RU2394825C2 - Пирролопиразины, пригодные в качестве ингибиторов киназы аврора а - Google Patents
Пирролопиразины, пригодные в качестве ингибиторов киназы аврора а Download PDFInfo
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- RU2394825C2 RU2394825C2 RU2007123360/04A RU2007123360A RU2394825C2 RU 2394825 C2 RU2394825 C2 RU 2394825C2 RU 2007123360/04 A RU2007123360/04 A RU 2007123360/04A RU 2007123360 A RU2007123360 A RU 2007123360A RU 2394825 C2 RU2394825 C2 RU 2394825C2
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| WO2006127587A1 (en) * | 2005-05-20 | 2006-11-30 | Vertex Pharmaceuticals Incorporated | Pyrrolopyridines useful as inhibitors of protein kinase |
| US8211919B2 (en) | 2005-09-02 | 2012-07-03 | Astellas Pharma Inc. | Amide derivatives as rock inhibitors |
| US8119655B2 (en) | 2005-10-07 | 2012-02-21 | Takeda Pharmaceutical Company Limited | Kinase inhibitors |
| WO2007076423A2 (en) * | 2005-12-22 | 2007-07-05 | Smithkline Beecham Corporation | INHIBITORS OF Akt ACTIVITY |
| CN102532133A (zh) | 2006-01-17 | 2012-07-04 | 沃泰克斯药物股份有限公司 | 适用作詹纳斯激酶抑制剂的吖吲哚类 |
| EP2044061A2 (en) * | 2006-07-20 | 2009-04-08 | Mehmet Kahraman | Benzothiophene inhibitors of rho kinase |
| CL2007002617A1 (es) * | 2006-09-11 | 2008-05-16 | Sanofi Aventis | Compuestos derivados de pirrolo[2,3-b]pirazin-6-ilo; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar inflamacion de las articulaciones, artritis reumatoide, tumores, linfoma de las celulas del manto. |
| SG158147A1 (en) | 2006-10-09 | 2010-01-29 | Takeda Pharmaceutical | Kinase inhibitors |
| AU2007338754A1 (en) | 2006-12-21 | 2008-07-03 | Vertex Pharmaceuticals Incorporated | 5-cyan0-4- (pyrrolo [2, 3B] pyridine-3-yl) -pyrimidine derivatives useful as protein kinase inhibitors |
| DK2124944T3 (da) | 2007-03-14 | 2012-04-23 | Ranbaxy Lab Ltd | Pyrazolo[3,4-b]pyridinderivater som phosphodiesteraseinhibitorer |
| CN101778825A (zh) * | 2007-03-22 | 2010-07-14 | 沃泰克斯药物股份有限公司 | 适用作詹纳斯激酶抑制剂的n-杂环类化合物 |
| JP5368485B2 (ja) * | 2008-02-25 | 2013-12-18 | エフ．ホフマン−ラ ロシュ アーゲー | ピロロピラジンキナーゼインヒビター |
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| WO2024155710A1 (en) | 2023-01-18 | 2024-07-25 | Biomea Fusion, Inc. | Crystalline forms of n-[4-[4-(4-morpholinyl)-7h-pyrrolo[2,3-d]pyrimidin-6- yl]phenyl]-4-[[3(r)-[(l-oxo-2-propen-l-yl)amino]-l-piperidinyl]methyl]-2-pyridinecarboxamide as a covalent inhibitor of menin-mll interaction |
| WO2025224050A1 (en) | 2024-04-22 | 2025-10-30 | Institut National de la Santé et de la Recherche Médicale | Methods of treatment of patients suffering from hypomelanosis of ito |
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- 2005-11-22 RU RU2007123360/04A patent/RU2394825C2/ru not_active IP Right Cessation
- 2005-11-22 KR KR1020077014367A patent/KR20070089201A/ko not_active Withdrawn
- 2005-11-22 EP EP05825395A patent/EP1814882A1/en not_active Withdrawn
- 2005-11-22 US US11/285,497 patent/US7795259B2/en not_active Expired - Fee Related
- 2005-11-22 CN CN2005800460428A patent/CN101098872B/zh not_active Expired - Fee Related
- 2005-11-22 WO PCT/US2005/042455 patent/WO2006058074A1/en not_active Ceased
- 2005-11-22 US US11/285,516 patent/US20060122185A1/en not_active Abandoned
- 2005-11-22 WO PCT/US2005/042537 patent/WO2006058120A1/en not_active Ceased
- 2005-11-22 AU AU2005309616A patent/AU2005309616A1/en not_active Abandoned
- 2005-11-22 EP EP10185488A patent/EP2316835A1/en not_active Withdrawn
- 2005-11-22 CA CA002587926A patent/CA2587926A1/en not_active Abandoned
- 2005-11-22 AU AU2005309566A patent/AU2005309566A1/en not_active Abandoned
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- 2005-11-22 JP JP2007543441A patent/JP2008520738A/ja active Pending
- 2005-11-22 ZA ZA200704888A patent/ZA200704888B/xx unknown
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- 2007-06-20 NO NO20073140A patent/NO20073140L/no not_active Application Discontinuation
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2008
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| US20060122185A1 (en) | 2006-06-08 |
| NZ555566A (en) | 2009-12-24 |
| EP1814882A1 (en) | 2007-08-08 |
| AU2005309566A1 (en) | 2006-06-01 |
| CA2587894A1 (en) | 2006-06-01 |
| US7795259B2 (en) | 2010-09-14 |
| WO2006058074A1 (en) | 2006-06-01 |
| WO2006058120A1 (en) | 2006-06-01 |
| NO20073140L (no) | 2007-06-20 |
| US20060258662A1 (en) | 2006-11-16 |
| AU2005309616A1 (en) | 2006-06-01 |
| KR20070089201A (ko) | 2007-08-30 |
| CA2587926A1 (en) | 2006-06-01 |
| MX2007006103A (es) | 2007-07-20 |
| CN101098872B (zh) | 2012-09-05 |
| JP2009024024A (ja) | 2009-02-05 |
| ZA200704888B (en) | 2009-02-25 |
| JP2008520745A (ja) | 2008-06-19 |
| US20110081364A1 (en) | 2011-04-07 |
| CN101098872A (zh) | 2008-01-02 |
| JP2008520738A (ja) | 2008-06-19 |
| EP1814883A1 (en) | 2007-08-08 |
| EP2316835A1 (en) | 2011-05-04 |
| US8372835B2 (en) | 2013-02-12 |
| RU2007123360A (ru) | 2009-01-27 |
| IL183318A0 (en) | 2007-09-20 |
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