MX9202449A - 3-aminoquinuclidinas substituidas. - Google Patents

3-aminoquinuclidinas substituidas.

Info

Publication number
MX9202449A
MX9202449A MX9202449A MX9202449A MX9202449A MX 9202449 A MX9202449 A MX 9202449A MX 9202449 A MX9202449 A MX 9202449A MX 9202449 A MX9202449 A MX 9202449A MX 9202449 A MX9202449 A MX 9202449A
Authority
MX
Mexico
Prior art keywords
aminoquinuclidines
substituted
compounds
disorders
antagonists
Prior art date
Application number
MX9202449A
Other languages
English (en)
Inventor
Fumitaka Ito
Thoshihde Kokura
Masami Nakane
Kunio Satake
Hiroaki Wakabayashi
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9202449A publication Critical patent/MX9202449A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Medicinal Preparation (AREA)
MX9202449A 1991-05-22 1992-05-22 3-aminoquinuclidinas substituidas. MX9202449A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP14682691 1991-05-22

Publications (1)

Publication Number Publication Date
MX9202449A true MX9202449A (es) 1993-03-01

Family

ID=15416402

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9202449A MX9202449A (es) 1991-05-22 1992-05-22 3-aminoquinuclidinas substituidas.

Country Status (25)

Country Link
EP (1) EP0585328B1 (es)
KR (1) KR100246065B1 (es)
CN (1) CN1041827C (es)
AT (1) ATE211743T1 (es)
AU (1) AU658898B2 (es)
BR (1) BR9206044A (es)
CA (1) CA2109415C (es)
CZ (1) CZ247993A3 (es)
DE (2) DE9290057U1 (es)
DK (1) DK0585328T3 (es)
EG (1) EG20218A (es)
ES (1) ES2168260T3 (es)
FI (1) FI935134A (es)
HU (1) HUT65771A (es)
IE (1) IE921662A1 (es)
IL (1) IL101960A (es)
MX (1) MX9202449A (es)
NO (1) NO305173B1 (es)
NZ (2) NZ272941A (es)
PL (4) PL171921B1 (es)
PT (1) PT100514B (es)
RU (1) RU2092486C1 (es)
UA (1) UA26401C2 (es)
WO (1) WO1992020676A1 (es)
ZA (1) ZA923773B (es)

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US5837711A (en) * 1992-10-28 1998-11-17 Pfizer Inc. Substituted quinuclidines as substance P antagonists
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EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
PE8798A1 (es) * 1995-07-17 1998-03-02 Pfizer Procedimiento de separacion de los enantiomeros del 1-azabiciclo[2.2.2] octan-3-amina, 2-(difenilmetil) -n- [[2-metoxi-5-(1-metiletil) fenil] metil]
TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
MX9706944A (es) * 1996-09-12 1998-08-30 Pfizer Quinuclidinas sustituidas con tetrazolilo como antagonistas de la sustancia p.
NZ329807A (en) * 1997-04-23 2000-07-28 Pfizer NK-1 receptor antagonists and P receptor antagonists 2-Diarylmethyl-3-amino-1-azabicyclo[2.2.2]octane derivatives and amino substituted N-containing rings as agents for treating irritable bowel syndrome
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US6861526B2 (en) 2002-10-16 2005-03-01 Pfizer Inc. Process for the preparation of (S,S)-cis-2-benzhydryl-3-benzylaminoquinuclidine
MX2007000428A (es) 2004-07-15 2008-03-05 Amr Technology Inc Tetrahidroisoquinolinas sustituidas con arilo y heteroarilo y uso de las mismas para bloquear la captacion de norepinefrina, dopamina y serotonina.
ES2382814T3 (es) 2005-05-17 2012-06-13 Merck Sharp & Dohme Ltd. Ácido cis-4-[(4-clorofenil)sulfonil]-4-(2,5-difluorofenil)ciclohexanopropanoico para el tratamiento del cáncer
MX2008000717A (es) 2005-07-15 2008-03-18 Amr Technology Inc Tetrahidrobenzazepinas substituidas con arilo y heteroarilo y uso de las mismas para bloquear la reabsorcion de norepinefrina, dopamina, y serotonina.
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EA200970706A1 (ru) 2007-01-24 2010-02-26 Глэксо Груп Лимитед Новые фармацевтические композиции
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UA105182C2 (ru) 2008-07-03 2014-04-25 Ньюрексон, Інк. Бензоксазины, бензотиазины и родственные соединения, которые имеют ингибирующую nos активность
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US9034899B2 (en) 2009-05-12 2015-05-19 Albany Molecular Research, Inc. Aryl, heteroaryl, and heterocycle substituted tetrahydroisoquinolines and use thereof
CN102638982B (zh) 2009-05-12 2015-07-08 百时美施贵宝公司 (S)-7-([1,2,4]三唑并[1,5-a]吡啶-6-基)-4-(3,4-二氯苯基)-1,2,3,4-四氢异喹啉的晶型及其用途
DK2429296T3 (en) 2009-05-12 2018-03-12 Albany Molecular Res Inc 7 - ([1,2,4,] TRIAZOLO [1,5, -A] PYRIDIN-6-YL) -4- (3,4-DICHLORPHENYL) -1,2,3,4- TETRAHYDROISOQUINOLINE AND USE thereof
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Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX18467A (es) * 1988-11-23 1993-07-01 Pfizer Agentes terapeuticos de quinuclidinas

Also Published As

Publication number Publication date
DE9290057U1 (de) 1994-01-05
EP0585328B1 (en) 2002-01-09
FI935134A0 (fi) 1993-11-19
PL170525B1 (en) 1996-12-31
IE921662A1 (en) 1992-12-02
ATE211743T1 (de) 2002-01-15
CA2109415C (en) 1998-12-29
NO305173B1 (no) 1999-04-12
ZA923773B (en) 1993-11-22
UA26401C2 (uk) 1999-08-30
ES2168260T3 (es) 2002-06-16
DE69232334D1 (de) 2002-02-14
PL172069B1 (pl) 1997-07-31
WO1992020676A1 (en) 1992-11-26
DE69232334T2 (de) 2002-11-14
NO934195D0 (no) 1993-11-19
CN1068571A (zh) 1993-02-03
IL101960A0 (en) 1994-04-12
CA2109415A1 (en) 1992-11-23
IL101960A (en) 1999-03-12
HUT65771A (en) 1994-07-28
PT100514A (pt) 1993-09-30
AU658898B2 (en) 1995-05-04
NO934195L (no) 1993-11-19
DK0585328T3 (da) 2002-02-11
KR100246065B1 (en) 2000-04-01
HU9303307D0 (en) 1994-03-28
NZ242880A (en) 1995-10-26
BR9206044A (pt) 1995-03-01
NZ272941A (en) 1997-05-26
CZ247993A3 (en) 1994-07-13
EG20218A (en) 1997-11-30
FI935134A (fi) 1993-11-19
PL171921B1 (pl) 1997-06-30
EP0585328A1 (en) 1994-03-09
AU1927592A (en) 1992-12-30
PL170513B1 (en) 1996-12-31
RU2092486C1 (ru) 1997-10-10
CN1041827C (zh) 1999-01-27
PT100514B (pt) 1999-06-30

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Legal Events

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FG Grant or registration
MM Annulment or lapse due to non-payment of fees