NO141800C - Analogifremgangsmaate for fremstilling av terapeutisk aktive benzomorfaner. - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive benzomorfaner.

Info

Publication number
NO141800C
NO141800C NO750773A NO750773A NO141800C NO 141800 C NO141800 C NO 141800C NO 750773 A NO750773 A NO 750773A NO 750773 A NO750773 A NO 750773A NO 141800 C NO141800 C NO 141800C
Authority
NO
Norway
Prior art keywords
benzomorphanes
preparation
therapeutic active
analogy procedure
analogy
Prior art date
Application number
NO750773A
Other languages
English (en)
Other versions
NO141800B (no
NO750773L (no
Inventor
Herbert Merz
Adolf Langbein
Gerhard Walther
Klaus Stockhaus
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of NO750773L publication Critical patent/NO750773L/no
Publication of NO141800B publication Critical patent/NO141800B/no
Publication of NO141800C publication Critical patent/NO141800C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
NO750773A 1974-03-09 1975-03-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive benzomorfaner. NO141800C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2411382A DE2411382C3 (de) 1974-03-09 1974-03-09 2-Tetrahydrofurfuryl-6,7-benzomorphane, Verfahren zur Herstellung und deren Verwendung

Publications (3)

Publication Number Publication Date
NO750773L NO750773L (no) 1975-09-10
NO141800B NO141800B (no) 1980-02-04
NO141800C true NO141800C (no) 1980-06-04

Family

ID=5909593

Family Applications (1)

Application Number Title Priority Date Filing Date
NO750773A NO141800C (no) 1974-03-09 1975-03-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive benzomorfaner.

Country Status (25)

Country Link
JP (1) JPS5827275B2 (no)
AT (1) AT344332B (no)
BE (1) BE826440A (no)
BG (3) BG24813A4 (no)
CA (1) CA1049511A (no)
CH (8) CH612425A5 (no)
CS (1) CS188221B2 (no)
DD (1) DD119236A5 (no)
DE (1) DE2411382C3 (no)
DK (1) DK137188C (no)
ES (6) ES440347A1 (no)
FI (1) FI63571C (no)
FR (1) FR2262984B1 (no)
GB (1) GB1496418A (no)
HU (1) HU177408B (no)
IE (1) IE40945B1 (no)
IL (1) IL46760A (no)
NL (1) NL7502724A (no)
NO (1) NO141800C (no)
PH (1) PH14127A (no)
PL (3) PL93700B1 (no)
RO (2) RO69617A (no)
SE (1) SE421919B (no)
SU (3) SU577982A3 (no)
ZA (1) ZA751394B (no)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2716687A1 (de) * 1977-04-15 1978-10-19 Boehringer Sohn Ingelheim 2'-hydroxy-2-(5-isoxazolylmethyl)-6,7benzomorphane, deren saeureadditionssalze und diese enthaltende arzneimittel
DE2828039A1 (de) * 1978-06-26 1980-01-10 Boehringer Sohn Ingelheim 2-(2-alkoxyethyl)-2'-hydroxy-6,7-benzomorphane deren saeureadditionssalze diese enthaltende arzneimittel und verfahren zu deren herstellung
US6492420B2 (en) 1995-03-10 2002-12-10 Photocure As Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
US6992107B1 (en) 1995-03-10 2006-01-31 Photocure Asa Esters of 5-aminolevulinic acid and their use as photosensitizing compounds in photochemotherapy
DE122006000051I2 (de) * 1995-03-10 2010-07-08 Photocure Asa Hoffsveien 48 Ester der 5-Aminolevulinsäure als Mittel zur Photosensibilisierung in der Chemotherapie
US7530461B2 (en) 1995-03-10 2009-05-12 Photocure Asa Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
GB0018528D0 (en) 2000-07-27 2000-09-13 Photocure Asa Compounds
US6723750B2 (en) 2002-03-15 2004-04-20 Allergan, Inc. Photodynamic therapy for pre-melanomas
JP5451611B2 (ja) 2007-07-26 2014-03-26 ヴァイティー ファーマシューティカルズ,インコーポレイテッド 11β−ヒドロキシステロイドデヒドロゲナーゼ1のサイクリックインヒビター
JP5769970B2 (ja) 2007-11-16 2015-08-26 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ベンゾモルファン及び関連骨格のアリール−及びヘテロアリールカルボニル誘導体、かかる化合物を含有する医薬及びこれらの使用
US8440658B2 (en) 2007-12-11 2013-05-14 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11β-hydroxysteroid dehydrogenase 1
TW200934490A (en) 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
WO2009094169A1 (en) 2008-01-24 2009-07-30 Vitae Pharmaceuticals, Inc. Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2254872A2 (en) 2008-02-15 2010-12-01 Vitae Pharmaceuticals, Inc. Cycloalkyl lactame derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
RU2531272C2 (ru) 2008-05-01 2014-10-20 Вайтаи Фармасьютиклз, Инк. Циклические ингибиторы 11бета-гидроксистероид-дегидрогеназы 1
US8569292B2 (en) 2008-05-01 2013-10-29 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1
CA2723034A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8765780B2 (en) 2008-05-13 2014-07-01 Boehringer Ingelheim International Gmbh Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use
JP5777030B2 (ja) 2008-07-25 2015-09-09 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 11β−ヒドロキシステロイドデヒドロゲナーゼ1の阻害剤
EP2324018B1 (en) 2008-07-25 2013-09-04 Boehringer Ingelheim International GmbH Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
UA109255C2 (ru) 2009-04-30 2015-08-10 Берінгер Інгельхайм Інтернешнл Гмбх Циклические ингибиторы 11бета-гидроксистероиддегидрогеназы 1
US8927539B2 (en) 2009-06-11 2015-01-06 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure
TWI531571B (zh) 2009-11-06 2016-05-01 維它藥物公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜芳基羰基衍生物
US8933072B2 (en) 2010-06-16 2015-01-13 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
TWI537258B (zh) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜環芳基羰基衍生物
WO2013025664A1 (en) 2011-08-17 2013-02-21 Boehringer Ingelheim International Gmbh Indenopyridine derivatives

Also Published As

Publication number Publication date
DE2411382B2 (de) 1979-01-18
NO141800B (no) 1980-02-04
CH612425A5 (en) 1979-07-31
SE7502592L (no) 1975-09-10
GB1496418A (en) 1977-12-30
FI63571B (fi) 1983-03-31
DK92975A (no) 1975-09-10
ES440350A1 (es) 1977-03-16
PL93699B1 (no) 1977-06-30
CH620681A5 (en) 1980-12-15
PH14127A (en) 1981-02-26
ZA751394B (en) 1976-11-24
BG24814A4 (en) 1978-05-12
SU577982A3 (ru) 1977-10-25
DD119236A5 (no) 1976-04-12
CH620440A5 (en) 1980-11-28
DE2411382A1 (de) 1975-09-18
AT344332B (de) 1978-07-10
CH622017A5 (en) 1981-03-13
FI63571C (fi) 1983-07-11
ES440346A1 (es) 1977-03-01
CH622016A5 (en) 1981-03-13
JPS5827275B2 (ja) 1983-06-08
DK137188C (da) 1978-07-03
BG25087A3 (en) 1978-07-12
IE40945L (en) 1975-09-09
CH620439A5 (en) 1980-11-28
CA1049511A (en) 1979-02-27
CH622015A5 (en) 1981-03-13
ES440348A1 (es) 1977-06-01
FI750652A (no) 1975-09-10
HU177408B (en) 1981-10-28
BE826440A (fr) 1975-09-08
PL93700B1 (no) 1977-06-30
ATA153875A (de) 1977-11-15
RO69617A (ro) 1980-08-15
AU7894275A (en) 1976-09-16
SU588916A3 (ru) 1978-01-15
RO70051A (ro) 1980-12-30
NO750773L (no) 1975-09-10
SU577983A3 (ru) 1977-10-25
CS188221B2 (en) 1979-02-28
FR2262984A1 (no) 1975-10-03
PL93499B1 (no) 1977-05-30
ES440347A1 (es) 1977-06-01
FR2262984B1 (no) 1978-07-28
CH622014A5 (en) 1981-03-13
NL7502724A (nl) 1975-09-11
JPS50123675A (no) 1975-09-29
IL46760A0 (en) 1975-05-22
ES440349A1 (es) 1977-03-01
SE421919B (sv) 1982-02-08
IE40945B1 (en) 1979-09-12
DK137188B (da) 1978-01-30
IL46760A (en) 1978-12-17
ES440345A1 (es) 1977-03-01
BG24813A4 (en) 1978-05-12
DE2411382C3 (de) 1979-09-06

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