ES443429A1 - Procedimiento para preparar derivados de acido 3-amino-inda-zolcarboxilico. - Google Patents

Procedimiento para preparar derivados de acido 3-amino-inda-zolcarboxilico.

Info

Publication number
ES443429A1
ES443429A1 ES443429A ES443429A ES443429A1 ES 443429 A1 ES443429 A1 ES 443429A1 ES 443429 A ES443429 A ES 443429A ES 443429 A ES443429 A ES 443429A ES 443429 A1 ES443429 A1 ES 443429A1
Authority
ES
Spain
Prior art keywords
formula
radical
amino
hydrogen
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES443429A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of ES443429A1 publication Critical patent/ES443429A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
ES443429A 1974-12-13 1975-12-12 Procedimiento para preparar derivados de acido 3-amino-inda-zolcarboxilico. Expired ES443429A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
ES443429A1 true ES443429A1 (es) 1977-04-16

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
ES443429A Expired ES443429A1 (es) 1974-12-13 1975-12-12 Procedimiento para preparar derivados de acido 3-amino-inda-zolcarboxilico.

Country Status (27)

Country Link
US (1) US4051252A (es)
JP (1) JPS5182266A (es)
AT (1) AT343653B (es)
BE (1) BE836528A (es)
CA (1) CA1059523A (es)
CH (1) CH622250A5 (es)
CS (1) CS189731B2 (es)
DD (1) DD125484A5 (es)
DE (1) DE2458965C3 (es)
DK (1) DK137082C (es)
ES (1) ES443429A1 (es)
FI (1) FI753493A (es)
FR (1) FR2293928A1 (es)
GB (1) GB1490306A (es)
HK (1) HK52580A (es)
HU (1) HU173557B (es)
IE (1) IE42208B1 (es)
IL (1) IL48642A (es)
KE (1) KE3078A (es)
LU (1) LU73993A1 (es)
NL (1) NL7514521A (es)
NO (1) NO145382C (es)
PL (1) PL99858B1 (es)
SE (1) SE419645B (es)
SU (1) SU604487A3 (es)
YU (1) YU315275A (es)
ZA (1) ZA757777B (es)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
WO2002022605A1 (en) 2000-09-15 2002-03-21 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
US6989385B2 (en) * 2000-12-21 2006-01-24 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
KR20040047869A (ko) 2001-09-26 2004-06-05 파마시아 이탈리아 에스.피.에이. 키나제 억제제로서 활성인 아미노인다졸 유도체, 이의제조방법 및 이를 함유하는 약제학적 조성물
RU2004126671A (ru) * 2002-02-06 2005-04-10 Вертекс Фармасьютикалз Инкорпорейтед (Us) Гетероарилсоединения, полезные в качестве ингибиторов gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
US20040009981A1 (en) 2002-03-15 2004-01-15 David Bebbington Compositions useful as inhibitors of protein kinases
ES2411655T3 (es) 2002-05-17 2013-07-08 Pfizer Italia S.R.L. Derivados de aminoindazol activos como inhibidores de quinasas, procedimiento para su preparación y composiciones farmacéuticas que los comprenden
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
EA200500299A1 (ru) 2002-08-02 2005-08-25 Вертекс Фармасьютикалз Инкорпорейтед Пиразольные композиции, используемые в качестве ингибиторов gsk-3
CA2502429A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
CN1902193B (zh) * 2003-12-04 2011-07-13 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的喹喔啉
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
WO2007022384A2 (en) 2005-08-18 2007-02-22 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
NZ594383A (en) 2005-11-03 2013-05-31 Vertex Pharma Aminopyrimidines useful as kinase inhibitors
MX2008013205A (es) * 2006-04-14 2008-10-22 Abbott Lab Procedimiento para la preparacion de indazolil ureas que inhibien receptores de vanilloides del subtipo 1 (vr1).
NZ576750A (en) 2006-11-02 2012-01-12 Vertex Pharma Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
EP2099787B1 (en) 2006-12-19 2010-07-21 Vertex Pharmaceuticals, Inc. Aminopyrimidines useful as inhibitors of protein kinases
RU2009137390A (ru) 2007-03-09 2011-04-20 Вертекс Фармасьютикалз Инкорпорейтед (Us) Аминопиримидины, пригодные в качестве ингибиторов протеинкиназ
CN101663295B (zh) 2007-03-09 2014-11-05 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的氨基嘧啶类化合物
NZ579483A (en) 2007-03-09 2012-07-27 Vertex Pharma Aminopyridines useful as inhibitors of protein kinases
MX2009011059A (es) 2007-04-13 2009-11-26 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasas.
JP5389785B2 (ja) * 2007-05-02 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害剤として有用なチアゾールおよびピラゾール
MX2009011811A (es) * 2007-05-02 2010-01-14 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasa.
AU2008247594A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
JP2010528021A (ja) * 2007-05-24 2010-08-19 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼのインヒビターとして有用なチアゾールおよびピラゾール
NZ582879A (en) * 2007-07-31 2012-03-30 Vertex Pharma Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
KR20110050549A (ko) * 2008-09-03 2011-05-13 버텍스 파마슈티칼스 인코포레이티드 공-결정 및 이를 포함하는 제약 제제
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
WO2014017936A2 (en) 2012-07-24 2014-01-30 Bial- Portela & Ca, S.A. Urea compounds and their use as enzyme inhibitors
JP2015528013A (ja) * 2012-07-27 2015-09-24 ビアル−ポルテラ エ コンパニア，ソシエダッド アノニマ 置換ウレア化合物の合成方法
CA2918993C (en) 2013-07-24 2021-08-24 Bial - Portela & Ca, S.A. Imidazolecarboxamides and their use as faah inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (es) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
HU173557B (hu) 1979-06-28
NO145382B (no) 1981-11-30
CA1059523A (en) 1979-07-31
US4051252A (en) 1977-09-27
FI753493A (es) 1976-06-14
DK567275A (da) 1976-06-14
GB1490306A (en) 1977-11-02
NO754024L (es) 1976-06-15
ATA939775A (de) 1977-10-15
ZA757777B (en) 1976-11-24
IL48642A0 (en) 1976-02-29
AT343653B (de) 1978-06-12
KE3078A (en) 1980-10-03
NL7514521A (nl) 1976-06-15
DE2458965B2 (de) 1979-02-22
DK137082B (da) 1978-01-16
HK52580A (en) 1980-09-26
LU73993A1 (es) 1976-11-11
SU604487A3 (ru) 1978-04-25
SE7513990L (sv) 1976-06-14
YU315275A (en) 1982-02-28
DK137082C (da) 1978-06-19
AU8717075A (en) 1977-06-09
BE836528A (fr) 1976-06-11
IL48642A (en) 1979-12-30
FR2293928B1 (es) 1979-09-21
CH622250A5 (es) 1981-03-31
JPS5182266A (en) 1976-07-19
NO145382C (no) 1982-03-10
CS189731B2 (en) 1979-04-30
FR2293928A1 (fr) 1976-07-09
IE42208B1 (en) 1980-06-18
PL99858B1 (pl) 1978-08-31
SE419645B (sv) 1981-08-17
DE2458965A1 (de) 1976-06-16
IE42208L (en) 1976-06-13
DD125484A5 (es) 1977-04-20
DE2458965C3 (de) 1979-10-11

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