MX2007006103A - Pirrolopirazinas y pirazolopirazinas de utilidad como inhibidores de proteinquinasas. - Google Patents
Pirrolopirazinas y pirazolopirazinas de utilidad como inhibidores de proteinquinasas.Info
- Publication number
- MX2007006103A MX2007006103A MX2007006103A MX2007006103A MX2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A
- Authority
- MX
- Mexico
- Prior art keywords
- optionally substituted
- compound according
- aliphatic
- independently
- membered
- Prior art date
Links
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63011504P | 2004-11-22 | 2004-11-22 | |
| PCT/US2005/042455 WO2006058074A1 (en) | 2004-11-22 | 2005-11-22 | Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007006103A true MX2007006103A (es) | 2007-07-20 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007006103A MX2007006103A (es) | 2004-11-22 | 2005-11-22 | Pirrolopirazinas y pirazolopirazinas de utilidad como inhibidores de proteinquinasas. |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US7795259B2 (https=) |
| EP (3) | EP1814883A1 (https=) |
| JP (3) | JP2008520745A (https=) |
| KR (1) | KR20070089201A (https=) |
| CN (1) | CN101098872B (https=) |
| AU (2) | AU2005309616A1 (https=) |
| CA (2) | CA2587926A1 (https=) |
| IL (1) | IL183318A0 (https=) |
| MX (1) | MX2007006103A (https=) |
| NO (1) | NO20073140L (https=) |
| NZ (1) | NZ555566A (https=) |
| RU (1) | RU2394825C2 (https=) |
| WO (2) | WO2006058074A1 (https=) |
| ZA (1) | ZA200704888B (https=) |
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| HN2005000795A (es) * | 2004-10-15 | 2010-08-19 | Aventis Pharma Inc | Pirimidinas como antagonistas del receptor de prostaglandina d2 |
| WO2006127587A1 (en) * | 2005-05-20 | 2006-11-30 | Vertex Pharmaceuticals Incorporated | Pyrrolopyridines useful as inhibitors of protein kinase |
| US8211919B2 (en) | 2005-09-02 | 2012-07-03 | Astellas Pharma Inc. | Amide derivatives as rock inhibitors |
| US8119655B2 (en) | 2005-10-07 | 2012-02-21 | Takeda Pharmaceutical Company Limited | Kinase inhibitors |
| WO2007076423A2 (en) * | 2005-12-22 | 2007-07-05 | Smithkline Beecham Corporation | INHIBITORS OF Akt ACTIVITY |
| CN102532133A (zh) | 2006-01-17 | 2012-07-04 | 沃泰克斯药物股份有限公司 | 适用作詹纳斯激酶抑制剂的吖吲哚类 |
| EP2044061A2 (en) * | 2006-07-20 | 2009-04-08 | Mehmet Kahraman | Benzothiophene inhibitors of rho kinase |
| CL2007002617A1 (es) * | 2006-09-11 | 2008-05-16 | Sanofi Aventis | Compuestos derivados de pirrolo[2,3-b]pirazin-6-ilo; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar inflamacion de las articulaciones, artritis reumatoide, tumores, linfoma de las celulas del manto. |
| SG158147A1 (en) | 2006-10-09 | 2010-01-29 | Takeda Pharmaceutical | Kinase inhibitors |
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| WO2022261159A1 (en) | 2021-06-09 | 2022-12-15 | Incyte Corporation | Tricyclic heterocycles as fgfr inhibitors |
| EP4352059A1 (en) | 2021-06-09 | 2024-04-17 | Incyte Corporation | Tricyclic heterocycles as fgfr inhibitors |
| IL310717A (en) | 2021-08-20 | 2024-04-01 | Biomea Fusion Inc | Crystalline form of N-[4-[4-(4-morpholinyl)-7H-PYRROLO[2,3-D]PYRIMIDIN-6-YL]PHENYL]-4-[[3(R)-[(1-OXO ] -2-PROPEN-1-YL)AMINO]-1-PIPERIDINYL]METHYL]-2-PYRIDINECARBOXAMIDE, IRREVERSIBLE MENIN-MLL INHIBITOR FOR CANCER TREATMENT |
| WO2024155710A1 (en) | 2023-01-18 | 2024-07-25 | Biomea Fusion, Inc. | Crystalline forms of n-[4-[4-(4-morpholinyl)-7h-pyrrolo[2,3-d]pyrimidin-6- yl]phenyl]-4-[[3(r)-[(l-oxo-2-propen-l-yl)amino]-l-piperidinyl]methyl]-2-pyridinecarboxamide as a covalent inhibitor of menin-mll interaction |
| WO2025224050A1 (en) | 2024-04-22 | 2025-10-30 | Institut National de la Santé et de la Recherche Médicale | Methods of treatment of patients suffering from hypomelanosis of ito |
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| MC2096A1 (fr) * | 1989-02-23 | 1991-02-15 | Hoffmann La Roche | Pyrroles substitues |
| JP2648372B2 (ja) * | 1989-09-18 | 1997-08-27 | キヤノン株式会社 | インクジェット記録装置 |
| HUP0202332A2 (en) * | 2000-02-05 | 2002-10-28 | Vertex Pharma | Pyrazole compositions useful as inhibitors of erk |
| MY130778A (en) * | 2001-02-09 | 2007-07-31 | Vertex Pharma | Heterocyclic inhibitiors of erk2 and uses thereof |
| GB0115109D0 (en) * | 2001-06-21 | 2001-08-15 | Aventis Pharma Ltd | Chemical compounds |
| EP1401762A1 (de) | 2001-06-22 | 2004-03-31 | Basf Aktiengesellschaft | Stäbchenförmige apatitkristalle mit einem bestimmten länge-zu-breite-verhältnis |
| US7101884B2 (en) * | 2001-09-14 | 2006-09-05 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| GB0206860D0 (en) * | 2002-03-22 | 2002-05-01 | Glaxo Group Ltd | Compounds |
| EP1545515A1 (en) * | 2002-08-12 | 2005-06-29 | Sugen, Inc. | 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors |
| JP2006507299A (ja) * | 2002-10-30 | 2006-03-02 | メルク エンド カムパニー インコーポレーテッド | Ａｋｔ活性の阻害薬 |
| EP1558607B1 (en) * | 2002-10-30 | 2010-05-05 | Vertex Pharmaceuticals Incorporated | Compositions useful as inhibitors of rock and other protein kinases |
| AR045595A1 (es) * | 2003-09-04 | 2005-11-02 | Vertex Pharma | Composiciones utiles como inhibidores de proteinas quinasas |
| AU2005219517A1 (en) * | 2004-02-27 | 2005-09-15 | F.Hoffmann-La Roche Ag | Heteroaryl-fused pyrazolo derivatives |
| KR100843526B1 (ko) | 2004-02-27 | 2008-07-03 | 에프. 호프만-라 로슈 아게 | 피라졸의 접합 유도체 |
| US7763843B2 (en) | 2004-03-01 | 2010-07-27 | Stanton Magnetics, Inc. | Optical navigation system for rotary control based non-contact controller |
| KR20070002081A (ko) * | 2004-04-02 | 2007-01-04 | 버텍스 파마슈티칼스 인코포레이티드 | Ｒｏｃｋ 및 기타 단백질 키나아제의 억제제로서 유용한아자인돌 |
| MX2007001126A (es) * | 2004-07-27 | 2007-09-25 | Sgx Pharmaceuticals Inc | Moduladores de heterociclo cinasa de anillo fusionado. |
| CN101389626A (zh) * | 2004-07-27 | 2009-03-18 | Sgx药物公司 | 稠环杂环激酶调节剂 |
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2005
- 2005-11-22 EP EP05825542A patent/EP1814883A1/en not_active Withdrawn
- 2005-11-22 RU RU2007123360/04A patent/RU2394825C2/ru not_active IP Right Cessation
- 2005-11-22 KR KR1020077014367A patent/KR20070089201A/ko not_active Withdrawn
- 2005-11-22 EP EP05825395A patent/EP1814882A1/en not_active Withdrawn
- 2005-11-22 US US11/285,497 patent/US7795259B2/en not_active Expired - Fee Related
- 2005-11-22 CN CN2005800460428A patent/CN101098872B/zh not_active Expired - Fee Related
- 2005-11-22 WO PCT/US2005/042455 patent/WO2006058074A1/en not_active Ceased
- 2005-11-22 US US11/285,516 patent/US20060122185A1/en not_active Abandoned
- 2005-11-22 WO PCT/US2005/042537 patent/WO2006058120A1/en not_active Ceased
- 2005-11-22 AU AU2005309616A patent/AU2005309616A1/en not_active Abandoned
- 2005-11-22 EP EP10185488A patent/EP2316835A1/en not_active Withdrawn
- 2005-11-22 CA CA002587926A patent/CA2587926A1/en not_active Abandoned
- 2005-11-22 AU AU2005309566A patent/AU2005309566A1/en not_active Abandoned
- 2005-11-22 MX MX2007006103A patent/MX2007006103A/es active IP Right Grant
- 2005-11-22 NZ NZ555566A patent/NZ555566A/en not_active IP Right Cessation
- 2005-11-22 CA CA002587894A patent/CA2587894A1/en not_active Abandoned
- 2005-11-22 JP JP2007543468A patent/JP2008520745A/ja active Pending
- 2005-11-22 JP JP2007543441A patent/JP2008520738A/ja active Pending
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2007
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2008
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| US20060122185A1 (en) | 2006-06-08 |
| NZ555566A (en) | 2009-12-24 |
| EP1814882A1 (en) | 2007-08-08 |
| AU2005309566A1 (en) | 2006-06-01 |
| CA2587894A1 (en) | 2006-06-01 |
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| WO2006058074A1 (en) | 2006-06-01 |
| WO2006058120A1 (en) | 2006-06-01 |
| NO20073140L (no) | 2007-06-20 |
| US20060258662A1 (en) | 2006-11-16 |
| AU2005309616A1 (en) | 2006-06-01 |
| KR20070089201A (ko) | 2007-08-30 |
| CA2587926A1 (en) | 2006-06-01 |
| CN101098872B (zh) | 2012-09-05 |
| JP2009024024A (ja) | 2009-02-05 |
| ZA200704888B (en) | 2009-02-25 |
| JP2008520745A (ja) | 2008-06-19 |
| US20110081364A1 (en) | 2011-04-07 |
| RU2394825C2 (ru) | 2010-07-20 |
| CN101098872A (zh) | 2008-01-02 |
| JP2008520738A (ja) | 2008-06-19 |
| EP1814883A1 (en) | 2007-08-08 |
| EP2316835A1 (en) | 2011-05-04 |
| US8372835B2 (en) | 2013-02-12 |
| RU2007123360A (ru) | 2009-01-27 |
| IL183318A0 (en) | 2007-09-20 |
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