965C3 (de) 1979-10-11
SU604487A3 (ru) 1978-04-25
LU73993A1 (OSRAM) 1976-11-11
ZA757777B (en) 1976-11-24
NO754024L (OSRAM) 1976-06-15
IL48642A0 (en) 1976-02-29
CA1059523A (en) 1979-07-31
ES443429A1 (es) 1977-04-16
NO145382B (no) 1981-11-30
IE42208L (en) 1976-06-13
IL48642A (en) 1979-12-30

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