CY1114518T1 - Πεπτιδο εποξυκετονες για αναστολη πρωτεασωματος - Google Patents
Πεπτιδο εποξυκετονες για αναστολη πρωτεασωματοςInfo
- Publication number
- CY1114518T1 CY1114518T1 CY20131100490T CY131100490T CY1114518T1 CY 1114518 T1 CY1114518 T1 CY 1114518T1 CY 20131100490 T CY20131100490 T CY 20131100490T CY 131100490 T CY131100490 T CY 131100490T CY 1114518 T1 CY1114518 T1 CY 1114518T1
- Authority
- CY
- Cyprus
- Prior art keywords
- prototasm
- peptido
- extractors
- destruction
- relates
- Prior art date
Links
- 230000006378 damage Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000004245 Proteasome Endopeptidase Complex Human genes 0.000 abstract 1
- 108090000708 Proteasome Endopeptidase Complex Proteins 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000037011 constitutive activity Effects 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000001506 immunosuppresive effect Effects 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/336—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having three-membered rings, e.g. oxirane, fumagillin
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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Applications Claiming Priority (2)
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|---|---|---|---|
| US81521806P | 2006-06-19 | 2006-06-19 | |
| EP07809745.8A EP2041158B1 (en) | 2006-06-19 | 2007-06-19 | Peptide epoxyketones for proteasome inhibition |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1114518T1 true CY1114518T1 (el) | 2016-10-05 |
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| CY20131100490T CY1114518T1 (el) | 2006-06-19 | 2013-06-18 | Πεπτιδο εποξυκετονες για αναστολη πρωτεασωματος |
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| JP6970085B2 (ja) | 2015-10-15 | 2021-11-24 | コーネル・ユニバーシティーCornell University | プロテアソーム阻害剤およびその用途 |
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- 2007-06-19 DK DK07809745.8T patent/DK2041158T3/da active
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2008
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2010
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2012
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