MX2008016512A - Epoxicetonas peptidicas para la inhibicion del proteasoma. - Google Patents
Epoxicetonas peptidicas para la inhibicion del proteasoma.Info
- Publication number
- MX2008016512A MX2008016512A MX2008016512A MX2008016512A MX2008016512A MX 2008016512 A MX2008016512 A MX 2008016512A MX 2008016512 A MX2008016512 A MX 2008016512A MX 2008016512 A MX2008016512 A MX 2008016512A MX 2008016512 A MX2008016512 A MX 2008016512A
- Authority
- MX
- Mexico
- Prior art keywords
- carbon atoms
- alkyl
- compound
- milliliters
- hydrogen
- Prior art date
Links
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- 230000005764 inhibitory process Effects 0.000 title description 18
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US81521806P | 2006-06-19 | 2006-06-19 | |
| PCT/US2007/014427 WO2007149512A2 (en) | 2006-06-19 | 2007-06-19 | Peptide epoxyketones for pr0teas0me inhibition |
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2008
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2010
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2011
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2012
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2013
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