DK567275A - 3-amino-indazolcarboxylsyrederivater samt deres fremstilling og anvendelse - Google Patents

3-amino-indazolcarboxylsyrederivater samt deres fremstilling og anvendelse

Info

Publication number
DK567275A
DK567275A DK567275A DK567275A DK567275A DK 567275 A DK567275 A DK 567275A DK 567275 A DK567275 A DK 567275A DK 567275 A DK567275 A DK 567275A DK 567275 A DK567275 A DK 567275A
Authority
DK
Denmark
Prior art keywords
amino
preparation
carboxylic acid
acid derivatives
indazole carboxylic
Prior art date
Application number
DK567275A
Other languages
English (en)
Other versions
DK137082C (da
DK137082B (da
Inventor
K H Mayer
S Petersen
E Klauke
F Hoffmeister
W Wuttke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of DK567275A publication Critical patent/DK567275A/da
Publication of DK137082B publication Critical patent/DK137082B/da
Application granted granted Critical
Publication of DK137082C publication Critical patent/DK137082C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK567275A 1974-12-13 1975-12-12 Analogifremgangsmaade til fremstilling af 3-aminoindazolcarboxylsyrederivater DK137082C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (3)

Publication Number Publication Date
DK567275A true DK567275A (da) 1976-06-14
DK137082B DK137082B (da) 1978-01-16
DK137082C DK137082C (da) 1978-06-19

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
DK567275A DK137082C (da) 1974-12-13 1975-12-12 Analogifremgangsmaade til fremstilling af 3-aminoindazolcarboxylsyrederivater

Country Status (27)

Country Link
US (1) US4051252A (da)
JP (1) JPS5182266A (da)
AT (1) AT343653B (da)
BE (1) BE836528A (da)
CA (1) CA1059523A (da)
CH (1) CH622250A5 (da)
CS (1) CS189731B2 (da)
DD (1) DD125484A5 (da)
DE (1) DE2458965C3 (da)
DK (1) DK137082C (da)
ES (1) ES443429A1 (da)
FI (1) FI753493A (da)
FR (1) FR2293928A1 (da)
GB (1) GB1490306A (da)
HK (1) HK52580A (da)
HU (1) HU173557B (da)
IE (1) IE42208B1 (da)
IL (1) IL48642A (da)
KE (1) KE3078A (da)
LU (1) LU73993A1 (da)
NL (1) NL7514521A (da)
NO (1) NO145382C (da)
PL (1) PL99858B1 (da)
SE (1) SE419645B (da)
SU (1) SU604487A3 (da)
YU (1) YU315275A (da)
ZA (1) ZA757777B (da)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
EP1317448B2 (en) * 2000-09-15 2011-05-04 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
ZA200301703B (en) * 2000-09-15 2004-03-02 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
DE60120219T2 (de) 2000-12-21 2007-04-12 Vertex Pharmaceuticals Inc., Cambridge Pyrazolverbindungen als protein-kinase-inhibitoren
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
EP1820503B1 (en) 2001-09-26 2012-02-22 Pfizer Italia S.r.l. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
JP4656838B2 (ja) * 2002-02-06 2011-03-23 バーテックス ファーマシューティカルズ インコーポレイテッド Ｇｓｋ−３の阻害剤として有用なヘテロアリール化合物
FR2836915B1 (fr) 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
ATE468336T1 (de) 2002-03-15 2010-06-15 Vertex Pharma Azolylaminoazine als proteinkinasehemmer
ES2411655T3 (es) 2002-05-17 2013-07-08 Pfizer Italia S.R.L. Derivados de aminoindazol activos como inhibidores de quinasas, procedimiento para su preparación y composiciones farmacéuticas que los comprenden
MY141867A (en) 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
PL374967A1 (en) 2002-08-02 2005-11-14 Vertex Pharmaceuticals Incorporated Pyrazole compositions useful as inhibitors of gsk-3
WO2004041285A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
WO2005056547A2 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
WO2007022384A2 (en) 2005-08-18 2007-02-22 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
WO2007056221A2 (en) 2005-11-03 2007-05-18 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
NZ571705A (en) * 2006-04-14 2012-03-30 Abbott Lab Process for the preparation of indazolyl ureas that inhibit vanilloid subtype 1 (VR1) receptors
MX2009004807A (es) 2006-11-02 2009-06-15 Vertex Pharma Aminopiridinas y aminopirimidinas utiles como inhibidores de proteina cinasa.
EP2099787B1 (en) 2006-12-19 2010-07-21 Vertex Pharmaceuticals, Inc. Aminopyrimidines useful as inhibitors of protein kinases
AU2008226461A1 (en) 2007-03-09 2008-09-18 Vertex Pharmaceuticals Incorporated Aminopyridines useful as inhibitors of protein kinases
CN101663295B (zh) 2007-03-09 2014-11-05 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的氨基嘧啶类化合物
AU2008226466B2 (en) 2007-03-09 2013-06-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
CA2683785A1 (en) 2007-04-13 2008-10-23 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2152694A2 (en) * 2007-05-02 2010-02-17 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
EP2155730A2 (en) * 2007-05-02 2010-02-24 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
AU2008247594A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CN101687852A (zh) * 2007-05-24 2010-03-31 沃泰克斯药物股份有限公司 可用作激酶抑制剂的噻唑类和吡唑类化合物
JP5553751B2 (ja) 2007-07-31 2014-07-16 バーテックス ファーマシューティカルズ インコーポレイテッド ５−フルオロ−１Ｈ−ピラゾロ［３，４−ｂ］ピリジン−３−アミンおよびその誘導体を調製するためのプロセス
RU2011112802A (ru) * 2008-09-03 2012-10-10 Вертекс Фармасьютикалз Инкорпорейтед (Us) Сокристаллы и содержащие их фармацевтические композиции
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
EP2890684B1 (en) 2012-07-24 2018-02-14 Bial-Portela & CA, S.A. Urea compounds and their use as enzyme inhibitors
CA2880299A1 (en) * 2012-07-27 2014-01-30 Bial - Portela & Ca, S.A. Process for the synthesis of substituted urea compounds
CN105793247B (zh) 2013-07-24 2018-03-16 比亚尔-珀特拉和Ca股份公司 咪唑甲酰胺类及其作为faah抑制剂的用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (da) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
US4051252A (en) 1977-09-27
HU173557B (hu) 1979-06-28
CA1059523A (en) 1979-07-31
GB1490306A (en) 1977-11-02
PL99858B1 (pl) 1978-08-31
SE7513990L (sv) 1976-06-14
JPS5182266A (en) 1976-07-19
IE42208L (en) 1976-06-13
ES443429A1 (es) 1977-04-16
NO145382C (no) 1982-03-10
SU604487A3 (ru) 1978-04-25
YU315275A (en) 1982-02-28
DE2458965C3 (de) 1979-10-11
DK137082C (da) 1978-06-19
NO754024L (da) 1976-06-15
HK52580A (en) 1980-09-26
DE2458965B2 (de) 1979-02-22
DD125484A5 (da) 1977-04-20
DK137082B (da) 1978-01-16
FR2293928B1 (da) 1979-09-21
AU8717075A (en) 1977-06-09
DE2458965A1 (de) 1976-06-16
CH622250A5 (da) 1981-03-31
NL7514521A (nl) 1976-06-15
IL48642A0 (en) 1976-02-29
BE836528A (fr) 1976-06-11
NO145382B (no) 1981-11-30
AT343653B (de) 1978-06-12
CS189731B2 (en) 1979-04-30
IE42208B1 (en) 1980-06-18
ATA939775A (de) 1977-10-15
SE419645B (sv) 1981-08-17
KE3078A (en) 1980-10-03
ZA757777B (en) 1976-11-24
FI753493A (da) 1976-06-14
IL48642A (en) 1979-12-30
FR2293928A1 (fr) 1976-07-09
LU73993A1 (da) 1976-11-11

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