FI935134A0 - Substituerade 3-aminokinuklidiner - Google Patents

Substituerade 3-aminokinuklidiner

Info

Publication number
FI935134A0
FI935134A0 FI935134A FI935134A FI935134A0 FI 935134 A0 FI935134 A0 FI 935134A0 FI 935134 A FI935134 A FI 935134A FI 935134 A FI935134 A FI 935134A FI 935134 A0 FI935134 A0 FI 935134A0
Authority
FI
Finland
Prior art keywords
compounds
aminoquinuclidine
substituent
disorders
antagonists
Prior art date
Application number
FI935134A
Other languages
English (en)
Other versions
FI935134A (fi
Inventor
Fumitaka Ito
Toshihide Kokura
Masami Nakane
Kunio Satake
Hiroaki Wakabayashi
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI935134A publication Critical patent/FI935134A/fi
Publication of FI935134A0 publication Critical patent/FI935134A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Medicinal Preparation (AREA)
FI935134A 1991-05-22 1993-11-19 Substituerade 3-aminokinuklidiner FI935134A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP14682691 1991-05-22
PCT/US1992/004002 WO1992020676A1 (en) 1991-05-22 1992-05-19 Substituted 3-aminoquinuclidines

Publications (2)

Publication Number Publication Date
FI935134A FI935134A (fi) 1993-11-19
FI935134A0 true FI935134A0 (fi) 1993-11-19

Family

ID=15416402

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935134A FI935134A0 (fi) 1991-05-22 1993-11-19 Substituerade 3-aminokinuklidiner

Country Status (25)

Country Link
EP (1) EP0585328B1 (fi)
KR (1) KR100246065B1 (fi)
CN (1) CN1041827C (fi)
AT (1) ATE211743T1 (fi)
AU (1) AU658898B2 (fi)
BR (1) BR9206044A (fi)
CA (1) CA2109415C (fi)
CZ (1) CZ247993A3 (fi)
DE (2) DE69232334T2 (fi)
DK (1) DK0585328T3 (fi)
EG (1) EG20218A (fi)
ES (1) ES2168260T3 (fi)
FI (1) FI935134A0 (fi)
HU (1) HUT65771A (fi)
IE (1) IE921662A1 (fi)
IL (1) IL101960A (fi)
MX (1) MX9202449A (fi)
NO (1) NO305173B1 (fi)
NZ (2) NZ242880A (fi)
PL (4) PL171921B1 (fi)
PT (1) PT100514B (fi)
RU (1) RU2092486C1 (fi)
UA (1) UA26401C2 (fi)
WO (1) WO1992020676A1 (fi)
ZA (1) ZA923773B (fi)

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JP2656699B2 (ja) * 1992-10-21 1997-09-24 ファイザー製薬株式会社 置換ベンジルアミノキヌクリジン
JP2656700B2 (ja) * 1992-10-28 1997-09-24 ファイザー製薬株式会社 置換キヌクリジン誘導体
US5837711A (en) * 1992-10-28 1998-11-17 Pfizer Inc. Substituted quinuclidines as substance P antagonists
WO1994013663A1 (en) * 1992-12-10 1994-06-23 Pfizer Inc. Aminomethylene substituted non-aromatic heterocycles and use as substance p antagonists
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US6083943A (en) * 1993-09-17 2000-07-04 Pfizer Inc Substituted azaheterocyclecarboxylic acid
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EP0653208A3 (en) * 1993-11-17 1995-10-11 Pfizer Substance P antagonists for the treatment or prevention of sunburn.
EP0659409A3 (en) * 1993-11-23 1995-08-09 Pfizer Substance P antagonists for the inhibition of angiogenesis.
EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
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TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
MX9706944A (es) * 1996-09-12 1998-08-30 Pfizer Quinuclidinas sustituidas con tetrazolilo como antagonistas de la sustancia p.
NZ329807A (en) * 1997-04-23 2000-07-28 Pfizer NK-1 receptor antagonists and P receptor antagonists 2-Diarylmethyl-3-amino-1-azabicyclo[2.2.2]octane derivatives and amino substituted N-containing rings as agents for treating irritable bowel syndrome
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WO2006123182A2 (en) 2005-05-17 2006-11-23 Merck Sharp & Dohme Limited Cyclohexyl sulphones for treatment of cancer
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US20110218176A1 (en) 2006-11-01 2011-09-08 Barbara Brooke Jennings-Spring Compounds, methods, and treatments for abnormal signaling pathways for prenatal and postnatal development
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Also Published As

Publication number Publication date
NO934195L (no) 1993-11-19
PL170513B1 (en) 1996-12-31
EG20218A (en) 1997-11-30
PL172069B1 (pl) 1997-07-31
DE69232334T2 (de) 2002-11-14
AU1927592A (en) 1992-12-30
CN1041827C (zh) 1999-01-27
EP0585328A1 (en) 1994-03-09
IL101960A0 (en) 1994-04-12
PT100514A (pt) 1993-09-30
NO934195D0 (no) 1993-11-19
PT100514B (pt) 1999-06-30
ATE211743T1 (de) 2002-01-15
IL101960A (en) 1999-03-12
MX9202449A (es) 1993-03-01
PL171921B1 (pl) 1997-06-30
FI935134A (fi) 1993-11-19
UA26401C2 (uk) 1999-08-30
CN1068571A (zh) 1993-02-03
CZ247993A3 (en) 1994-07-13
NO305173B1 (no) 1999-04-12
RU2092486C1 (ru) 1997-10-10
CA2109415C (en) 1998-12-29
KR100246065B1 (en) 2000-04-01
CA2109415A1 (en) 1992-11-23
BR9206044A (pt) 1995-03-01
ES2168260T3 (es) 2002-06-16
WO1992020676A1 (en) 1992-11-26
PL170525B1 (en) 1996-12-31
DK0585328T3 (da) 2002-02-11
DE69232334D1 (de) 2002-02-14
AU658898B2 (en) 1995-05-04
HU9303307D0 (en) 1994-03-28
ZA923773B (en) 1993-11-22
DE9290057U1 (de) 1994-01-05
IE921662A1 (en) 1992-12-02
HUT65771A (en) 1994-07-28
NZ272941A (en) 1997-05-26
EP0585328B1 (en) 2002-01-09
NZ242880A (en) 1995-10-26

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