NL8701226A - Imidazochinolinyletherderivaten met geneesmiddelwerking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze derivaten bevatten. - Google Patents

Imidazochinolinyletherderivaten met geneesmiddelwerking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze derivaten bevatten. Download PDF

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Publication number
NL8701226A
NL8701226A NL8701226A NL8701226A NL8701226A NL 8701226 A NL8701226 A NL 8701226A NL 8701226 A NL8701226 A NL 8701226A NL 8701226 A NL8701226 A NL 8701226A NL 8701226 A NL8701226 A NL 8701226A
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NL
Netherlands
Prior art keywords
formula
aromatic
methyl
ortho
oxo
Prior art date
Application number
NL8701226A
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English (en)
Unknown language (lm)
Dutch (nl)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of NL8701226A publication Critical patent/NL8701226A/nl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NL8701226A 1986-05-23 1987-05-22 Imidazochinolinyletherderivaten met geneesmiddelwerking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze derivaten bevatten. NL8701226A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86681386 1986-05-23
US06/866,813 US4775674A (en) 1986-05-23 1986-05-23 Imidazoquinolinylether derivatives useful as phosphodiesterase and blood aggregation inhibitors

Publications (1)

Publication Number Publication Date
NL8701226A true NL8701226A (nl) 1987-12-16

Family

ID=25348473

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8701226A NL8701226A (nl) 1986-05-23 1987-05-22 Imidazochinolinyletherderivaten met geneesmiddelwerking, werkwijzen ter bereiding daarvan alsmede farmaceutische preparaten die deze derivaten bevatten.

Country Status (24)

Country Link
US (1) US4775674A (ko)
JP (1) JPS62283972A (ko)
KR (1) KR900008567B1 (ko)
AT (1) AT392790B (ko)
AU (1) AU603577B2 (ko)
BE (1) BE1002033A4 (ko)
CA (1) CA1289137C (ko)
CH (1) CH675246A5 (ko)
DE (1) DE3717291A1 (ko)
DK (1) DK166084C (ko)
ES (1) ES2005588A6 (ko)
FI (1) FI86723C (ko)
FR (1) FR2603586B1 (ko)
GB (1) GB2190676B (ko)
GR (1) GR870803B (ko)
HU (1) HU197570B (ko)
IL (1) IL82612A0 (ko)
IT (1) IT1205031B (ko)
LU (1) LU86896A1 (ko)
NL (1) NL8701226A (ko)
NZ (1) NZ220345A (ko)
PT (1) PT84938B (ko)
SE (1) SE465163B (ko)
ZA (1) ZA873583B (ko)

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US5187188A (en) * 1992-04-03 1993-02-16 Bristol-Myers Squibb Company Oxazole carboxylic acid derivatives
US5158958A (en) * 1992-04-03 1992-10-27 Bristol-Myers Squibb Company Imidazo[4,5-b]quinolinyl oxy alkyl sulfonyl piperidine derivatives
US5552267A (en) * 1992-04-03 1996-09-03 The Trustees Of Columbia University In The City Of New York Solution for prolonged organ preservation
US5196428A (en) * 1992-04-03 1993-03-23 Bristol-Myers Squibb Company Imidazo[4,5-b]qinolinyl oxy alkyl ureas
US5348960A (en) * 1992-04-03 1994-09-20 Bristol-Myers Squibb Company Imidazo[4,5-b]quinolinyl oxy alkyl tetrazolyl piperidine derivatives
US5208237A (en) * 1992-04-03 1993-05-04 Bristol-Meyers Squibb Company 7-oxypropylsulfonamido-imidazo[4,5-b]quinolin-2-ones
TW593317B (en) 1993-06-21 2004-06-21 Janssen Pharmaceutica Nv Positive cardiac inotropic and lusitropic pyrroloquinolinone derivatives
US6331539B1 (en) 1999-06-10 2001-12-18 3M Innovative Properties Company Sulfonamide and sulfamide substituted imidazoquinolines
US6573273B1 (en) 1999-06-10 2003-06-03 3M Innovative Properties Company Urea substituted imidazoquinolines
US6756382B2 (en) 1999-06-10 2004-06-29 3M Innovative Properties Company Amide substituted imidazoquinolines
US6541485B1 (en) 1999-06-10 2003-04-01 3M Innovative Properties Company Urea substituted imidazoquinolines
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JP2006509790A (ja) * 2002-11-27 2006-03-23 アルテシアン セラピューティック，インコーポレイティド 心不全の治療のための混合されたＰＤＥ阻害およびβアドレナリン拮抗薬活性または部分的作用薬活性を有する化合物
JP2007502293A (ja) 2003-08-12 2007-02-08 スリーエム イノベイティブ プロパティズ カンパニー ヒドロキシルアミン置換イミダゾ含有化合物
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US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
AR046046A1 (es) 2003-10-03 2005-11-23 3M Innovative Properties Co Imidazoquinolinas alcoxi sustituidas. composiciones farmaceuticas.
CA2545774A1 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Oxime substituted imidazo ring compounds
CA2545825A1 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Hydroxylamine substituted imidazo ring compounds
BRPI0416936A (pt) 2003-11-25 2007-01-16 3M Innovative Properties Co sistemas de anel de imidazo substituìdos e métodos
EP1701955A1 (en) 2003-12-29 2006-09-20 3M Innovative Properties Company Arylalkenyl and arylalkynyl substituted imidazoquinolines
EP1699788A2 (en) 2003-12-30 2006-09-13 3M Innovative Properties Company Imidazoquinolinyl, imidazopyridinyl and imidazonaphthyridinyl sulfonamides
AU2005228150A1 (en) 2004-03-24 2005-10-13 3M Innovative Properties Company Amide substituted imidazopyridines, imidazoquinolines, and imidazonaphthyridines
WO2005123080A2 (en) 2004-06-15 2005-12-29 3M Innovative Properties Company Nitrogen-containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
WO2006065280A2 (en) 2004-06-18 2006-06-22 3M Innovative Properties Company Isoxazole, dihydroisoxazole, and oxadiazole substituted imidazo ring compounds and methods
WO2006038923A2 (en) 2004-06-18 2006-04-13 3M Innovative Properties Company Aryl substituted imidazonaphthyridines
WO2006009826A1 (en) 2004-06-18 2006-01-26 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted thiazoloquinolines and thiazolonaphthyridines
US8034938B2 (en) 2004-12-30 2011-10-11 3M Innovative Properties Company Substituted chiral fused [1,2]imidazo[4,5-c] ring compounds
JP5543068B2 (ja) 2004-12-30 2014-07-09 スリーエム イノベイティブ プロパティズ カンパニー キラル縮合［１，２］イミダゾ［４，５−ｃ］環状化合物
US9248127B2 (en) 2005-02-04 2016-02-02 3M Innovative Properties Company Aqueous gel formulations containing immune response modifiers
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US7943610B2 (en) 2005-04-01 2011-05-17 3M Innovative Properties Company Pyrazolopyridine-1,4-diamines and analogs thereof
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WO2013106547A1 (en) 2012-01-10 2013-07-18 President And Fellows Of Harvard College Beta-cell replication promoting compounds and methods of their use

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US3932407A (en) * 1973-11-19 1976-01-13 Bristol-Myers Company Optionally substituted 1,2,3,5-tetrahydroimidezo(2,1-b)-quinazolin-2-ones and 6(H)-1,2,3,4-tetrahydropyimido(2,1-b)quinazolin-2-ones
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Also Published As

Publication number Publication date
GB8711839D0 (en) 1987-06-24
FI86723C (fi) 1992-10-12
AT392790B (de) 1991-06-10
SE465163B (sv) 1991-08-05
KR870011137A (ko) 1987-12-21
DE3717291A1 (de) 1987-11-26
HUT43602A (en) 1987-11-30
FR2603586B1 (fr) 1990-12-28
FI86723B (fi) 1992-06-30
BE1002033A4 (fr) 1990-05-29
HU197570B (en) 1989-04-28
GB2190676B (en) 1990-05-30
AU603577B2 (en) 1990-11-22
GR870803B (en) 1987-09-24
DK263587A (da) 1987-11-24
DK166084C (da) 1993-08-02
JPS62283972A (ja) 1987-12-09
KR900008567B1 (ko) 1990-11-24
NZ220345A (en) 1990-10-26
DK166084B (da) 1993-03-08
CH675246A5 (ko) 1990-09-14
AU7299387A (en) 1987-11-26
ES2005588A6 (es) 1989-03-16
GB2190676A (en) 1987-11-25
FR2603586A1 (fr) 1988-03-11
US4775674A (en) 1988-10-04
ZA873583B (en) 1988-04-27
IT1205031B (it) 1989-03-10
PT84938A (en) 1987-06-01
FI872220A0 (fi) 1987-05-20
FI872220A (fi) 1987-11-24
IL82612A0 (en) 1987-11-30
PT84938B (pt) 1990-02-08
SE8702158D0 (sv) 1987-05-22
CA1289137C (en) 1991-09-17
LU86896A1 (fr) 1988-01-20
ATA132087A (de) 1990-11-15
IT8720650A0 (it) 1987-05-22
SE8702158L (sv) 1987-11-24
DK263587D0 (da) 1987-05-22

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