MX2007006103A - Pirrolopirazinas y pirazolopirazinas de utilidad como inhibidores de proteinquinasas. - Google Patents
Pirrolopirazinas y pirazolopirazinas de utilidad como inhibidores de proteinquinasas.Info
- Publication number
- MX2007006103A MX2007006103A MX2007006103A MX2007006103A MX2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A MX 2007006103 A MX2007006103 A MX 2007006103A
- Authority
- MX
- Mexico
- Prior art keywords
- optionally substituted
- compound according
- aliphatic
- independently
- membered
- Prior art date
Links
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Classifications
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63011504P | 2004-11-22 | 2004-11-22 | |
| PCT/US2005/042455 WO2006058074A1 (en) | 2004-11-22 | 2005-11-22 | Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007006103A true MX2007006103A (es) | 2007-07-20 |
Family
ID=35953926
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007006103A MX2007006103A (es) | 2004-11-22 | 2005-11-22 | Pirrolopirazinas y pirazolopirazinas de utilidad como inhibidores de proteinquinasas. |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US7795259B2 (enExample) |
| EP (3) | EP1814882A1 (enExample) |
| JP (3) | JP2008520745A (enExample) |
| KR (1) | KR20070089201A (enExample) |
| CN (1) | CN101098872B (enExample) |
| AU (2) | AU2005309616A1 (enExample) |
| CA (2) | CA2587926A1 (enExample) |
| IL (1) | IL183318A0 (enExample) |
| MX (1) | MX2007006103A (enExample) |
| NO (1) | NO20073140L (enExample) |
| NZ (1) | NZ555566A (enExample) |
| RU (1) | RU2394825C2 (enExample) |
| WO (2) | WO2006058074A1 (enExample) |
| ZA (1) | ZA200704888B (enExample) |
Families Citing this family (141)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HN2005000795A (es) * | 2004-10-15 | 2010-08-19 | Aventis Pharma Inc | Pirimidinas como antagonistas del receptor de prostaglandina d2 |
| EP1881983B1 (en) * | 2005-05-20 | 2012-01-11 | Vertex Pharmaceuticals, Inc. | Pyrrolopyridines useful as inhibitors of protein kinase |
| CA2620818A1 (en) | 2005-09-02 | 2007-03-08 | Astellas Pharma Inc. | Amide derivatives as rock inhibitors |
| US8119655B2 (en) | 2005-10-07 | 2012-02-21 | Takeda Pharmaceutical Company Limited | Kinase inhibitors |
| JP2009521504A (ja) * | 2005-12-22 | 2009-06-04 | スミスクライン・ビーチャム・コーポレイション | Ａｋｔ活性阻害剤 |
| NZ601687A (en) | 2006-01-17 | 2014-03-28 | Vertex Pharma | Azaindoles useful as inhibitors of janus kinases |
| US20080021217A1 (en) * | 2006-07-20 | 2008-01-24 | Allen Borchardt | Heterocyclic inhibitors of rho kinase |
| CL2007002617A1 (es) * | 2006-09-11 | 2008-05-16 | Sanofi Aventis | Compuestos derivados de pirrolo[2,3-b]pirazin-6-ilo; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar inflamacion de las articulaciones, artritis reumatoide, tumores, linfoma de las celulas del manto. |
| JP2010505962A (ja) | 2006-10-09 | 2010-02-25 | 武田薬品工業株式会社 | キナーゼ阻害剤 |
| CA2673472A1 (en) * | 2006-12-21 | 2008-07-03 | Vertex Pharmaceuticals Incorporated | 5-cyan0-4- (pyrrolo) [2, 3b] pyridine-3-yl) -pyrimidine derivatives useful as protein kinase inhibitors |
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| CN119816500A (zh) | 2021-08-20 | 2025-04-11 | 拜欧米富士恩公司 | 用于治疗癌症的不可逆menin-MLL抑制剂N-[4-[4-(4-吗啉基)-7H-吡咯并[2,3-d]嘧啶-6-基]苯基]-4-[[3(R)-[(1-氧代-2-丙烯-1-基)氨基]-1-哌啶基]甲基]-2-吡啶甲酰胺的结晶形式 |
| WO2024155719A1 (en) | 2023-01-18 | 2024-07-25 | Biomea Fusion, Inc. | Crystalline forms of n-[4-[4-(4-morpholinyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]-4-[[3(r)-[(l-oxo-2-propen-l-yl)amino]-l-piperidinyl]methyl]-2- pyridinecarboxamide as a covalentinhibitor of menin-mll interaction |
| WO2025224050A1 (en) | 2024-04-22 | 2025-10-30 | Institut National de la Santé et de la Recherche Médicale | Methods of treatment of patients suffering from hypomelanosis of ito |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| MC2096A1 (fr) * | 1989-02-23 | 1991-02-15 | Hoffmann La Roche | Pyrroles substitues |
| JP2648372B2 (ja) * | 1989-09-18 | 1997-08-27 | キヤノン株式会社 | インクジェット記録装置 |
| BR0104424A (pt) * | 2000-02-05 | 2002-01-08 | Vertex Pharma | Composições de pirazol úteis como inibidores de erk |
| MY130778A (en) * | 2001-02-09 | 2007-07-31 | Vertex Pharma | Heterocyclic inhibitiors of erk2 and uses thereof |
| GB0115109D0 (en) * | 2001-06-21 | 2001-08-15 | Aventis Pharma Ltd | Chemical compounds |
| JP2004538228A (ja) | 2001-06-22 | 2004-12-24 | ビーエーエスエフ アクチェンゲゼルシャフト | 特定の長さ幅比を有する棒状アパタイト結晶 |
| US7101884B2 (en) * | 2001-09-14 | 2006-09-05 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| GB0206860D0 (en) * | 2002-03-22 | 2002-05-01 | Glaxo Group Ltd | Compounds |
| CA2495216A1 (en) * | 2002-08-12 | 2004-02-19 | Sugen, Inc. | 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors |
| DE60332475D1 (de) * | 2002-10-30 | 2010-06-17 | Vertex Pharma | Zusammensetzungen verwendbar für die hemmung von rock und anderen kinasen |
| AU2003284981B2 (en) * | 2002-10-30 | 2009-05-28 | Merck Sharp & Dohme Corp. | Inhibitors of Akt activity |
| AR045595A1 (es) | 2003-09-04 | 2005-11-02 | Vertex Pharma | Composiciones utiles como inhibidores de proteinas quinasas |
| KR100843526B1 (ko) * | 2004-02-27 | 2008-07-03 | 에프. 호프만-라 로슈 아게 | 피라졸의 접합 유도체 |
| BRPI0508220A (pt) * | 2004-02-27 | 2007-07-17 | Hoffmann La Roche | derivados de pirazol heteroarila fundidos |
| US7763843B2 (en) | 2004-03-01 | 2010-07-27 | Stanton Magnetics, Inc. | Optical navigation system for rotary control based non-contact controller |
| AR049333A1 (es) * | 2004-04-02 | 2006-07-19 | Vertex Pharma | Azaindoles inhibidores de proteinquinasas rock y otras proteinas quinasas. composiciones farmaceuticas. |
| CN101389626A (zh) * | 2004-07-27 | 2009-03-18 | Sgx药物公司 | 稠环杂环激酶调节剂 |
| AU2005269387A1 (en) * | 2004-07-27 | 2006-02-09 | Sgx Pharmaceuticals, Inc. | Fused ring heterocycle kinase modulators |
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2005
- 2005-11-22 EP EP05825395A patent/EP1814882A1/en not_active Withdrawn
- 2005-11-22 US US11/285,497 patent/US7795259B2/en not_active Expired - Fee Related
- 2005-11-22 CA CA002587926A patent/CA2587926A1/en not_active Abandoned
- 2005-11-22 CA CA002587894A patent/CA2587894A1/en not_active Abandoned
- 2005-11-22 US US11/285,516 patent/US20060122185A1/en not_active Abandoned
- 2005-11-22 EP EP10185488A patent/EP2316835A1/en not_active Withdrawn
- 2005-11-22 NZ NZ555566A patent/NZ555566A/en not_active IP Right Cessation
- 2005-11-22 JP JP2007543468A patent/JP2008520745A/ja active Pending
- 2005-11-22 RU RU2007123360/04A patent/RU2394825C2/ru not_active IP Right Cessation
- 2005-11-22 EP EP05825542A patent/EP1814883A1/en not_active Withdrawn
- 2005-11-22 AU AU2005309616A patent/AU2005309616A1/en not_active Abandoned
- 2005-11-22 MX MX2007006103A patent/MX2007006103A/es active IP Right Grant
- 2005-11-22 WO PCT/US2005/042455 patent/WO2006058074A1/en not_active Ceased
- 2005-11-22 ZA ZA200704888A patent/ZA200704888B/xx unknown
- 2005-11-22 KR KR1020077014367A patent/KR20070089201A/ko not_active Withdrawn
- 2005-11-22 AU AU2005309566A patent/AU2005309566A1/en not_active Abandoned
- 2005-11-22 JP JP2007543441A patent/JP2008520738A/ja active Pending
- 2005-11-22 WO PCT/US2005/042537 patent/WO2006058120A1/en not_active Ceased
- 2005-11-22 CN CN2005800460428A patent/CN101098872B/zh not_active Expired - Fee Related
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2007
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2008
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| AU2005309566A1 (en) | 2006-06-01 |
| US8372835B2 (en) | 2013-02-12 |
| JP2009024024A (ja) | 2009-02-05 |
| US20060122185A1 (en) | 2006-06-08 |
| RU2394825C2 (ru) | 2010-07-20 |
| CN101098872A (zh) | 2008-01-02 |
| IL183318A0 (en) | 2007-09-20 |
| EP1814883A1 (en) | 2007-08-08 |
| US7795259B2 (en) | 2010-09-14 |
| JP2008520738A (ja) | 2008-06-19 |
| ZA200704888B (en) | 2009-02-25 |
| WO2006058120A1 (en) | 2006-06-01 |
| US20060258662A1 (en) | 2006-11-16 |
| WO2006058074A1 (en) | 2006-06-01 |
| NZ555566A (en) | 2009-12-24 |
| NO20073140L (no) | 2007-06-20 |
| JP2008520745A (ja) | 2008-06-19 |
| CN101098872B (zh) | 2012-09-05 |
| KR20070089201A (ko) | 2007-08-30 |
| EP1814882A1 (en) | 2007-08-08 |
| RU2007123360A (ru) | 2009-01-27 |
| US20110081364A1 (en) | 2011-04-07 |
| CA2587926A1 (en) | 2006-06-01 |
| CA2587894A1 (en) | 2006-06-01 |
| EP2316835A1 (en) | 2011-05-04 |
| AU2005309616A1 (en) | 2006-06-01 |
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